Zu "K04277" wurden 357 Artikel gefunden!
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Delta9-THCP-d3 (CRM)
Artikelnummer: Cay44430-100
Delta9-THCP-d3 (CRM) (Cay-44430) is intended for use as an internal standard for the quantification of Delta9-THCP (Cay-33691, Cay-41267, Cay-30171) by GC- or LC-MS. Delta9-THCP is categorized as a phytocannabinoid and has been found in Cannabis. Delta9-THCP-d3 is regulated as a Schedule I compound in the United...
| Schlagworte: | Delta9-Tetrahydrocannabiphorol-d3, Delta9-THC-C7-d3, Delta9-THC-heptyl-d3,... |
| Anwendung: | Certified reference material, GC-MS, LC-MS internal standard, quantification, phytocannabinoid |
| MW: | 345.54 D |
428,00 €
N-Arachidonoyl Dopamine
Artikelnummer: Cay90057-5
N-Arachidonoyl dopamine (NADA) is an arachidonoyl amino acid and cannabinoid (CB) receptor 1 agonist (Ki = 250 nM in rat brain membranes, which highly express CB1 receptors). It is selective for CB1 over CB2 receptors (Ki = 12,000 nM in rat spleen membranes, which highly express CB2 receptors). NADA induces...
| Schlagworte: | NADA, N-[2-(3,4-dihydroxyphenyl)ethyl]-5Z,8Z,11Z,14Z-eicosatetraenamide |
| Anwendung: | CB1 agonist |
| CAS | 199875-69-9 |
| MW: | 439.6 D |
ab 81,00 €
AM251
Artikelnummer: Cay71670-10
AM251 is a cannabinoid 1 (CB1) receptor 1 antagonist. It binds to CB1 receptors in rat forebrain membrane preparations (Ki = 7.5 nM) and is selective over CB2 receptors in mouse spleen preparations (Ki = 2,290 nM) in radioligand binding assays. AM251 inhibits GTPgammaS binding induced by the CB receptor agonist CP...
| Schlagworte: | 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-1-piperidinyl-1H-pyrazole-3-carboxamide |
| Anwendung: | SR 141716A analog |
| CAS | 183232-66-8 |
| MW: | 555.2 D |
ab 83,00 €
CHO-K1/CB1/Galpha15 Stable Cell Line
Artikelnummer: GSC-M00299
The cannabinoid receptor CNR1 is Gs-coupled GPCRs expressed in primarily CNS and some peripheral neurones, particularly prevalent in basal ganglia, hippocampus, cerebellum, cerebral cortex and also presented in some non-neuronal cells and tissues, for example leukocytes and testis. A shorter human splice variant...
| Schlagworte: | CNR1, CANN6, Cannabinoid receptor 1 |
11.424,00 €
ADB-5'F-BUTINACA
Artikelnummer: Cay37761-1
ADB-5'F-BUTINACA (Cay-37761) is an analytical reference standard categorized as a synthetic cannabinoid. This product is intended for research and forensic applications.Formal Name: (S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-1-butyl-5-fluoro-1H-indazole-3-carboxamide. Molecular Formula: C18H25FN4O2. Formula...
| Schlagworte: | ADB-B-5'F-INACA, ADB-BUT-5'F-INACA, (S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-1-butyl-5-fluoro-1H-indazole-3-carboxamide |
| Anwendung: | Analytical reference standard, synthetic cannabinoid |
| MW: | 348.4 D |
ab 122,00 €
Anti-CB1 Receptor (C-Term)
Artikelnummer: Cay10006590-1
The CB1 receptor is a G-protein coupled receptor that binds the active component of cannabis, Delta9-tetrahydrocannabinol. This antibody has been raised against the C-terminal (amino acids 461-472) intracellular region of the human CB1 receptor and can be used for western blotting. Human and rat CB1 receptors...
| Schlagworte: | Anti-CNR, Anti-CB1, Anti-CB1, Anti-CNR1, Anti-CB-R, Anti-CB-R, Anti-CANN6, Anti-CANN6, Anti-Cannabinoid receptor 1,... |
| Anwendung: | IHC, WB |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human |
542,00 €
Anti-CB1 Receptor
Artikelnummer: Cay101500-1
The CB1 receptor and the splice variant CB1a are localized mainly in the brain. The CB1 receptor is a G-protein coupled receptor that binds the active component of cannabis, Delta9-tetrahydrocannabinol. Human and rat CB1 receptors exhibit 97.3% homology at the amino acid level over the complete protein, and 100%...
| Schlagworte: | Anti-CNR, Anti-CB1, Anti-CB1, Anti-CNR1, Anti-CB-R, Anti-CB-R, Anti-CANN6, Anti-CANN6, Anti-Cannabinoid receptor 1,... |
| Anwendung: | WB, IHC |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human, mouse, rat |
468,00 €
Rimonabant
Artikelnummer: Cay9000484-10
Rimonabant is a cannabinoid 1 (CB1) receptor antagonist (Ki = 5.6 nM). It is selective for CB1 over CB2 receptors (Ki = >1,000 nM), as well as a panel of 37 other receptors and channels (IC50s = >1,000 nM). Rimonabant (10 µM) inhibits phytohemagglutinin-induced proliferation of isolated human peripheral blood...
| Schlagworte: | SR141716, 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-1-piperidinyl-1H-pyrazole-3-carboxamide |
| Anwendung: | CB1 receptor inverse agonist |
| CAS | 168273-06-1 |
| MW: | 463.8 D |
ab 40,00 €
9(R)-Hexahydrocannabinol (CRM)
Artikelnummer: Cay37913-1
9(R)-Hexahydrocannabinol (CRM) (Cay-37913) is a certified reference material that is structurally similar to known phytocannabinoids. 9(R)-Hexahydrocannabinol induces immobility, severe stupor, ataxia, full ptosis, and crouched posture, markers of psychotropic activity, in rhesus monkeys. This product is intended...
| Schlagworte: | 9beta-HHC, 11beta-Hexahydrocannabinol, trans-(6aR,9R,10aR)-HHC, 11beta-HHC, 9(R)-HHC, 9beta-Hexahydrocannabinol,... |
| Anwendung: | Certified reference material, phytocannabinoid |
| CAS | 36403-90-4 |
| MW: | 316.5 D |
475,00 €
R-1 Methanandamide
Artikelnummer: Cay90070-5
R-1 methanandamide is a potent cannabinoid (CB) receptor 1 agonist in the methanandamide series. It is selective for CB1 over CB2 receptors with Ki values ranging from 17.9 to 28.3 and 815 to 868 nM, respectively.{7912, 10685} R-1 methanandamide is more potent than arachidonoyl ethanolamide (AEA, Cay-90050). In...
| Schlagworte: | (R)-(+)-Arachidonyl-1'-Hydroxy-2'-Propylamide, AM356, N-(2-hydroxy-1R-methylethyl)-5Z,8Z,11Z,14Z-eicosatetraenamide |
| Anwendung: | CB1 receptor agonist |
| CAS | 157182-49-5 |
| MW: | 361.6 D |
ab 77,00 €
2-Linoleoyl Glycerol
Artikelnummer: Cay62260-1
2-Arachidonoyl glycerol (2-AG) has been isolated from porcine brain, and has been characterized as the natural endocannabinoid ligand for the CB1 receptor. The congener of 2-AG in which a linoleoyl group replaces the arachidonoyl group is 2-linoleoyl glycerol (2-LG), and this compound also appears in vivo in...
| Schlagworte: | 2-LG, 9Z,12Z-octadecadienoic acid, 2-glyceryl ester |
| Anwendung: | CB1 receptor ligand |
| CAS | 3443-82-1 |
| MW: | 354.5 D |
ab 25,00 €
JD5037
Artikelnummer: Cay12053-1
JD5037 is an inverse agonist of peripheral cannabinoid 1 (CB1) receptors (Ki = 0.35 nM). It displays >700-fold selectivity for CB1 over CB2, >1,000-fold selectivity over a panel of 70 receptors, transporters, and ion channels, and low blood-brain barrier penetrance. JD5037 is orally bioavailable and reduces food...
| Schlagworte: | 2S-[[[(4S)-3-(4-chlorophenyl)-4,5-dihydro-4-phenyl-1H-pyrazol-1-yl][[(4-chlorophenyl)sulfonyl]amino]methylene]amino]-3-met... |
| Anwendung: | CB1 receptor inverse agonist |
| CAS | 1392116-14-1 |
| MW: | 572.5 D |
ab 38,00 €