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AR (human) Reporter Assay Kit
Artikelnummer: IB-IB03001
This nuclear receptor assay system utilizes proprietary non-human mammalian cells engineered to provide constitutive, high-level expression of full-length, unmodified human androgen receptor (NR3C4), a ligand-dependent transcription factor commonly referred to as AR. INDIGO's reporter cells include the luciferase...
| Schlagworte: | AR, DHTR, Androgen receptor, Dihydrotestosterone receptor, Nuclear receptor subfamily 3 group C member 4 |
| Anwendung: | Functional activity screening |
| Spezies-Reaktivität: | human |
ab 1.588,00 €
NEU
Testosterone Enanthate (exempt preparation)
Artikelnummer: Cay46044-1
Testosterone enanthate (exempt preparation) (Cay46044) is an analytical reference standard categorized as an anabolic androgenic steroid. Testosterone enanthate is a prodrug form of testosterone (CayISO60154, CayISO00154, Cay15645). It has been found in performance-enhancing drug (PED) samples seized by law...
| Schlagworte: | NSC 17591, 17beta-[(1-oxoheptyl)oxy]-androst-4-en-3-one |
| Anwendung: | Analytical reference standard, anabolic androgenic steroid |
| CAS | 315-37-7 |
| MW: | 400.6 D |
299,00 €
NEU
Testosterone Cypionate (exempt preparation)
Artikelnummer: Cay46045-1
Testosterone cypionate (exempt preparation) (Cay46045) is an analytical reference standard categorized as an anabolic androgenic steroid. Testosterone cypionate is a prodrug form of testosterone (CayISO60154, CayISO00154, Cay15645). It has been detected in hair samples from competition athletes and plasma samples...
| Schlagworte: | NSC 9157, 17beta-(3-cyclopentyl-1-oxopropoxy)-androst-4-en-3-one |
| Anwendung: | Analytical reference standard, anabolic androgenic steroid |
| CAS | 58-20-8 |
| MW: | 412.61 D |
299,00 €
NEU
Testosterone Isobutyrate
Artikelnummer: Cay41937-1
Testosterone isobutyrate (Cay41937) is an analytical reference standard categorized as an anabolic androgenic steroid. Testosterone isobutyrate is a prodrug form of testosterone (CayISO60154, CayISO00154, Cay15645). Testosterone isobutyrate is regulated as a Schedule III compound in the United States. This product...
| Schlagworte: | Testosterone 17-isobutyrate, Testosterone 2-methylpropanoate, 17beta-(2-methyl-1-oxopropoxy)-androst-4-en-3-one |
| Anwendung: | Analytical reference standard, anabolic androgenic steroid |
| CAS | 1169-49-9 |
| MW: | 358.51 D |
ab 249,00 €
ARD-266
Artikelnummer: Cay45321-1
ARD-266 is a proteolysis-targeting chimera (PROTAC) containing an androgen receptor antagonist conjugated to a VHL ligand via a piperidine-alkyne linker. It induces degradation of the androgen receptor in LNCaP, VCaP, and 22Rv1 prostate cancer cells with half-maximal degradation concentration (DC50) values of 0.54,...
| Schlagworte: | (2S,4R)-N-[(1S)-3-[4-[2-[4-[[[trans-3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]amino]carbonyl]phenyl]ethyny... |
| Anwendung: | Androgen receptor (AR/NR3C4) degradation driving PROTAC |
| CAS | 2666951-70-6 |
| MW: | 915.53 D |
ab 139,00 €
Rezvilutamide
Artikelnummer: Cay45332-10
Rezvilutamide is a non-steroidal androgen receptor antagonist. It reduces secretion of prostate-specific androgen (PSA) from LNCaP prostate cancer cells (IC50 = 22 nM) and reduces proliferation of the same cells (IC50 = 33 nM). Formulations containing rezvilutamide have been used in the treatment of prostate...
| Schlagworte: | SHR-3680,... |
| Anwendung: | Non-steroidal androgen receptor antagonist |
| CAS | 1572045-62-5 |
| MW: | 479.47 D |
ab 271,00 €
MK-0773
Artikelnummer: Cay43202-1
MK-0773 is a selective androgen receptor modulator (SARM). It selectively binds to the androgen receptor (AR, IC50 = 6.6 nM) over the glucocorticoid and progesterone receptors (IC50s = >2 µM for both). It is a partial agonist of AR that increases AR-dependent transcription in a reporter assay using MDA-MB-453 cells...
| Schlagworte: | PF-05314882, (4aS,4bS,6aS,7S,9aS,9bS,11aR)-3-fluoro-2,4a,4b,5,6,6a,7,... |
| Anwendung: | Selective androgen receptor modulator (SARM) |
| CAS | 606101-58-0 |
| MW: | 479.6 D |
ab 105,00 €
Anti-Androgen Receptor, clone r2F12
Artikelnummer: NSJ-V5924SAF-100UG
1 mg/ml in 1X PBS, BSA free, sodium azide free. Androgen receptor (AR), encoded by the AR gene and also known as nuclear receptor subfamily 3 group C member 4 (NR3C4), is a ligand-activated nuclear hormone receptor that mediates cellular responses to androgens such as testosterone and dihydrotestosterone. AR...
| Schlagworte: | Anti-AR, Anti-Androgen receptor, Anti-Dihydrotestosterone receptor, Anti-Nuclear receptor subfamily 3 group C member 4,... |
| Anwendung: | IHC |
| Wirt: | Mouse |
| Spezies-Reaktivität: | human |
810,00 €
Anti-Androgen Receptor, clone r2F12
Artikelnummer: NSJ-V5924-100UG
0.2 mg/ml in 1X PBS with 0.05% BSA, 0.05% sodium azide. Androgen receptor (AR), encoded by the AR gene and also known as nuclear receptor subfamily 3 group C member 4 (NR3C4), is a ligand-activated nuclear hormone receptor that mediates cellular responses to androgens such as testosterone and dihydrotestosterone. AR...
| Schlagworte: | Anti-AR, Anti-Androgen receptor, Anti-Dihydrotestosterone receptor, Anti-Nuclear receptor subfamily 3 group C member 4,... |
| Anwendung: | IHC |
| Wirt: | Mouse |
| Spezies-Reaktivität: | human |
ab 375,00 €
Anti-Androgen Receptor, clone MSVA-367R
Artikelnummer: NSJ-V6092-100UG
Antibody in 1X PBS with 0.05% BSA, 0.05% sodium azide. Androgen receptor (AR), encoded by the AR gene and also known as nuclear receptor subfamily 3 group C member 4 (NR3C4), is a ligand-activated nuclear hormone receptor that mediates cellular responses to androgens such as testosterone and dihydrotestosterone. AR...
| Schlagworte: | Anti-AR, Anti-Androgen receptor, Anti-Dihydrotestosterone receptor, Anti-Nuclear receptor subfamily 3 group C member 4,... |
| Anwendung: | IHC |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human |
ab 684,00 €
Enzalutamide-d3
Artikelnummer: Cay45044-1
An internal standard for the quantification of enzalutamide by GC- or LC-MS. SMILES: S=C1N(C2=CC(F)=C(C=C2)C(NC([2H])([2H])[2H])=O)C(C)(C(N1C3=CC(C(F)(F)F)=C(C=C3)C#N)=O)C. InChi Code:...
| Schlagworte: | 4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-thioxo-1-imidazolidinyl]-2-fluoro-N-(methyl-d3)-benzamide |
| Anwendung: | GC-MS, LC-MS, internal standard, quantification, non-steroidal androgen receptor antagonist |
| CAS | 1443331-82-5 |
| MW: | 467.46 D |
535,00 €
Anti-Zebrafish Androgen receptor / AR
Artikelnummer: NSJ-RZ1202
0.5mg/ml if reconstituted with 0.2ml sterile DI water. Androgen receptor (AR) is a nuclear hormone receptor that functions as a ligand-activated transcription factor, mediating the biological effects of androgens such as testosterone and 11-ketotestosterone. In zebrafish (Danio rerio), AR plays a critical role in...
| Schlagworte: | Anti-ar, Anti-Androgen receptor, Anti-Dihydrotestosterone receptor, Anti-Nuclear receptor subfamily 3 group C member 4,... |
| Anwendung: | WB |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | zebrafish |
948,00 €