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CFMTI
Artikelnummer: TGM-T3482-100mg
Description: CFMTI is a potent and selective metabotropic glutamate receptor (mGluR) 1 allosteric antagonist (IC50: 2.6 nM). The selectivity of CFMTI to mGluR1 is higher 2000-fold than mGluR5. Target: GluR. Smiles: Cc1c(nnn1-c1cccnc1F)-c1ccc2C(=O)N(Cc2c1)C1CC1. References: Satow A et al. Unique antipsychotic...
| Anwendung: | mGluR1 allosteric antagonist |
| CAS | 864864-17-5 |
| MW: | 349.36 D |
ab 55,00 €
CFMTI
Artikelnummer: Cay37546-10
CFMTI is a metabotropic glutamate receptor 1 (mGluR1) allosteric antagonist (IC50 = 2.6 nM in CHO cells expressing the human receptor). It is selective for mGluR1 over mGluR5 by greater than 2,000-fold, as well as over mGluR2, -4, -6, -7, or -8 at 10 µM in CHO cells expressing the human receptors. CFTMI reduces...
| Schlagworte: | 2-cyclopropyl-5-[1-(2-fluoro-3-pyridinyl)-5-methyl-1H-1,2,3-triazol-4-yl]-2,3-dihydro-1H-isoindol-1-one |
| Anwendung: | mGluR1 allosteric antagonist |
| CAS | 864864-17-5 |
| MW: | 349.4 D |
ab 138,00 €
