Zu "K22599" wurden 28 Artikel gefunden!
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COVID-19 Forschung
Ritonavir
Artikelnummer: Cay13872-10
Ritonavir is an HIV protease inhibitor. It inhibits recombinant HIV-1 protease by 79% when used at a concentration of 0.5 nM. It inhibits HIV-13B-induced cell death in MT-4 human T cell leukemia cells (EC50 = 25 nM) as well as cell death induced by HIV-1LAI, HIV-2ROD, and HIV-2EHO in human MT-2 cells (IC50s = 0.045,...
| Schlagworte: | A-84538, ABT-538, NSC 693184, RTV,... |
| Anwendung: | Antiviral, HIV protease inhibitor |
| CAS | 155213-67-5 |
| MW: | 720.9 D |
ab 42,00 €
Saquinavir (mesylate)
Artikelnummer: Cay9001893-5
Saquinavir is an HIV protease inhibitor (Kis = 0.12 and 50 = 2 nM). It also inhibits the activity of the severe acute respiratory coronavirus 2 (SARS-CoV-2) main protease (Mpro), also known as 3C-like protease (3CLpro), with an IC50 value of 9.92 µM.Formal Name:...
| Schlagworte: | Ro 31-8959/003,... |
| Anwendung: | HIV protease inhibitor |
| CAS | 149845-06-7 |
| MW: | 767 D |
ab 67,00 €
Tipranavir
Artikelnummer: Cay21028-1
Tipranavir is a potent, orally bioavailable nonpeptidic HIV aspartyl protease inhibitor (Ki = 95%. Formulation: (Request formulation change), A crystalline solid. Solubility: Chloroform: slightly soluble, Methanol: slightly soluble. lambdamax: 254 nm. SMILES:...
| Schlagworte: | PNU-140690,... |
| Anwendung: | HIV protease inhibitor |
| CAS | 174484-41-4 |
| MW: | 602.7 D |
ab 238,00 €
COVID-19 Forschung
Nelfinavir . mesylate
Artikelnummer: AG-CR1-3726-M010
Soluble in DMSO (15mg/ml), DMF (20mg/ml) or ethanol (20mg/ml). Nelfinavir is an orally bioavailable competitive inhibitor of the human immunodeficiency virus. It potently inhibits HIV-1 (Ki=2nM) and HIV-2 protease in vitro. HIV-1 protease is important for the replication of the virus within the cell and the release...
| Schlagworte: | AG-1343, Nelfin, Viracep |
| Anwendung: | Antiviral, HIV protease inhibitor |
| CAS | 159989-65-8 |
| MW: | 663.89 D |
ab 55,00 €
COVID-19 Forschung
Saquinavir . mesylate
Artikelnummer: AG-CR1-3727-M010
Soluble in DMSO (10mg/ml). Saquinavir is an antiretroviral inhibitor of the human immunodeficiency virus. It potently inhibits HIV-1 (Ki=0.12nM) and HIV-2 (Ki<0.1nM) protease in vitro. HIV-1 protease is important for the replication of the virus within the cell and the release of mature viral particles from the...
| Schlagworte: | Ro 31-8959 |
| Anwendung: | Antiviral, HIV protease inhibitor |
| CAS | 149845-06-7 |
| MW: | 766.95 D |
ab 55,00 €
Indinavir sulfate
Artikelnummer: TGM-T5863-25mg
Description: Indinavir sulfate (L735524 sulfate) is a HIV protease inhibitor.It inhibits the HIV-1 protease with an IC50 value of 0.41 nM and Ki value of 0.24 nM. Target: SARS-CoV, HIV Protease. Smiles: OS(O)(=O)=O.CC(C)(C)NC(=O)[C@@H]1CN(Cc2cccnc2)CCN1C[C@@H](O)C[C@@H](Cc1ccccc1)C(=O)N[C@@H]1[C@H](O)Cc2ccccc12....
| Schlagworte: | MK-639 sulfate, L735524 sulfate |
| Anwendung: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 157810-81-6 |
| MW: | 711.87 D |
ab 33,00 €
Fosamprenavir (calcium salt)
Artikelnummer: Cay21609-1
Fosamprenavir is a prodrug form of the HIV-1 protease inhibitor amprenavir (Cay-15369). It is converted to amprenavir by alkaline phosphatase in the intestinal epithelium. Formulations containing fosamprenavir have been used in the treatment of HIV infections.Formal Name:...
| Schlagworte: | GW 433908G,... |
| Anwendung: | Antiviral, HIV protease inhibitor prodrug |
| CAS | 226700-81-8 |
| MW: | 623.7 D |
ab 38,00 €
Des(benzylpyridyl) Atazanavir
Artikelnummer: LKT-D1872.1
Atazanavir metabolite, HIV protease inhibitor.
| Anwendung: | Atazanavir metabolite, HIV protease inhibitor |
| CAS | 1192224-24-0 |
| MW: | 537.66 D |
ab 204,00 €
Saquinavir-d9
Artikelnummer: Cay28906-1
Saquinavir-d9 is intended for use as an internal standard for the quantification of saquinavir (Cay-9001893) by GC- or LC-MS. Saquinavir is an HIV protease inhibitor (Kis = 0.12 and 50 = 2 nM). It also inhibits the activity of the severe acute respiratory coronavirus 2 (SARS-CoV-2) main protease (Mpro), also known...
| Schlagworte: | (2S)-N1-[(1S,2R)-3-[(3S,4aS,8aS)-3-[[(1,1-di(methyl-d3)ethyl-2,2,2-d3)amino]carbonyl]octahydro-2(1H)-isoquinolinyl]-2-hydr... |
| Anwendung: | GC-MS, LC-MS, internal standard, quantification, HIV protease inhibitor |
| CAS | 1356355-11-7 |
| MW: | 679.9 D |
533,00 €
Tipranavir-d4
Artikelnummer: Cay28907-1
Tipranavir-d4 is intended for use as an internal standard for the quantification of tipranavir (Cay-21028) by GC- or LC-MS. Tipranavir is a potent, orally bioavailable nonpeptidic HIV aspartyl protease inhibitor (Ki = 99% deuterated forms (d1-d4). Formulation: (Request formulation change), A solid. Solubility:...
| Schlagworte: | N-(3-((R)-1-((R)-4-hydroxy-2-oxo-6-phenethyl-6-(propyl-1,1,2,2-d4)-5,6-dihydro-2H-pyran-3-yl)propyl)phenyl)-5-(trifluorome... |
| Anwendung: | GC-MS, LC-MS, internal standard, quantification, HIV protease inhibitor |
| CAS | 1217819-15-2 |
| MW: | 606.7 D |
588,00 €
COVID-19 Forschung
Darunavir
Artikelnummer: AG-CR1-3712-M010
Soluble in DMSO (30mg/ml) or DMF (30mg/ml). Darunavir is a highly potent HIV protease inhibitor (IC50=3-6nM, depending on laboratory HIV-1 strain), an antiretroviral medication used to treat and prevent HIV/AIDS. Darunavir is a second generation HIV-1 protease inhibitor that inhibits replication of various...
| Schlagworte: | TMC114, TMC41629, UIC-94017, HSDB 7788, Prezista |
| Anwendung: | Antiviral, HIV protease inhibitor |
| CAS | 206361-991 |
| MW: | 547.7 D |
143,00 €
COVID-19 Forschung
Lopinavir
Artikelnummer: AG-CR1-3715-M025
Soluble in ethanol (20mg/ml), DMSO (15mg/ml) or dimtheylformamide (15mg/ml). The antiviral agent Lopinavir is a potent inhibitor of HIV-1 protease (Ki=1.3pM for wild-type enzyme) and has been shown to block the replication of clinical isolates of HIV (EC50s=5-52nM). Lopinavir is an antiretroviral of the protease...
| Schlagworte: | A-157378.0, ABT-378, Aluviran |
| Anwendung: | Antiviral, HIV protease inhibitor |
| CAS | 192725-17-0 |
| MW: | 628.8 D |
ab 39,00 €