GNE 2861

Item number	Size	Delivery time	Price
TGM-T16429-1mg	1 mg	7 - 10 business days*	35.00€
TGM-T16429-2mg	2 mg	7 - 10 business days*	48.00€
TGM-T16429-5mg	5 mg	7 - 10 business days*	75.00€
TGM-T16429-1mL	1 ml	7 - 10 business days*	79.00€
TGM-T16429-10mg	10 mg	7 - 10 business days*	125.00€
TGM-T16429-25mg	25 mg	7 - 10 business days*	256.00€
TGM-T16429-50mg	50 mg	7 - 10 business days*	430.00€
TGM-T16429-100mg	100 mg	7 - 10 business days*	635.00€

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Description: GNE 2861 inhibits PAK4, PAK5, and PAK6 (IC50s: 7.5, 36, 126 nM, respectively). GNE... more

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Product information "GNE 2861"

Description: GNE 2861 inhibits PAK4, PAK5, and PAK6 (IC50s: 7.5, 36, 126 nM, respectively). GNE 2861 is a PAK inhibitor that shows group II selectivity. Target: PAK. Smiles: COCCNc1nc2ccc(cc2n1-c1ccnc(N)n1)C#CC1(O)CCCCC1. References: Karpov AS, et al. Optimization of a Dibenzodiazepine Hit to a Potent and Selective Allosteric PAK1 Inhibitor. ACS Med Chem Lett. 2015 May 22,6(7):776-81.

Supplier:	TargetMol
Supplier-Nr:	T16429

Properties

Application:	Group 2 p21-activated kinase (PAK4, PAK5, PAK6) inhibitor
MW:	406.48 D
Formula:	C22H26N6O2

Database Information

CAS :	1394121-05-1\| Matching products
KEGG ID :	K05734 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+20°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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