Zu "K04819" wurden 134 Artikel gefunden!
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Anti-5-HT3C / 5-hydroxytryptamine receptor 3C / HTR3C
Artikelnummer: NSJ-RQ8700
0.5mg/ml if reconstituted with 0.2ml sterile DI water. 5-hydroxytryptamine receptor 3C is a protein that in humans is encoded by the HTR3C gene. The product of this gene belongs to the ligand-gated ion channel receptor superfamily. This gene encodes subunit C of the type 3 receptor for 5-hydroxytryptamine...
| Schlagworte: | Anti-HTR3C, Anti-Serotonin receptor 3C, Anti-5-hydroxytryptamine receptor 3C, 5-HT3C Antibody / 5-hydroxytryptamine... |
| Anwendung: | WB, IF, ELISA |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human, mouse, rat |
790,00 €
Anti-HTR3E / 5-hydroxytryptamine receptor 3E
Artikelnummer: NSJ-FY12377
Adding 0.2 ml of distilled water will yield a concentration of 500 ug/ml. The HTR3E antibody targets 5-hydroxytryptamine receptor 3E, a serotonin receptor subunit encoded by the HTR3E gene. This protein belongs to the ligand-gated ion channel family and contributes to the formation of functional 5-HT3 receptor...
| Schlagworte: | Anti-HTR3E, Anti-Serotonin receptor 3E, Anti-5-hydroxytryptamine receptor 3E, HTR3E Antibody / 5-hydroxytryptamine... |
| Anwendung: | WB, IHC, ELISA |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human, mouse, rat |
790,00 €
MDL 72222
Artikelnummer: Cay43507-10
A 5-HT3 receptor antagonist (IC50 = 0.82 nM), selective for 5-HT3 over 5-HT1 and 5-HT2 receptors and alpha1-, alpha2-, and beta-adrenergic receptors (IC50s = >10,000 nM for all), as well as the histamine H1 receptor (IC50 = 3,800 nM), intraplantar administration inhibits formalin-induced paw licking and complete...
| Schlagworte: | Bemesetron, 3,5-dichloro-benzoic acid, (3-endo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl ester |
| Anwendung: | 5-HT3 receptor antagonist |
| CAS | 40796-97-2 |
| MW: | 314.21 D |
ab 83,00 €
Granisetron (hydrochloride)
Artikelnummer: Cay21239-100
Granisetron is an antagonist of the serotonin (5-HT) receptor subtype 5-HT3 (Ki = 3.9 nM) with antiemetic activity. It is selective for 5-HT3 over 5-HT4 receptors (Ki = >1,000 nM). Granisetron (0.3, 1, and 3 mg/kg, p.o.) increases the latency to first vomiting episode and reduces the number of vomiting episodes in a...
| Schlagworte: | BRL 43694, 1-methyl-N-[(3-endo)-9-methyl-9-azabicyclo[3.3.1]non-3-yl]-1H-indazole-3-carboxamide, monohydrochloride |
| Anwendung: | 5-HT3 receptor antagonist |
| CAS | 107007-99-8 |
| MW: | 348.9 D |
ab 85,00 €
Vortioxetine (hydrobromide)
Artikelnummer: Cay23694-5
Vortioxetine is a multimodal serotonergic agent that acts as a serotonin (5-HT, Cay-14332) reuptake inhibitor (Ki = 1.6 nM) and binds to the 5-HT1A, 5-HT1B, 5-HT3A, and 5-HT7 receptors (Kis = 15, 33, 3.7, and 19 nM, respectively). It also binds to the beta1-adrenergic receptor (Ki = 46 nM). It acts as an antagonist...
| Schlagworte: | 1-[2-[(2,4-dimethylphenyl)thio]phenyl]-piperazine, monohydrobromide |
| Anwendung: | Serotonergic agent |
| CAS | 960203-27-4 |
| MW: | 379.4 D |
ab 50,00 €
Alosetron (hydrochloride)
Artikelnummer: Cay22434-25
Alosetron is an antagonist of the serotonin (5-HT) receptor subtype 5-HT3 (Kis = 0.3 and 0.4 nM for the rat cortical and human recombinant receptors, respectively). It is selective for 5-HT3 over 5-HT2 and 5-HT1A receptors (Kis = 6.3 and >100 µM, respectively), as well as alpha1-, beta1-, and beta2- adrenergic, M1,...
| Schlagworte: | GR 68755, 2,3,4,5-tetrahydro-5-methyl-2-[(4-methyl-1H-imidazol-5-yl)methyl]-1H-pyrido[4,3-b]indol-1-one, monohydrochloride |
| Anwendung: | Serotonin 5-HT3 receptor antagonist |
| CAS | 122852-69-1 |
| MW: | 330.8 D |
ab 38,00 €
Ramosetron (hydrochloride)
Artikelnummer: Cay15548-10
Ramosetron is a potent and selective antagonist of the serotonin (5-HT) receptor subtype 5-HT3 (Ki = 0.06 nM). It has little or no effect at other 5-HT receptor subtypes or at adrenergic or histamine receptors. Ramosetron competitively blocks serotonin-mediated contraction of the colon. It has applications in...
| Schlagworte: | (1-methyl-1H-indol-3-yl)[(6R)-4,5,6,7-tetrahydro-1H-benzimidazol-6-yl]-methanone, monohydrochloride |
| Anwendung: | 5-HT3 receptor antagonist |
| CAS | 132907-72-3 |
| MW: | 315.8 D |
ab 102,00 €
Tropisetron (hydrochloride)
Artikelnummer: Cay21240-50
Tropisetron is an antagonist of the serotonin (5-HT) receptor subtype 5-HT3 (Ki = 0.8 nM for the mouse receptor). It is selective for 5-HT3 over the 5-HT4 receptor subtype (Ki = 156 nM for the porcine receptor). Tropisetron is also an antagonist of the alpha9 nicotinic acetylcholine receptor (nAChR, IC50 = 166 nM...
| Schlagworte: | ICS 205-930, SDZ-ICS 930, 1H-indole-3-carboxylic acid (3-endo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl ester, monohydrochloride |
| Anwendung: | 5-HT3 receptor antagonist |
| CAS | 105826-92-4 |
| MW: | 320.8 D |
ab 49,00 €
Ondansetron Hydrochloride Dihydrate
Artikelnummer: LKT-O5212.100
5-HT3 antagonist.
| Schlagworte: | Zofran, Zophren, 1,2,3,9-Tetrahydro-9-methyl-3-[(2-methyl-1H- imidazol-1-yl)methyl]-4H-carbazol-4-one hydrochloride dihydrate |
| Anwendung: | 5-HT3-receptor antagonist |
| CAS | 103639-04-9 |
| MW: | 365.86 D |
ab 204,00 €
Vortioxetine
Artikelnummer: Cay30183-10
Vortioxetine is a multimodal serotonergic agent that acts as a serotonin (5-HT, Cay-14332) reuptake inhibitor (Ki = 1.6 nM) and binds to the 5-HT1A, 5-HT1B, 5-HT3A, and 5-HT7 receptors (Kis = 15, 33, 3.7, and 19 nM, respectively). It also binds to the beta1-adrenergic receptor (Ki = 46 nM). It acts as an antagonist...
| Schlagworte: | 1-[2-[(2,4-dimethylphenyl)thio]phenyl]-piperazine |
| Anwendung: | Serotonin receptor antagonist |
| CAS | 508233-74-7 |
| MW: | 298.4 D |
ab 56,00 €
Granisetron-d3
Artikelnummer: Cay31786-1
Granisetron-d3 is intended for use as an internal standard for the quantification of granisetron (Cay-21239) by GC- or LC-MS. Granisetron is an antagonist of the serotonin (5-HT) receptor subtype 5-HT3 (Ki = 3.9 nM) with antiemetic activity. It is selective for 5-HT3 over 5-HT4 receptors (Ki = >1,000 nM)....
| Schlagworte: | 1-(methyl-d3)-N-[(3-endo)-9-methyl-9-azabicyclo[3.3.1]non-3-yl]-1H-indazole-3-carboxamide |
| Anwendung: | GC-MS, LC-MS, quantification internal standard, 5-HT3 receptor antagonist |
| CAS | 1224925-76-1 |
| MW: | 315.4 D |
480,00 €
Anti-Serotonin receptor 3A / HTR3A, Internal
Artikelnummer: ARG64018.100
Protein function: This is one of the several different receptors for 5- hydroxytryptamine (serotonin), a biogenic hormone that functions as a neurotransmitter, a hormone, and a mitogen. This receptor is a ligand-gated ion channel, which when activated causes fast, depolarizing responses in neurons. It is a...
| Schlagworte: | Anti-HTR3A, Anti-5HT3R, Anti-5-HT3A, Anti-5-HT3R, Anti-5-HT-3, Anti-5-HT3-A, Anti-Serotonin receptor 3A,... |
| Anwendung: | ELISA, WB |
| Wirt: | Goat |
| Spezies-Reaktivität: | human, rat |
871,00 €