Zu "K04268" wurden 33 Artikel gefunden!

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5'-Deoxy-5'-methylthioadenosine
5'-Deoxy-5'-methylthioadenosine

Artikelnummer: Cay15593-50

5'-Deoxy-5'-methylthioadenosine (MTA) is an intermediate in the generation of adenine and methionine that is produced by the decarboxylation of S-adenosylmethionine. This nucleoside is a potent agonist of adenosine receptors (Kis = 0.15, 1.13, 13.9, and 0.68 µM for A1, A2A, A2B, and A3, respectively). At higher...
Schlagworte: 5'-S-Methylthioadenosine, MTA, NSC 335422, Vitamin L2, 5'-S-methyl-5'-thio-adenosine
Anwendung: Intermediate, Adenosine receptor agonist
CAS 2457-80-9
MW: 297.3 D
ab 42,00 €
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MRS1523
MRS1523

Artikelnummer: Cay17128-1

MRS1523 is a selective adenosine A3 receptor antagonist (Kis = 18.9 and 113 nM for human and rat A3 receptors, respectively, versus Kis = 15.6 and 2.05 µM for rat A1 and A2A receptors, respectively). As activation of the A3 receptor is linked to several second messenger systems for signaling pathways involving...
Schlagworte: 6-ethyl-5-[(ethylthio)carbonyl]-2-phenyl-4-propyl-3-pyridinecarboxylic acid propyl ester
Anwendung: Adenosine A3 receptor agonist
CAS 212329-37-8
MW: 399.5 D
ab 55,00 €
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CGS 15943
CGS 15943

Artikelnummer: Cay22073-5

CGS 15943 is an orally bioavailable non-xanthine antagonist at adenosine (A) receptors with IC50 values of 3.5, 4.2, 16, and 51 nM in CHO cells transfected with human recombinant A1, A2A, A2B, and A3 receptors, respectively. It also binds to the phosphatidylinositol 3-kinase (PI3K) catalytic subunit p110gamma, and...
Schlagworte: CGS 15943A, 9-chloro-2-(2-furanyl)-[1,2,4]triazolo[1,5-c]quinazolin-5-amine
Anwendung: Adenosine receptor antagonist
CAS 104615-18-1
MW: 285.7 D
ab 33,00 €
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HEMADO
HEMADO

Artikelnummer: Cay21015-5

HEMADO is a selective agonist of the adenosine A3 receptor (Kis = 1.1, 327, and 1,230 nM for A3, A1, and A2A receptors, respectively). HEMADO reduces release of lactate dehydrogenase (LDH) and creatine kinase-MB (CK-MB) from myocardium in isolated rat hearts subjected to ischemia-reperfusion injury. Formal Name:...
Schlagworte: 2-(1-hexyn-1-yl)-N-methyl-adenosine
Anwendung: High affinity and selective adenosine A3 receptor agonist
CAS 403842-38-6
MW: 361.4 D
ab 32,00 €
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2-Cl-IB-MECA
2-Cl-IB-MECA

Artikelnummer: Cay27336-25

2-Cl-IB-MECA is an adenosine A3 receptor agonist. It binds selectively to adenosine A3 receptors (Ki = 0.33 nM) over A1 and A2A receptors (Kis = 820 and 470 nM, respectively) and inhibits adenylate cyclase activity with an IC50 value of 66.8 nM in CHO cell membranes expressing rat A3 receptors. 2-Cl-IB-MECA (10 and...
Schlagworte: 2-Chloro-IB-MECA, CF 102, Namodenoson,...
Anwendung: Adenosine receptor A3 agonist
CAS 163042-96-4
MW: 544.7 D
ab 112,00 €
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VUF 5574
VUF 5574

Artikelnummer: Cay27676-5

VUF 5574 is an antagonist of the adenosine A3 receptor (Ki = 4.03 nM for the recombinant human receptor). It is greater than 2,500-fold selective for adenosine A3 over A1 and A2A receptors. VUF 5574 (100 nM) decreases phosphorylation of ERK1/2 induced by adenosine (Cay-21232) in isolated porcine coronary artery...
Schlagworte: N-(2-methoxyphenyl)-N'-[2-(3-pyridinyl)-4-quinazolinyl]-urea
Anwendung: Adenosine A3 receptor antagonist
CAS 280570-45-8
MW: 371.4 D
ab 32,00 €
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Anti-ADORA3
Anti-ADORA3

Artikelnummer: ABD-8G204.50

Custom conjugation services for this antibody as available (eg. labeling of Anti-ADORA3 with HRP. Available labels are AF: AF350, AF488, AF555, AF594, AF647, AF680, AF700, AF750. Proteins: HRP, Alkaline Phosphatase, Streptavidin. Tandems: APC, APC/Cy7, APC/AF750, APC/iFluor(TM) 700, APC/iFluor(TM) 750, PE, PE/Cy5,...
Schlagworte: Anti-Transmembrane domain-containing protein TMIGD3, ADORA3 Antibody
Anwendung: IF, ELISA
Reaktivität: Human, Mouse
230,00 €
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Anti-ADORA3
Anti-ADORA3

Artikelnummer: ABD-8G021.50

Custom conjugation services for this antibody as available (eg. labeling of Anti-ADORA3 with HRP. Available labels are AF: AF350, AF488, AF555, AF594, AF647, AF680, AF700, AF750. Proteins: HRP, Alkaline Phosphatase, Streptavidin. Tandems: APC, APC/Cy7, APC/AF750, APC/iFluor(TM) 700, APC/iFluor(TM) 750, PE, PE/Cy5,...
Schlagworte: Anti-Transmembrane domain-containing protein TMIGD3, ADORA3 Antibody
Anwendung: IF, ELISA
Reaktivität: Human, Mouse
230,00 €
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Rat Adenosine A3 Receptor / ADORA3 ELISA Kit
Rat Adenosine A3 Receptor / ADORA3 ELISA Kit

Artikelnummer: G-RTFI00555.96

Anwendung: ELISA
Reaktivität: Rat
629,00 €
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Human ADORA3 (Adenosine A3 Receptor) ELISA Kit
Human ADORA3 (Adenosine A3 Receptor) ELISA Kit

Artikelnummer: E-EL-H5633.96

The kit is a Sandwich enzyme immunoassay for in vitro quantitative measurement of ADORA3 in serum, plasma and other biological fluids. Detection Range: 0.63--40ng/mL. Sensitivity: 0.38ng/mL. Protein function: Isoform 2: Receptor for adenosine. The activity of this receptor is mediated by G proteins which inhibits...
Schlagworte: Adenosine receptor A3
Anwendung: ELISA
Reaktivität: Human
554,00 €
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Rat ADORA3 (Adenosine A3 Receptor) ELISA Kit
Rat ADORA3 (Adenosine A3 Receptor) ELISA Kit

Artikelnummer: E-EL-R2510.96

The kit is a Sandwich enzyme immunoassay for in vitro quantitative measurement of ADORA3 in serum, plasma and other biological fluids. Detection Range: 0.31--20ng/mL. Sensitivity: 0.19ng/mL. Protein function: Receptor for adenosine. The activity of this receptor is mediated by G proteins which inhibits adenylyl...
Schlagworte: TGPCR1, Adora3, Adenosine receptor A3
Anwendung: ELISA
Reaktivität: Rat
554,00 €
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2-Cl-IB-MECA
2-Cl-IB-MECA

Artikelnummer: 159522.5

2-Cl-IB-MECA acts as an A3 adenosine receptor-selective nucleoside. Solubility: >20 mg/ml in DMSO.
Schlagworte: 1-[2-Chloro-6-[[(3-iodophenyl)methyl]amino]-9H-purin-9-yl]-1-deoxy-N-methyl- -D-ribofuranuronamide,...
Anwendung: ADORA3 agonist
CAS 163042-96-4
MW: 544.73 D
472,00 €
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