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Usmarapride
Usmarapride

Artikelnummer: TGM-T63069-100mg

Description: Usmarapride (SUVN-D4010) is a selective, orally active, potent 5-HT4 receptor partial agonist with blood-brain barrier permeability and an EC50 value of 44 nM, used to study cognitive deficits associated with Alzheimer's disease. Target: Others. Smiles:...
Anwendung: 5-HT4 partial agonist
CAS 1428862-33-2
MW: 473.53 D
ab 1.200,00 €
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Usmarapride (oxalate)
Usmarapride (oxalate)

Artikelnummer: Cay35867-1

Usmarapride is a partial agonist of the serotonin (5-HT) receptor subtype 5-HT4. It induces reporter gene expression in CHO cells expressing recombinant human 5-HT4E receptors (EC50 = 44 nM). In vivo, usmarapride (1 and 3 mg/kg) increases novel object exploration time in rats. It also reverses scopolamine-induced...
Schlagworte: SUVN-D4010, 3-[5-[1-(3-methoxypropyl)-4-piperidinyl]-1,3,4-oxadiazol-2-yl]-1-(1-methylethyl)-1H-indazol, monoethanedioate
Anwendung: 5-HT4 partial agonist
CAS 1428862-33-2
MW: 473.5 D
ab 81,00 €
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