PROTAC AR-V7 degrader-1

Please request pricing for this article.
Request Pricing

Item number	Size	Datasheet	Manual	SDS	Delivery time	Quantity	Price
TGM-T74410-5mg	5 mg				7 - 10 business days*		-
TGM-T74410-50mg	50 mg				7 - 10 business days*		-

If you have any questions, please use our Contact Form.
You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk

Description: PROTAC AR-V7 degrader-1 (Compound 6) is an orally bioavailable, potent, and... more

Close menu

Product information "PROTAC AR-V7 degrader-1"

Description: PROTAC AR-V7 degrader-1 (Compound 6) is an orally bioavailable, potent, and selective degrader targeting the androgen receptor (AR) variant V7, achieving degradation with a DC50 of 0.32 µM by directing the VHL E3 ligase to the AR DNA-binding domain (DBD). It demonstrates efficacy in the 22Rv1 cell line expressing AR-V7, with an EC50 of 0.88 µM [1]. Target: PROTACs

Supplier:	TargetMol
Supplier-Nr:	T74410

Properties

MW:	789.02 D
Formula:	C41H52N6O6S2

Database Information

CAS :

2767440-24-2| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+20°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

Information about the product reference will follow. more

Close menu

You will get a certificate here

Go back

Read, write and discuss reviews... more

Close menu

Customer review for "PROTAC AR-V7 degrader-1"

Write a review