Zu "1884712-47-3" wurden 2 Artikel gefunden!
Für die Filterung wurden keine Ergebnisse gefunden!
CPI-637
Artikelnummer: TGM-T6811-100mg
Description: CPI-637 is a selective and cell-active benzodiazepinone CBP/EP300 bromodomain inhibitor. Target: Histone Acetyltransferase, Epigenetic Reader Domain. Smiles: C[C@@H]1CC(=O)Nc2cccc(-c3ccc4n(C)nc(-c5cnn(C)c5)c4c3)c2N1. References: Taylor AM, et al. ACS Med Chem Lett. 2016, 7(5):531-6.
| Schlagworte: | CPI 637 |
| Anwendung: | CREB-binding protein / Histone acetyltransferase p300 inhibitor |
| CAS | 1884712-47-3 |
| MW: | 386.45 D |
ab 34,00 €
CPI-637
Artikelnummer: Cay23500-1
CPI-637 is an inhibitor of cyclic-AMP response element binding protein (CBP) and adenoviral E1A binding protein of 300 kDa (EP300), a homologous pair of bromodomain-containing proteins (IC50s = 30 and 51 nM in a time-resolved-FRET (TR-FRET) assay). It is selective for CBP and EP300 over the BET family of...
| Schlagworte: | (4R)-1,3,4,5-tetrahydro-4-methyl-6-[1-methyl-3-(1-methyl-1H-pyrazol-4-yl)-1H-indazol-5-yl]-2H-1,5-benzodiazepin-2-one |
| Anwendung: | CREB-binding protein / Histone acetyltransferase p300 inhibitor |
| CAS | 1884712-47-3 |
| MW: | 386.5 D |
ab 44,00 €
