CK2/ERK8-IN-1

Item number	Size	Datasheet	Manual	SDS	Delivery time	Quantity	Price
TGM-T10827-5mg	5 mg				7 - 10 business days*		30.00€
TGM-T10827-10mg	10 mg				7 - 10 business days*		-

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Description: CK2/ERK8-IN-1 (TMCB) is a dual inhibitor of casein kinase 2 (CK2) (Ki: 0.25 µM) and... more

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Product information "CK2/ERK8-IN-1"

Description: CK2/ERK8-IN-1 (TMCB) is a dual inhibitor of casein kinase 2 (CK2) (Ki: 0.25 µM) and ERK8 (IC50s: 0.50 µM) with pro-apoptotic efficacy. CK2/ERK8-IN-1 also binds to PIM1, DYRK1A, and HIPK2 (Kis: 8.65 µM, 11.9 µM, and 15.25 µM). Target: Casein Kinase, DYRK, ERK, Apoptosis, Pim. Smiles: CN(C)c1nc2c(Br)c(Br)c(Br)c(Br)c2n1CC(O)=O. References: Pagano MA, et al. The selectivity of inhibitors of protein kinase CK2: an update. Biochem J. 2008 Nov 1,415(3):353-65.

Keywords:	TMCB
Supplier:	TargetMol
Supplier-Nr:	T10827

Properties

MW:	534.82 D
Formula:	C11H9Br4N3O2

Database Information

CAS :

1085822-09-8| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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