SAFit2

Item number	Size	Delivery time	Price
TGM-T16836-1mg	1 mg	7 - 10 business days*	79.00€
TGM-T16836-5mg	5 mg	7 - 10 business days*	195.00€
TGM-T16836-1mL	1 ml	7 - 10 business days*	259.00€
TGM-T16836-10mg	10 mg	7 - 10 business days*	294.00€
TGM-T16836-25mg	25 mg	7 - 10 business days*	501.00€
TGM-T16836-50mg	50 mg	7 - 10 business days*	714.00€
TGM-T16836-100mg	100 mg	7 - 10 business days*	934.00€

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Description: SAFit2 is a highly effective and selective fk506 binding protein 51(FKBP51)... more

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Product information "SAFit2"

Description: SAFit2 is a highly effective and selective fk506 binding protein 51(FKBP51) inhibitor (Ki: 6 nM). SAFit2 can enhance AKT2-AS160 binding and participate in the downstream response of glucocorticoid release in vivo, and is a candidate compound for the treatment of obesity, chronic pain, depression and anxiety. Target: FKBP. Smiles: COc1ccc(CC[C@@H](OC(=O)[C@@H]2CCCCN2C(=O)[C@@H](C2CCCCC2)c2cc(OC)c(OC)c(OC)c2)c2cccc(OCCN3CCOCC3)c2)cc1OC. References: Balsevich G, et al. Stress-responsive FKBP51 regulates AKT2-AS160 signaling and metabolic function. Nat Commun. 2017 Nov 23,8(1):1725.

Supplier:	TargetMol
Supplier-Nr:	T16836

Properties

Application:	FKBP5 inhibitor
MW:	802.99 D
Formula:	C46H62N2O10

Database Information

CAS :	1643125-33-0\| Matching products
KEGG ID :	K09571 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+20°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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