Produkte von TargetMol

TargetMol aus Boston (Massachusetts) wurde 2015 gegründet und ist ein Experte für Wirkstoffscreening in der Life Science-Community. Das Unternehmen bietet diverse Substanzbibliotheken, darunter FDA-zugelassene Bibliotheken, an und deckt ein breites Spektrum an niedermolekularen Verbindungen wie Inhibitoren und Agonisten sowie rekombinante Proteine und Naturstoffe ab. Die Produkte von TargetMol werden von Forschenden weltweit in Bereichen wie Krebsforschung, Neurobiologie, Inflammation, Immunologie oder Metabolismus eingesetzt.

Mehr Informationen unter: www.targetmol.com

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MS117

Artikelnummer: TGM-T60662-100mg

Description: MS117 is a first-in-class, cell-active, irreversible covalent inhibitor of protein arginine methyltransferase 6 (PRMT6) with an IC50 of 18 nM [1]. Target: Others

MW:

298.38 D

ab 1.023,00 €

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GSD-11

Artikelnummer: TGM-T60672-100mg

Description: GSD-11 inhibits the Akt/mTOR signaling pathway. GSD-11 inhibits the PANC-1 cells migration and colony formation. GSD-11 is a potent and selective anti-austerity agent that has the potential for the pancreatic cancer research [1]. Target: Others

MW:

300.44 D

ab 1.440,00 €

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FPDT

Artikelnummer: TGM-T60676-100mg

Description: FPDT shows anti-glioblastoma activity which is linked to downregulation of the AKT pathway. FPDT has the IC 50 values >100 µM for astrocytes and 45-68 µM for GBM cells [1]. Target: Others

MW:

301.34 D

ab 1.440,00 €

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Elongation factor P-IN-2

Artikelnummer: TGM-T60682-100mg

Description: Elongation factor P-IN-2, a beta-lysine derivative, is a potent inhibitor of elongation factor P (EFP) that affects E. coli proliferation rates [1]. Target: Others

MW:

301.47 D

ab 1.440,00 €

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A1AR antagonist 1

Artikelnummer: TGM-T60687-100mg

Description: A1AR antagonist 1 (compound 18g) is a potent A1 adenosine receptor (AR) antagonist with Ki values of 2.08, 6.91, and 31.2 nM for hA1, hA2A, and hA2B, respectively [1]. Target: Others

MW:

302.33 D

ab 1.440,00 €

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Glutamate-5-kinase-IN-1

Artikelnummer: TGM-T60693-100mg

Description: Glutamate-5-kinase-IN-1 (compound 50) is a potent G5K inhibitor that modifies the ATP binding site architecture for enzyme recognition (MIC = 4.1 µM) and has potential for anti-TB research [1]. Target: Others

MW:

302.37 D

ab 1.440,00 €

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Cedazuridine hydrochloride

Artikelnummer: TGM-T60708-100mg

Description: Cedazuridine (E7727) (Compound 7a) hydrochloride, an orally active cytidine deaminase (CDA) inhibitor with an IC50 of 0.4 µM, can be used for cancer research [1]. Target: Others

MW:

304.68 D

ab 1.440,00 €

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TK-129

Artikelnummer: TGM-T60713-100mg

Description: TK-129 is an orally active, potent inhibitor of KDM5B with an IC50 of 44 nM and is low-toxicity. TK-129 exhibits cardioprotective effects by inhibiting KDM5B and blocking the KDM5B-associated Wnt pathway. TK-129 can be used in cardiovascular disease studies to reduce isoprenaline-induced myocardial...

MW:

305.38 D

ab 747,00 €

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Prohibitin ligand 1

Artikelnummer: TGM-T60722-100mg

Description: Prohibitin ligand 1 (Compound 22i) is a cardioprotective prohibitin ligand that shows in vitro cardioprotective activities at nanomolar concentrations, inducing the pro-survival factor STAT3 phosphorylation [1]. Target: Others

MW:

306.4 D

ab 1.440,00 €

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URAT1 inhibitor 3

Artikelnummer: TGM-T60724-100mg

Description: URAT1 inhibitor 3 is a potent, orally active, selective inhibitor of URAT1 (IC50 = 0.8 nM) demonstrating urate-lowering efficacy, suitable for research in gout and hyperuricemia [1]. Target: Others

MW:

307.13 D

ab 1.440,00 €

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TMX-4113

Artikelnummer: TGM-T60740-100mg

Description: TMX-4113 has potential to be used in cancer that is a phosphodiesterase 6D(PDE6D) and casein kinase 1alpha(CK1alpha) degrader [1]. Target: Others

MW:

308.38 D

ab 1.327,00 €

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HDAC10-IN-2

Artikelnummer: TGM-T60760-100mg

Description: HDAC10-IN-2 (compound 10c) is a potent and highly selective HDAC10 inhibitor (IC50 = 20 nM) that regulates autophagy in aggressive FLT3-ITD positive acute myeloid leukemia cells [1]. Target: Others

MW:

310.39 D

ab 1.440,00 €

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