Ogerin

Item number	Size	Delivery time	Price
TGM-T16378-1mg	1 mg	7 - 10 business days*	30.00€
TGM-T16378-2mg	2 mg	7 - 10 business days*	42.00€
TGM-T16378-5mg	5 mg	7 - 10 business days*	65.00€
TGM-T16378-1mL	1 ml	7 - 10 business days*	74.00€
TGM-T16378-10mg	10 mg	7 - 10 business days*	110.00€
TGM-T16378-25mg	25 mg	7 - 10 business days*	225.00€
TGM-T16378-50mg	50 mg	7 - 10 business days*	378.00€
TGM-T16378-100mg	100 mg	7 - 10 business days*	564.00€

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Description: Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83) that blocks... more

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Product information "Ogerin"

Description: Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83) that blocks recall in fear conditioning in mice. It exhibits inverse agonist and antagonist activity (Ki, 220 nM) at the A2A receptor and weak antagonist activity (Ki, 736 nM) at the 5-HT2B receptor. Target: 5-HT Receptor, Adenosine Receptor, Others. Smiles: Nc1nc(NCc2ccccc2)nc(n1)-c1ccccc1CO. References: Huang XP, et al. Allosteric ligands for the pharmacologically dark receptors GPR68 and GPR65. Nature. 2015 Nov 26,527(7579):477-83.

Supplier:	TargetMol
Supplier-Nr:	T16378

Properties

Application:	GPR68 positive allosteric modulator
MW:	307.35 D
Formula:	C17H17N5O

Database Information

CAS :	1309198-71-7\| Matching products
KEGG ID :	K08408 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+20°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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