Zu "K08421" wurden 29 Artikel gefunden!
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ZQ-16
Artikelnummer: Cay43951-10
ZQ-16 is an agonist of G protein-coupled receptor 84 (GPR84). It induces calcium mobilization in HEK293 cells expressing GPR84 and Galpha16 (EC50 = 0. µM). ZQ-16 is selective for GPR84 over free fatty acid receptor 1 (FFAR1/GPR40), FFAR3/GPR41, GPR119, and FFAR4/GPR120 at 100 µM. ZQ-16 also inhibits...
| Schlagworte: | 2-HTP |
| Anwendung: | GPR84 agonist |
| CAS | 376616-73-8 |
| MW: | 228.31 D |
ab 127,00 €
GPR84 Antagonist 8
Artikelnummer: Cay43485-10
GPR84 antagonist 8 is an antagonist of G protein-coupled receptor 84 (GPR84). It inhibits calcium mobilization induced by 6-OAU (Cay17687) in HEK293 cells expressing human GPR84 and Galpha16 (IC50 = 716 nM). GPR84 antagonist 8 (10 µM) inhibits 6-OAU-enhanced phagocytosis of E. coli by primary mouse bone...
| Schlagworte: | EN 818470, G Protein-coupled Receptor 84 Antagonist 8,... |
| Anwendung: | GPR84 antagonist |
| CAS | 1445846-30-9 |
| MW: | 421.45 D |
ab 294,00 €
6-OAU
Artikelnummer: Cay17687-1
GPR84 is a Galphai protein-coupled receptor that is activated by medium-chain free fatty acids, but only at micromolar concentrations. GPR84 is expressed in leukocytes and its expression is further induced by LPS. 6-OAU is a synthetic agonist for GPR84 (EC50 = 512 nM). It has insignificant actions at a panel of 69...
| Schlagworte: | 6-(octylamino)-2,4(1H,3H)-pyrimidinedione |
| Anwendung: | GPR84 agonist |
| CAS | 83797-69-7 |
| MW: | 239.3 D |
ab 139,00 €
OX04528
Artikelnummer: Cay42377-10
A G protein-biased agonist of GPR84, inhibits forskolin-induced cAMP production in CHO cells expressing human GPR84 (EC50 = 0.00598 nM), does not induce ß-arrestin recruitment at concentrations up to 80 µM. Formulation: A solid. InChI:...
| Schlagworte: | 5-[3-[3,5-bis(trifluoromethyl)phenyl]propyl]-3-pyridinol, 1-oxide |
| Anwendung: | GPR84 G protein-biased agonist |
| CAS | 3028055-45-7 |
| MW: | 365.27 D |
ab 116,00 €
2-hydroxy Lauric Acid
Artikelnummer: Cay24586-25
2-hydroxy Lauric acid is a naturally occuring hydroxylated fatty acid that is found in Acinetobacter species. It acts as a partial agonist of free fatty acid receptor 1 (FFAR1/GPR40) and GPR84 receptors in vitro (EC50s = 6.7 and 12.8 µM, respectively). 2-hydroxy Lauric acid also inhibits bovine hepatic ligase (Ki =...
| Schlagworte: | (±)-2-hydroxy Dodecanoic Acid, (±)-alpha-hydroxy Dodecanoic Acid, (±)-alpha-hydroxy Lauric Acid, NSC 39025,... |
| Anwendung: | Hydroxylated fatty acid, GPR40/GPR84 partial agonist |
| CAS | 2984-55-6 |
| MW: | 216.3 D |
ab 97,00 €
GTPL-5846
Artikelnummer: LKT-G7862.1
GPR84 agonist.
| Schlagworte: | 6-n-octylaminouracil, 6-OAU |
| Anwendung: | GPR84 agonist |
| CAS | 83797-69-7 |
| MW: | 239.32 D |
ab 94,00 €
Anti-GPR84
Artikelnummer: G-PACO40638.50
GPR84 Antibody is a IgG polyclonal antibody from Assay Genie with reactivity against Human and for use in ELISA, IF applications. GPR84 Antibody is a high quality polyclonal antibody for research use only.. Protein function: Receptor for medium-chain free fatty acid (FFA) with carbon chain lengths of C9 to C14....
| Schlagworte: | Anti-EX33, Anti-GPR84, Anti-G-protein coupled receptor 84, Anti-Inflammation-related G-protein coupled receptor EX33 |
| Anwendung: | ELISA, IF |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human |
313,00 €
G-protein coupled receptor 84 (GPR84), partial, human,...
Artikelnummer: CSB-YP865107HU2.1
Organism: Homo sapiens (Human). Source: Yeast. Expression Region: 1-26aa. Protein Length: Partial. Tag Info: C-terminal hFc-tagged. Target Protein Sequence: MWNSSDANFS CYHESVLGYR YVAVSW. Purity: Greater than 85% as determined by SDS-PAGE. Endotoxin: Not test. Biological Activity: n/a. Form: Liquid or Lyophilized...
| Schlagworte: | EX33, GPR84, G-protein coupled receptor 84, Inflammation-related G-protein coupled receptor EX33, Recombinant Human... |
| Anwendung: | Activity not tested |
| Exprimiert in: | Yeast |
| Ursprungsart: | human |
| MW: | 31.2 kD |
ab 347,00 €
Human GPR84 Protein, hFc Tag
Artikelnummer: DIM-PME101470.10
Recombinant human GPR84 Protein with C-terminal human Fc tag. GPR84(Met1-Tyr21) hFc(Glu99-Ala330), Protein function: Receptor for medium-chain free fatty acid (FFA) with carbon chain lengths of C9 to C14. Capric acid (C10:0), undecanoic acid (C11:0) and lauric acid (C12:0) are the most potent agonists. Not activated...
| Schlagworte: | EX33, GPCR4 |
| Exprimiert in: | Human cells |
| Ursprungsart: | human |
| CAS | 12 |
| MW: | 28.7 kD |
ab 139,00 €
GPR84 (human) full length protein-synthetic nanodisc
Artikelnummer: DIM-FLP100129.10
Discover a breakthrough in membrane protein research and drug development with DIMA Biotech's Synthetic Nanodiscs. Traditional methods struggle with challenges in obtaining water-soluble and bioactive forms of multi-transmembrane proteins. Our innovative polymer-based Nanodisc platform offers a game-changing...
| Schlagworte: | EX33, GPR84, G-protein coupled receptor 84, Inflammation-related G-protein coupled receptor EX33, EX33, GPCR4, Human... |
| Anwendung: | Full length transmembrane protein, FA, ELISA, screening, immunization, cell-based assays, crystallization |
| Exprimiert in: | Human cells |
| Ursprungsart: | human |
| MW: | 43.7 kD |
ab 1.317,00 €
6-OAU
Artikelnummer: TGM-T2036-100mg
Description: 6-OAU (GTPL5846)(GTPL5846, 6-n-octylaminouracil) is a surrogate agonist of GPR84, activates human GPR84 in the presence of Gqi5 chimera in HEK293 cells with an EC50 of 105 nM in the PI assay. Target: GPR. Smiles: CCCCCCCCNc1cc(=O)[nH]c(=O)[nH]1. References: Suzuki M, et al. J Biol Chem. 2013 Apr...
| Schlagworte: | GTPL5846 |
| Anwendung: | GPR84 agonist |
| CAS | 83797-69-7 |
| MW: | 239.31 D |
ab 153,00 €
GPR84 Protein, Human, Recombinant (hFc)
Artikelnummer: TGM-TMPH-01410-100ug
Description: Receptor for medium-chain free fatty acid (FFA) with carbon chain lengths of C9 to C14. Capric acid (C10:0), undecanoic acid (C11:0) and lauric acid (C12:0) are the most potent agonists. Not activated by short-chain and long-chain saturated and unsaturated FFAs. Activation by medium-chain free fatty...
| Schlagworte: | Inflammation-related G-protein coupled receptor EX33, G-protein coupled receptor 84, GPR84 |
| MW: | 31.2 kD |
ab 321,00 €