Produkte von TargetMol
TargetMol aus Boston (Massachusetts) wurde 2015 gegründet und ist ein Experte für Wirkstoffscreening in der Life Science-Community. Das Unternehmen bietet diverse Substanzbibliotheken, darunter FDA-zugelassene Bibliotheken, an und deckt ein breites Spektrum an niedermolekularen Verbindungen wie Inhibitoren und Agonisten sowie rekombinante Proteine und Naturstoffe ab. Die Produkte von TargetMol werden von Forschenden weltweit in Bereichen wie Krebsforschung, Neurobiologie, Inflammation, Immunologie oder Metabolismus eingesetzt.
Mehr Informationen unter: www.targetmol.com
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Tirofiban hydrochloride monohydrate
Artikelnummer: TGM-T2537-100mg
Description: Tirofiban hydrochloride monohydrate (MK-383 Hydrochloride) is a potent non-peptide, glycoprotein IIb/IIIa (integrins alphaIIbbetaIII) antagonist. Target: Integrin, ATPase. Smiles: O.Cl.CCCCS(=O)(=O)N[C@@H](Cc1ccc(OCCCCC2CCNCC2)cc1)C(O)=O. References: Winter JP, Juergens CP. Cardiovasc Hematol Disord...
| Schlagworte: | Tirofiban Hydrochloride, MK-383 Hydrochloride |
| Anwendung: | Platelet aggregation inhibitor, Glycoprotein IIb/IIIa receptor antagonist |
| CAS | 150915-40-5 |
| MW: | 495.07 D |
ab 39,00 €
Prucalopride
Artikelnummer: TGM-T2542-100mg
Description: Prucalopride (R-93877) is a selective, high-affinity 5-HT4A/4B receptor agonist (Ki: 2.5/8 nM). It has >290-fold selectivity for 5-HT4A/4B receptor than other 5-HT receptor subtypes. Target: 5-HT Receptor. Smiles: COCCCN1CCC(CC1)NC(=O)c1cc(Cl)c(N)c2CCOc12. References: Briejer MR, et al. Eur J Pharmacol,...
| Schlagworte: | R-93877 |
| Anwendung: | Targets 5-hydroxytryptamine receptor 4 (HTR4) |
| CAS | 179474-81-8 |
| MW: | 367.87 D |
ab 30,00 €
Cabazitaxel
Artikelnummer: TGM-T2543-1mL
Description: Cabazitaxel (taxoid XRP6258) is a taxane and antineoplastic agent which is currently used in the therapy of castration-resistant metastatic prostate cancer after failure of docetaxel. Target: Autophagy, Microtubule Associated. Smiles:...
| Schlagworte: | RPR-116258A, XRP6258, taxoid XRP6258, TXD 258 |
| Anwendung: | Targets tubulin beta (TUBB) |
| CAS | 183133-96-2 |
| MW: | 835.93 D |
48,00 €
Bazedoxifene acetate
Artikelnummer: TGM-T2544-100mg
Description: Bazedoxifene acetate (WAY-TES 424) is a novel selective estrogen receptor modulator (SERM). Target: Estrogen/progestogen Receptor, Estrogen Receptor/ERR. Smiles: C(=O)(C)O.c1c(cc2c(c1)n(c(c2C)c1ccc(cc1)O)Cc1ccc(cc1)OCCN1CCCCCC1)O. References: Miller CP, et al. J Med Chem, 2001, 44(11), 1654-1657.
| Schlagworte: | WAY-140424, TSE 424, WAY-TES 424 |
| Anwendung: | Osteoporosis agent, Selective estrogen receptor modulator (SERM) |
| CAS | 198481-33-3 |
| MW: | 530.67 D |
ab 38,00 €
Pimozide
Artikelnummer: TGM-T2546-1mL
Description: Pimozide (R6238) is a diphenylbutylpiperidine derivative and a dopamine antagonist with the antipsychotic property. Pimozide selectively inhibits type 2 dopaminergic receptors in the central nervous system (CNS), thereby decreasing dopamine neurotransmission and reducing the occurrence of the motor and...
| Schlagworte: | R6238 |
| Anwendung: | Targets dopamine receptor D2 (DRD2) |
| CAS | 2062-78-4 |
| MW: | 461.55 D |
ab 30,00 €
Diflorasone
Artikelnummer: TGM-T2548-100mg
Description: Diflorasone is a synthetic glucocorticoid with anti-inflammatory and immunosuppressive properties. Like other glucocorticoids, diflorasone enters the cell by diffusion across the cell membrane and binds to the glucocorticoid receptor (GR) in the cytoplasm. The receptor complex subsequently translocates...
| Anwendung: | Targets glucocorticoid receptor (NR3C1, GR) |
| CAS | 2557-49-5 |
| MW: | 410.45 D |
ab 35,00 €
Robenidine hydrochloride
Artikelnummer: TGM-T2549-100mg
Description: Robenidine hydrochloride (Robenidine Hydrochoride) is an anticoccidial agent mainly used in poultry. Target: Antibacterial, Parasite, Antibiotic. Smiles: Cl.Clc1ccc(\C=N\NC(=N)N\N=C\c2ccc(Cl)cc2)cc1. References: Yeom H, et al. Arch Pharm Res. 2013 Mar,36(3):359-65.
| Schlagworte: | Dexium, Robenidine Hydrochoride, Toraxine, Nugatex, Rasexinium |
| Anwendung: | Coccidiostat (for poultry) |
| CAS | 25875-50-7 |
| MW: | 370.66 D |
ab 35,00 €
Etofenamate
Artikelnummer: TGM-T2553-1mL
Description: Etofenamate is a non-steroidal anti-inflammatory drug (NSAID) used for the treatment of joint and muscular pain. Target: COX. Smiles: N(C1=C(C(OCCOCCO)=O)C=CC=C1)C2=CC(C(F)(F)F)=CC=C2. References: Bender T, et al. Arzneimittelforschung. 2001,51(6):489-92.
| Anwendung: | Targets prostaglandin-endoperoxide synthase 1 [EC:1.14.99.1] (PTGS1, COX1) |
| CAS | 30544-47-9 |
| MW: | 369.33 D |
ab 35,00 €
Aclidinium bromide
Artikelnummer: TGM-T2555-100mg
Description: Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis or emphysema. Aclidinium has not been implicated in causing liver enzyme elevations or clinically apparent acute liver injury. Target: AChR....
| Schlagworte: | LAS 34273, LAS-W 330 |
| Anwendung: | Bronchodilator, Muscarinic acetylcholine receptor antagonist |
| CAS | 320345-99-1 |
| MW: | 564.55 D |
ab 32,00 €
JNJ-3534
Artikelnummer: TGM-T25557-100mg
Description: JNJ-3534 is an oral active modulator of RORgammat. Target: Others. Smiles: NA
| Schlagworte: | JNJ3534, JNJ 3534 |
Bitte fragen Sie den aktuellen Preis für diesen Artikel an.
Cladribine
Artikelnummer: TGM-T2558-100mg
Description: Cladribine (2CdA), an adenosine deaminase inhibitor, is utilized in the treatment of lymphoproliferative diseases. Target: Adenosine deaminase, Apoptosis. Smiles: Nc1nc(Cl)nc2n(cnc12)[C@H]1C[C@H](O)[C@@H](CO)O1. References: Ma J, et al. BMC Cancer. 2011, 11, 255.
| Schlagworte: | 2-Chloro-2'-deoxyadenosine, CldAdo, 2-chlorodeoxyadenosine, 2CdA |
| Anwendung: | Targets ribonucleoside-diphosphate reductase subunit M1 [EC:1.17.4.1] (RRM1) |
| CAS | 4291-63-8 |
| MW: | 285.69 D |
ab 33,00 €
Allylestrenol
Artikelnummer: TGM-T2559-1mL
Description: Allylestrenol (Gestanin) is a synthetic steroid with progestational activity. Target: Estrogen/progestogen Receptor. Smiles: [H][C@@]12CC[C@@](O)(CC=C)[C@@]1(C)CC[C@]1([H])[C@@]3([H])CCCC=C3CC[C@@]21[H]. References: Madauss KP, et al. Med Res Rev. 2007 May,27(3):374-400.
| Schlagworte: | Gestanin, Gestanon, Gestanol |
| Anwendung: | Targets progesterone receptor (PGR, NR3C3) |
| CAS | 432-60-0 |
| MW: | 300.48 D |
29,00 €