Zu "1610882-30-8" wurden 2 Artikel gefunden!
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TCS-OX2-29 HCl
Artikelnummer: TGM-T4965L-10mg
Description: TCS-OX2-29 is a selective orexin-2 receptor antagonist (IC50 = 40 nM), which plays an important role in pain modulation. Target: Others. Smiles: C([C@@H](NCC=1C=CN=CC1)C(C)(C)C)(=O)N2CC=3C(=CC(OC)=C(OC)C3)CC2.Cl
| Schlagworte: | TCS-OX229, TCS OX229, TCSOX 229, TCS OX2 29, TCSOX-229, TCSOX229 |
| Anwendung: | OX2R antagonist |
| CAS | 1610882-30-8 |
| MW: | 433.97 D |
ab 242,00 €
TCS-OX2-29
Artikelnummer: Cay17419-10
Orexin receptors R1 (OX1R) and OX2R mediate the action of the neuropeptides orexin A and orexin B. TCX-OX2-29 is an antagonist of OX2R (pKi = 7.5) that exhibits >250-fold selectivity for hOX2R compared with hOX1R (IC50s = 40 nM and >10,000 nM, respectively). It blocks the inhibitory action of orexin A on...
| Schlagworte: | (2S)-1-(3,4-dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)-3,3-dimethyl-2-[(4-pyridinylmethyl)amino]-1-butanone,... |
| Anwendung: | OX2R antagonist |
| CAS | 1610882-30-8 |
| MW: | 434 D |
ab 133,00 €
