Produkte von TargetMol

TargetMol aus Boston (Massachusetts) wurde 2015 gegründet und ist ein Experte für Wirkstoffscreening in der Life Science-Community. Das Unternehmen bietet diverse Substanzbibliotheken, darunter FDA-zugelassene Bibliotheken, an und deckt ein breites Spektrum an niedermolekularen Verbindungen wie Inhibitoren und Agonisten sowie rekombinante Proteine und Naturstoffe ab. Die Produkte von TargetMol werden von Forschenden weltweit in Bereichen wie Krebsforschung, Neurobiologie, Inflammation, Immunologie oder Metabolismus eingesetzt.

Mehr Informationen unter: www.targetmol.com

Zu den Katalogen von TargetMol

Für die Filterung wurden keine Ergebnisse gefunden!

KB-5492 FA

Artikelnummer: TGM-T62396L-10mg

Description: KB-5492 FA is a selective sigma receptor inhibitor with antiulcerogenic effects.CAS ??128-52-56-8. Target: Sigma receptor. Smiles: O=C(CN1CCN(CC1)CC2=CC(OC)=C(C(OC)=C2)OC)OC3=CC=C(C=C3)OC.[H]C(O)=O. References: Morimoto Y,et al. Effects of KB-5492, a new anti-ulcer agent, on ethanol- and acidified...

Schlagworte:	KB-5492 FA(113594-64-2 Free base)
MW:	476.52 D

ab 53,00 €

Detailansicht

Bewerten

KDM1/CDK1-IN-1

Artikelnummer: TGM-T62405-100mg

Description: KDM1/CDK1-IN-1 (compound 4) is a potent inhibitor of KDM1 (IC50: 0.096 µM) and CDK1 (IC50: 0.078 µM), blocking the cell cycle of HOP-92 cells in the G2/M phase and inducing apoptosis. It is highly cytotoxic to CCRF-CEM cells (IC50: 16.34 µM), HOP-92 cells (IC50: 3.45 µM), and Hep-G2 cells (IC50: 7.79...

MW:

431.47 D

ab 1.440,00 €

Detailansicht

Bewerten

AD012

Artikelnummer: TGM-T62831-100mg

Description: AD012 is a dual inhibitor of cACE/NEP that utilizes the previously reported C-domain selective ACE inhibitor lenopril-tryptophan synthesis, potentially offering potent anti-hypertensive and cardioprotective effects. Target: Others

MW:

456.53 D

ab 1.440,00 €

Detailansicht

Bewerten

Antitumor agent-54

Artikelnummer: TGM-T62835-100mg

Description: Antitumor agent-54 (Compound C11) is a 14-3-3eta protein inhibitor (KD: 35 µM). antitumor agent-54 inhibits several typical human hepatocellular carcinoma cell lines. antitumor agent-54 blocks the cell cycle in the G1-S phase and induces apoptosis, showing good metabolic stability. It exhibits good...

MW:

456.58 D

ab 1.440,00 €

Detailansicht

Bewerten

Artikelnummer: TGM-T62836-100mg

Description: Hit 1, an activator of insulin-degrading enzymes (IDE) (EC50: 5.5 µM), reduces glucose-stimulated insulin secretion. Target: Others

MW:

456.58 D

ab 1.440,00 €

Detailansicht

Bewerten

AR antagonist 4

Artikelnummer: TGM-T62838-100mg

Description: AR antagonist 4 (Compound 67-b) is an orally active androgen receptor (AR) antagonist with an IC50 of 246.6 nM for wild-type AR. Target: Others

MW:

456.62 D

ab 1.440,00 €

Detailansicht

Bewerten

5-HT1A antagonist 1

Artikelnummer: TGM-T62843-100mg

Description: 5-HT1A antagonist 1 (compound 6f) is a potent and selective 5-HT1A receptor antagonist (Ki: 35 nM) and can be utilized in the study of central nervous system disorders. Target: Others

MW:

456.97 D

ab 1.440,00 €

Detailansicht

Bewerten

Freselestat quarterhydrate

Artikelnummer: TGM-T62846-100mg

Description: Freselestat quarterhydrate (ONO-6818 quarterhydrate) is a potent, orally active inhibitor of neutrophil elastase (Ki: 12.2 nM). The quarterhydrate is more than 100-fold less active against other proteases, including trypsin, proteinase 3, pancreatic elastase, thrombin, fibrin, collagenase, histone G,...

MW:

457.03 D

ab 1.080,00 €

Detailansicht

Bewerten

GSK2945 hydrochloride

Artikelnummer: TGM-T62852-100mg

Description: GSK2945 hydrochloride is a tertiary amine and a highly specific antagonist of Rev-erbalpha/REV-ERBalpha (mouse/human reverse erythropoietic virus alpha) with an EC50 value of 21.5 µM and 20.8 µM, respectively.GSK2945 hydrochloride increases cholesterol 7alpha-hydroxylase ( The EC50 values were 21 µM and...

MW:

457.8 D

Bitte fragen Sie den aktuellen Preis für diesen Artikel an.

Detailansicht

Bewerten

K203

Artikelnummer: TGM-T62857-100mg

Description: K203 is a potent tabun-inhibited AChE reactivator and is an important antidote to organophosphorus poisoning. Target: Others

MW:

458.15 D

ab 1.440,00 €

Detailansicht

Bewerten

CK2-IN-3

Artikelnummer: TGM-T62862-100mg

Description: CK2-IN-3 is a potent and selective CK2 inhibitor (Kd: 12 nM) with IC50 values of 1.51 µM for CK2alpha and 7.64 µM for CK2alpha'. CK2-IN-3 can be used in cancer research. Target: Others

MW:

458.46 D

ab 1.440,00 €

Detailansicht

Bewerten

844-TFM

Artikelnummer: TGM-T62866-100mg

Description: 844-TFM is an NBTI (novel bacterial topoisomerase inhibitor) DNA gyrase inhibitor (IC50: 1.5 µM). 844-TFM exhibits bactericidal activity against Mycobacterium abscessus. Target: Others

MW:

458.48 D

ab 1.440,00 €

Detailansicht

Bewerten

12309 von 12311 Seiten