GSK270822A

GSK270822A
Item number Size Datasheet Manual SDS Delivery time Quantity Price
Cay43717-1 1 mg -

6 - 10 business days*

147.00€
Cay43717-5 5 mg -

6 - 10 business days*

697.00€
Cay43717-10 10 mg -

6 - 10 business days*

1,322.00€
Cay43717-25 25 mg -

6 - 10 business days*

2,934.00€
 
GSK270822A is an inhibitor of G protein-coupled receptor kinase 2 (GRK2, IC50 = 12. µM). It is... more
Product information "GSK270822A"
GSK270822A is an inhibitor of G protein-coupled receptor kinase 2 (GRK2, IC50 = 12. µM). It is selective for GRK2 over GRK1, GRK5, and PKA (IC50s = 794, 63. and 50. µM, respectively). InChI: InChI=1S/C24H20N4O2/c1-14-23(24(30)27-19-8-9-21-18(11-19)13-25-28-21)20(12-22(29)26-14)17-7-6-15-4-2-3-5-16(15)10-17/h2-11,13,20H,12H2,1H3,(H,25,28)(H,26,29)(H,27,30), InChIKey: ODLNBFNBEPOFNC-UHFFFAOYSA-N, SMILES: O=C(CC1C2=CC3=C(C=CC=C3)C=C2)NC(C)=C1C(NC4=CC5=C(C=C4)NN=C5)=O
Keywords: 1,4,5,6-tetrahydro-N-1H-indazol-5-yl-2-methyl-4-(2-naphthalenyl)-6-oxo-3-pyridinecarboxamide
Supplier: Cayman Chemical
Supplier-Nr: 43717

Properties

Application: GRK2 inhibitor
MW: 396.45 D
Formula: C24H20N4O2
Purity: >98%
Format: Solid

Database Information

CAS : 864082-23-5| Matching products
KEGG ID : K00910 | Matching products

Handling & Safety

Storage: -20°C
Shipping: +20°C (International: -20°C)
Caution
Our products are for laboratory research use only: Not for administration to humans!
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