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Mezlocillin Sodium
Item number: TGM-T6582-100mg
Description: Mezlocillin Sodium (Baycipen) is a penicillin beta-lactam antibiotic used in the treatment of bacterial infections caused by susceptible, usually gram-positive, organisms. Target: Antibacterial, Antibiotic. Smiles:...
| Keywords: | Baycipen |
| CAS | 42057-22-7 |
| MW: | 561.56 D |
From 34.00€
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MG 149
Item number: TGM-T6584-100mg
Description: MG 149 (Tip60 HAT inhibitor) is a selective and potent Tip60 inhibitor with IC50 of 74 uM, similar potentcy for MOF(IC50= 47 uM). Target: Histone Acetyltransferase, Others, Epigenetic Reader Domain, Apoptosis. Smiles: CCCCCCCc1ccc(CCc2cccc(O)c2C(O)=O)cc1. References: Ghizzoni M, et al....
| Keywords: | Tip60 HAT inhibitor, MG149 |
| Application: | KAT5 inhibitor |
| CAS | 1243583-85-8 |
| MW: | 340.46 D |
From 46.00€
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SAR405838
Item number: TGM-T6585-100mg
Description: MI-773 (SAR405838 (MI 773)) is an orally available MDM2 antagonist with Ki of 0.88 nM. Phase 1. Target: E1/E2/E3 Enzyme, Mdm2. Smiles: CC(C)(C)C[C@@H]1N[C@H]([C@H](c2cccc(Cl)c2F)[C@]11C(=O)Nc2cc(Cl)ccc12)C(=O)N[C@H]1CC[C@H](O)CC1. References: Wang S, et al. Cancer Res. 2014, 74(20), 5855-5865.
| Keywords: | MI-77301, MI-773, MI773, MI 773 |
| Application: | MDM2-p53 interaction inhibitor |
| CAS | 1303607-60-4 |
| MW: | 562.5 D |
From 43.00€
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Mildronate dihydrate
Item number: TGM-T6586-100mg
Description: Mildronate dihydrate is an inhibitor of biosynthesis of L-carnitine by gamma-butyrobetaine (GBB) hydroxylase and as a competitive inhibitor of renal carnitine reabsorption. Target: Others, Mitochondrial Metabolism. Smiles: O.O.C[N+](C)(C)NCCC([O-])=O. References: Simkhovich BZ, et al. Biochem...
| Keywords: | Meldonium , Mildronate |
| MW: | 182.22 D |
From 29.00€
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Nodinitib-1
Item number: TGM-T6591-100mg
Description: Nodinitib-1 (CID-1088438) is a potent and selective NOD1 inhibitor with an IC50 of 0.56 µM. Target: NOD, NOD-like Receptor (NLR), TNF. Smiles: Cc1ccc(cc1)S(=O)(=O)n1c(N)nc2ccccc12. References: Khan PM et al. ACS Med Chem Lett, 2011, 2(10), 780-785.
| Keywords: | CID-1088438, ML130 |
| Application: | NOD1 inhibitor |
| CAS | 799264-47-4 |
| MW: | 287.34 D |
From 48.00€
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ML133 hydrochloride
Item number: TGM-T6592-100mg
Description: ML133 hydrochloride (ML133 HCl) is a selective potassium channel inhibitor for Kir2.1 with IC50 of 1.8 µM (pH 7.4) and 290 nM (pH 8.5), has no effect on Kir1.1 and weak activity for Kir4.1 and Kir7.1. Target: Potassium Channel. Smiles: Cl.COC1=CC=C(CNCC2=CC=CC3=CC=CC=C23)C=C1. References: Wang HR, et...
| Keywords: | ML133 HCl |
| Application: | Kir2 channel inhibitor |
| CAS | 1222781-70-5 |
| MW: | 313.82 D |
From 41.00€
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Paroxypropione
Item number: TGM-T66154-1mL
Description: It is an inhibitor of the Human Apurinic/apyrimidinic Endonuclease 1 (APE1). Target: Others. Smiles: CCC(=O)c1ccc(O)cc1
| Application: | Antioxidant |
| CAS | 70-70-2 |
| MW: | 150.17 D |
From 29.00€
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Ondansetron hydrochloride
Item number: TGM-T6616-100mg
Description: Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiation therapy. Target: 5-HT Receptor. Smiles: Cl.CN1C2=CC=CC=C2C2=C1CCC(CN1C=CN=C1C)C2=O. References: Pinelli A, et al. Eur J Pharmacol,1997, 340(2-3),...
| Keywords: | SN 307, Ondansetron HCl, Zofran, NSC 665799, Emeset, GR 38032 HCl |
| Application: | Serotonin 5-HT3 receptor antagonist, metabolic studies |
| CAS | 99614-01-4 |
| MW: | 329.82 D |
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Ceftriaxone Sodium
Item number: TGM-T66175-100mg
Description: Ceftriaxone Sodium is a broad-spectrum beta-lactam tertiary cephalosporin antibiotic with anti-inflammatory, antitumor, antibacterial, and antioxidant activities.Ceftriaxone Sodium is a covalent GSK3beta and Aurora B inhibitor used in the study of sepsis and infective endocarditis. Target: GSK-3,...
| CAS | 958633-51-7 |
| MW: | 576.562 D |
From 38.00€
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Desmethyl Erlotinib hydrochloride
Item number: TGM-T6619-100mg
Description: Desmethyl Erlotinib hydrochloride (OSI 420) is an active metabolite of erlotinib which is an orally active EGFR tyrosin kinase inhibitor with IC50 of 2 and 20 nM for human EGFR and EGFR autophosphorylation in tumor cells. Target: EGFR, Drug Metabolite. Smiles:...
| Keywords: | DesMethyl Erlotinib (CP-473420) HCl, OSI420, OSI-420, OSI 420, Desmethyl Erlotinib, CP-473420 |
| CAS | 183320-51-6 |
| MW: | 415.87 D |
From 51.00€
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Oxacillin sodium monohydrate
Item number: TGM-T6622-100mg
Description: Oxacillin sodium monohydrate (Stapenor monohydrate) is an antibacterial agent and is a narrow spectrum beta-lactam antibiotic of the penicillin class. Target: Antibiotic, Antibacterial. Smiles: O.[Na+].[H][C@]12SC(C)(C)[C@@H](N1C(=O)[C@H]2NC(=O)C1=C(C)ON=C1C1=CC=CC=C1)C([O-])=O. References: Ehinger AM,...
| Keywords: | Stapenor monohydrate , Sodium oxacillin monohydrate , Methicillin , Bactocill monohydrate |
| Application: | Antibacterial, Cell wall biosynthesis inhibitor |
| CAS | 7240-38-2 |
| MW: | 441.43 D |
From 30.00€
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Oxibendazole
Item number: TGM-T6623-100mg
Description: Oxibendazole is a benzimidazole drug that interferes with metabolic pathways, used to protect against roundworms, strongyles, threadworms, pinworms and lungworm infestations in horses and some domestic pets. Target: Parasite, Apoptosis. Smiles: N(C(OC)=O)C=1NC=2C(N1)=CC(OCCC)=CC2. References: Lyons ET,...
| Application: | Anthelmintic |
| CAS | 20559-55-1 |
| MW: | 249.27 D |
From 30.00€
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