Morantel (tartrate)

Morantel is a positive allosteric modulator of neuronal nicotinic acetylcholine receptors (nAChRs). It enhances channel gating of the alpha3beta2 nAChR subtype by binding to non-canonical sites. Formulations containing morantel are used to treat nematode infections in livestock.Formal Name: 1,4,5,6-tetrahydro-1-methyl-2-[(2E)-2-(3-methyl-2-thienyl)ethenyl]-pyrimidine, 2R,3R-dihydroxybutanedioate. CAS Number: 26155-31-7. Synonyms: CP 12,009-18, UK 2964-18. Molecular Formula: C12H16N2S . C4H6O6. Formula Weight: 370.4. Purity: >98%. Formulation: (Request formulation change), A crystalline solid. Solubility: DMF: 33 mg/ml, DMSO: 20 mg/ml, Ethanol: 1 mg/ml, PBS (pH 7.2): 10 mg/ml. lambdamax: 238, 323 nm. SMILES: CN1CCCN=C1/C=C/C2=C(C)C=CS2.OC([C@H](O)[C@@H](O)C(O)=O)=O. InChi Code: InChI=1S/C12H16N2S.C4H6O6/c1-10-6-9-15-11(10)4-5-12-13-7-3-8-14(12)2,5-1(3(7)8)2(6)4(9)10/h4-6,9H,3,7-8H2,1-2H3,1-2,5-6H,(H,7,8)(H,9,10)/b5-4+,/t,1-,2-/m.1/s1. InChi Key: GGXQONWGCAQGNA-UUSVNAAPSA-N.