GSK778

Item number	Size	Delivery time	Price
TGM-T9703-1mL	1 ml	7 - 10 business days*	38.00€
TGM-T9703-1mg	1 mg	7 - 10 business days*	153.00€
TGM-T9703-5mg	5 mg	7 - 10 business days*	310.00€
TGM-T9703-10mg	10 mg	7 - 10 business days*	500.00€
TGM-T9703-25mg	25 mg	7 - 10 business days*	1,004.00€
TGM-T9703-50mg	50 mg	7 - 10 business days*	1,592.00€
TGM-T9703-100mg	100 mg	7 - 10 business days*	2,209.00€

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Description: GSK778 is a potent and selective inhibitor of BD1 bromodomain such as BRD2 BD1... more

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Product information "GSK778"

Description: GSK778 is a potent and selective inhibitor of BD1 bromodomain such as BRD2 BD1 (IC50s = 75 nM), BRD3 BD1 (IC50s = 41 nM), BRD4 BD1 (IC50s = 41 nM), and BRDT BD1 (IC50s = 143 nM). GSK778 inhibits proliferation, induces a cell cycle arrest and apoptosis. Target: Epigenetic Reader Domain. Smiles: COCc1nc2cnc3cc(-c4c(C)noc4C)c(OC[C@H]4CCNC4)cc3c2n1[C@H](C)c1ccccc1. References: Omer G, et, al. Selective targeting of BD1 and BD2 of the BET proteins in cancer and immunoinflammation. Science. 2020 Apr 24, 368(6489): 387-394.

Supplier:	TargetMol
Supplier-Nr:	T9703

Properties

MW:	511.61 D
Formula:	C30H33N5O3

Database Information

CAS :

2451862-42-1| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+20°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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