G-5758

Item number	Size	Datasheet	Manual	SDS	Delivery time	Price
TGM-T87983-25mg	25 mg	-	-	-	7 - 10 business days*	1,668.00€
TGM-T87983-50mg	50 mg	-	-	-	7 - 10 business days*	2,228.00€
TGM-T87983-100mg	100 mg	-	-	-	7 - 10 business days*	2,817.00€

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Description: G-5758 is an orally active IRE1alpha inhibitor with an IC50 of 38 nM for XBP1s. It... more

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Product information "G-5758"

Description: G-5758 is an orally active IRE1alpha inhibitor with an IC50 of 38 nM for XBP1s. It is used in studies involving multiple myeloma models [KMS-11], demonstrating good tolerance in rats at oral doses up to 500 mg/kg. G-5758 exhibits pharmacodynamic effects comparable to those induced by IRE1 knockdown. Target: IRE1, Liposome. Smiles: O(C1=C(C=CC=N1)C2=NC(N[C@H]3C[C@H](F)CNC3)=NC=C2)C4=C(F)C(F)=C(NS(CC5=CC=CC=C5)(=O)=O)C(F)=C4

Supplier:	TargetMol
Supplier-Nr:	T87983

Properties

MW:	588.58 D
Formula:	C27H24F4N6O3S

Database Information

Handling & Safety

Storage:	+4°C
Shipping:	+20°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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