Zu "K08655" wurden 25 Artikel gefunden!
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1G244
Artikelnummer: Cay18306-10
1G244 is an inhibitor of dipeptidyl peptidase 8 (DPP-8) and DPP-9 (IC50s = 14 and 53 nM, respectively). It is selective for DPP-8 and DPP-9 over DPP-4, DPP-2, and fibroblast activation protein (FAP, IC50s = >100 µM for all). 1G244 (20 µM) inhibits the differentiation of 3T3-L1 cells into adipocytes. It induces...
| Schlagworte: | PTX1210, 2S-amino-4-[4-[bis(4-fluorophenyl)methyl]-1-piperazinyl]-1-(1,3-dihydro-2H-isoindol-2-yl)-1,4-butanedione |
| Anwendung: | DPP8/DPP9 inhibitor |
| CAS | 847928-32-9 |
| MW: | 504.6 D |
ab 112,00 €
DPP8 assay kit
Artikelnummer: BPS-80208
The DPP8 Fluorescent Activity Assay kit is designed to measure DPP8 activity using purified DPP8 or DPP8 extracts. It comes in a convenient 96-well format, with purified DPP8 enzyme, DPP8 substrate, and DPP8 assay buffer for 100 enzyme reactions. The Key to DPP8 Fluorescent Activity Assay is the fluorogenic...
| Schlagworte: | Dipeptidylpeptidase 8, MSTP141, |
| Anwendung: | DPP8 assays, inhibitor screening, HTS |
812,00 €
DPP8, active human recombinant protein
Artikelnummer: BPS-80080
Active human DPP8 (Dipeptidylpeptidase 8) (GenBank Accession No. NM_197960), (full length) with N-terminal GST tag, MW=129.3 kDa, expressed in a Baculovirus infected Sf9 cell expression system.
| Schlagworte: | DP8, DPRP1, DPRP-1, MSTP097, DPP VIII, Dipeptidyl peptidase 8, Prolyl dipeptidase DPP8, Dipeptidyl peptidase VIII,... |
| Anwendung: | Enzyme kinetics, inhibitor screening |
| MW: | 129.3 kD |
678,00 €
Talabostat (mesylate)
Artikelnummer: Cay29007-25
Talabostat is a non-selective inhibitor of dipeptidyl peptidases (DPPs), including DPP-4, DPP-7, DPP-8, DPP-9, fibroblast activation protein (FAP), and prolyl endopeptidase (PREP, IC50s = >4, 310, 4, 11, 560, and 390 nM, respectively). It inhibits proliferation of superantigen-stimulated human peripheral blood...
| Schlagworte: | Val-boro-Pro, B-[(2R)-1-[(2S)-2-amino-3-methyl-1-oxobutyl]-2-pyrrolidinyl]-boronic acid, methanesulfonate |
| Anwendung: | Dipeptidyl peptidase inhibitor |
| CAS | 150080-09-4 |
| MW: | 310.2 D |
ab 73,00 €
Anti-DPP8
Artikelnummer: ARG40130.100
Protein function: Dipeptidyl peptidase that cleaves off N-terminal dipeptides from proteins having a Pro or Ala residue at position 2. [The UniProt Consortium]
| Schlagworte: | Anti-DP8, Anti-DPP8, Anti-DPRP1, Anti-DPRP-1, Anti-MSTP097, Anti-DPP VIII, Anti-Dipeptidyl peptidase 8, Anti-Prolyl... |
| Anwendung: | FC, IHC (paraffin), WB |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human |
616,00 €
Anti-DPP8
Artikelnummer: ATA-HPA008706.100
Protein function: Dipeptidyl peptidase that cleaves off N-terminal dipeptides from proteins having a Pro or Ala residue at position 2. [The UniProt Consortium] Buffer: 40% glycerol and PBS (pH 7.2). 0.02% sodium azide is added as preservative. Highest antigen sequence identity to mouse: 96% and to rat: 95%
| Schlagworte: | Anti-DP8, Anti-DPP8, Anti-DPRP1, Anti-DPRP-1, Anti-MSTP097, Anti-DPP VIII, Anti-Dipeptidyl peptidase 8, Anti-Prolyl... |
| Anwendung: | ICC, IHC |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human |
ab 369,00 €
Talabostat . mesylate
Artikelnummer: AG-CR1-3541-M010
Talabostat is an orally bioavailable non-selective inhibitor of dipeptidyl-peptidases (DPPs), including DPP-4, DPP-7/QPP, DPP-8, DPP-9, fibroblast activation protein (FAP) and prolyl endopeptidase (PREP, PEP) (IC50s = >4, 310, 4, 11, 560 and 390 nM, respectively). Talabostat induces powerful anti-tumor immune...
| Schlagworte: | Valinyl-L-boroproline, Val-boro-Pro, BXCL 701, PT-100, B-[(2R)-1-[(2S)-2-Amino-3-methyl-1-oxobutyl]-2-pyrrolidinyl]boronic... |
| Anwendung: | Dipeptidyl-peptidases (DPP) inhibitor |
| CAS | 150080-09-4 |
| MW: | 310,2 D |
ab 66,00 €
Human DPP8 (Dipeptidyl Peptidase 8) ELISA Kit
Artikelnummer: ELK-ELK4591.48
The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Human DPP8. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Human DPP8. Next,...
| Schlagworte: | DP8, DPRP1, DPRP-1, MSTP097, DPP VIII, Dipeptidyl peptidase 8, Prolyl dipeptidase DPP8, Dipeptidyl peptidase VIII,... |
| Anwendung: | ELISA |
| Spezies-Reaktivität: | human |
ab 374,00 €
Mouse DPP8 (Dipeptidyl Peptidase 8) ELISA Kit
Artikelnummer: ELK-ELK6504.48
The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Mouse DPP8. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Mouse DPP8. Next,...
| Schlagworte: | DP8, DPP VIII, Dipeptidyl peptidase 8, Dipeptidyl peptidase VIII |
| Anwendung: | ELISA |
| Spezies-Reaktivität: | mouse |
ab 374,00 €
Talabostat
Artikelnummer: TGM-T37861-10mg
Description: Talabostat (PT100, Val-boroPro) is a potent, nonselective and orally available dipeptidyl peptidase IV (DPP-IV) inhibitor with a Ki of 0.18 nM. Target: Others. Smiles: CC(C)[C@H](N)C(=O)N1CCC[C@H]1B(O)O. References: Connolly BA, et al. Dipeptide boronic acid inhibitors of dipeptidyl peptidase IV:...
| Anwendung: | Targets dipeptidyl-peptidase 8 [EC:3.4.14.5] (DPP8) |
| CAS | 149682-77-9 |
| MW: | 214.07 D |
ab 101,00 €
Talabostat mesylate
Artikelnummer: TGM-T4042-10mg
Description: Talabostat mesylate (PT100) is an orally active, selective inhibitor of dipeptidyl peptidases IV (DPP4, IC50: 0.18 nM), including tumor-associated fibroblast activation protein. This agent may also stimulate the production of colony stimulating factors, such as granulocyte colony-stimulating factor...
| Schlagworte: | PT100, Val-boroPro |
| Anwendung: | Targets dipeptidyl-peptidase 8 [EC:3.4.14.5] (DPP8) |
| CAS | 150080-09-4 |
| MW: | 310.18 D |
ab 48,00 €
DPP8 (human), recombinant protein
Artikelnummer: ABS-PP-5158-L.100
Protein function: Dipeptidyl peptidase that cleaves off N-terminal dipeptides from proteins having a Pro or Ala residue at position 2. [The UniProt Consortium]
| Schlagworte: | Dipeptidyl peptidase 8, DP8, Dipeptidyl peptidase IV-related protein 1, DPRP-1, Dipeptidyl peptidase VIII, DPP VIII,... |
| Exprimiert in: | E.coli |
| Ursprungsart: | human |
| MW: | 52.5 kD |
ab 115,00 €