Pyrotinib dimaleate

Item number	Size	Delivery time	Price
TGM-T12594-1mg	1 mg	5 - 10 business days*	148.00€
TGM-T12594-5mg	5 mg	5 - 10 business days*	455.00€
TGM-T12594-10mg	10 mg	5 - 10 business days*	606.00€
TGM-T12594-1mL	1 ml	5 - 10 business days*	616.00€
TGM-T12594-25mg	25 mg	5 - 10 business days*	943.00€
TGM-T12594-50mg	50 mg	5 - 10 business days*	1,298.00€
TGM-T12594-100mg	100 mg	5 - 10 business days*	1,754.00€

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Description: Pyrotinib dimaleate (SHR-1258 dimaleate) is a potent, selective dual inhibitor of... more

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Product information "Pyrotinib dimaleate"

Description: Pyrotinib dimaleate (SHR-1258 dimaleate) is a potent, selective dual inhibitor of EGFR and HER2, with IC50 values of 13 nM and 38 nM, respectively. Target: HER, EGFR. Smiles: OC(=O)\C=C/C(O)=O.OC(=O)\C=C/C(O)=O.CCOc1cc2ncc(C#N)c(Nc3ccc(OCc4ccccn4)c(Cl)c3)c2cc1NC(=O)\C=C\[C@H]1CCCN1C. References: Li X, et al. Discovery and development of Pyrotinib: A novel irreversible EGFR/HER2 dual tyrosine kinase inhibitor with favorable safety profiles for the treatment of breast cancer. Eur J Pharm Sci. 2017 Jan 21. pii: S0928-0987(17)30043-X.

Keywords:	SHR-1258 dimaleate
Supplier:	TargetMol
Supplier-Nr:	T12594

Properties

MW:	815.22 D
Formula:	C40H39ClN6O11

Database Information

CAS :

1397922-61-0| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+20°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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