Zu "K04266" wurden 99 Artikel gefunden!
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Regadenoson hydrate
Artikelnummer: TGM-T26054-100mg
Description: Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing. Target: Others. Smiles: NC1=C2C(N(C=N2)[C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)=NC(=N1)N4C=C(C(NC)=O)C=N4.O. References: Johnson NP, Gould KL. Regadenoson versus dipyridamole hyperemia for...
| Schlagworte: | CVT 3146, Lexiscan, CVT-3146, CVT3146, Regadenoson |
| Anwendung: | Targets adenosine receptor A2a (ADORA2A, ADOR) |
| CAS | 875148-45-1 |
| MW: | 408.37 D |
ab 1.520,00 €
CGS 21680 Hydrochloride
Artikelnummer: TGM-T6441-100mg
Description: CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor. Target: Adenosine Receptor. Smiles: Cl.CCNC(=O)[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)nc(NCCc3ccc(CCC(O)=O)cc3)nc12. References: Hutchison AJ, et al. J...
| Schlagworte: | CGS 21680 HCl |
| Anwendung: | Adenosine A2A receptor agonist |
| CAS | 124431-80-7 |
| MW: | 535.98 D |
ab 34,00 €
Istradefylline
Artikelnummer: TGM-T6552-100mg
Description: Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails. It has been used in trials studying the treatment and basic science of Drug Abuse, Sleep Disorder, Hepatic Impairment, Parkinson's Disease, and Restless Legs...
| Schlagworte: | KW-6002 |
| Anwendung: | Targets adenosine receptor A2a (ADORA2A, ADOR) |
| CAS | 155270-99-8 |
| MW: | 384.43 D |
ab 37,00 €
Sonedenoson
Artikelnummer: TGM-T34685-100mg
Description: Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2,-O-ribose methyltransferase, and may be used in the study of diabetic foot ulcers. Target: Adenosine Receptor, SARS-CoV. Smiles:...
| Schlagworte: | MRE 0094, MRE0094, MRE-0094 |
| Anwendung: | Targets adenosine receptor A2a (ADORA2A, ADOR) |
| CAS | 131865-88-8 |
| MW: | 421.84 D |
ab 292,00 €
ST-1535
Artikelnummer: TGM-T28861-100mg
Description: ST 1535 is a potent and orally active antagonist of the A2A adenosine receptor, exhibiting antiparkinsonian activity and antitremorigenic effects, with potential for Parkinson's disease research. Target: Adenosine Receptor. Smiles: CCCCc1nc(N)c2nc(-n3nccn3)n(C)c2n1. References: Maria Antonietta Stasi,...
| Anwendung: | Adenosine A2A receptor antagonist |
| CAS | 496955-42-1 |
| MW: | 272.31 D |
ab 40,00 €
Evodenoson
Artikelnummer: TGM-T31731-100mg
Description: Evodenoson (ATL313) is a potent and selective adenosine A2a receptor (A2aR) agonist for the treatment of eye diseases, tumors, and immune system disorders, and may be used in studies of open-angle glaucoma and blood tumors. Target: Adenosine Receptor. Smiles:...
| Schlagworte: | ATL313, DE112, ATL-313, ATL 313, DE 112, DE-112 |
| Anwendung: | Targets adenosine receptor A2a (ADORA2A, ADOR) |
| CAS | 844873-47-8 |
| MW: | 499.52 D |
ab 248,00 €
Apadenoson
Artikelnummer: TGM-T26641-25mg
Description: Apadenoson is a potent Adenosine A2 receptor agonist with inhibitory effects on Adenosine A3 receptors with an IC of 45 nM. Apadenoson has anti-inflammatory activity and can be used to study neurological diseases. Target: Others. Smiles:...
| Schlagworte: | BMS-068645, BMS068645, ATL-146e, ATL146e, BMS 068645, ATL 146e |
| Anwendung: | Targets adenosine receptor A2a (ADORA2A, ADOR) |
| CAS | 250386-15-3 |
| MW: | 486.52 D |
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Inupadenant
Artikelnummer: TGM-T37014-25mg
Description: Inupadenant is an orally active, highly selective A2A receptor antagonist with potent anti-tumor activity [1] and is not brain-penetrant. Target: Others. Smiles: CS(=O)CCOc1cc(N2CCN(CCn3c4nc(N)n5nc(nc5c4sc3=O)-c3ccco3)CC2)c(F)cc1F. References: Laurence Buisseret, et al. Phase 1 trial of the adenosine...
| Anwendung: | Targets adenosine receptor A2a (ADORA2A, ADOR) |
| CAS | 2246607-08-7 |
| MW: | 604.65 D |
2.573,00 €
AZD4635
Artikelnummer: TGM-T4265-100mg
Description: AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM). Target: Adenosine Receptor. Smiles: Cc1cc(cc(Cl)n1)-c1nnc(N)nc1-c1ccc(F)cc1. References: Alexandra Borodovsky, et al. Abstract 5580: PreClinicalal pharmacodynamics and antitumor activity of AZD4635, a novel adenosine 2A...
| Schlagworte: | HTL1071 |
| Anwendung: | Adenosine 2A receptor (A2AR) antagonist |
| CAS | 1321514-06-0 |
| MW: | 315.73 D |
ab 31,00 €
Preladenant
Artikelnummer: TGM-T4290-100mg
Description: Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine receptors. Target: Adenosine Receptor. Smiles: COCCOc1ccc(cc1)N1CCN(CCn2ncc3c2nc(N)n2nc(nc32)-c2ccco2)CC1. References: Hodgson RA, et al....
| Schlagworte: | SCH-420814 |
| Anwendung: | Targets adenosine receptor A2a (ADORA2A, ADOR) |
| CAS | 377727-87-2 |
| MW: | 503.56 D |
ab 31,00 €
Adenosine receptor inhibitor 1
Artikelnummer: TGM-T61850-100mg
Description: Adenosine receptor inhibitor 1 is a highly potent and selective antagonist of adenosine receptor (AR), exhibiting exceptional affinity for A1 AR, A2A AR, A2B AR, and A3 AR, with respective Ki values of >1000, 68.5, >1000, >1000 nM. This compound demonstrates notable antinociceptive, anti-inflammatory,...
| Anwendung: | Adenosine receptor inhibitor |
| CAS | 2550400-52-5 |
| MW: | 395.82 D |
ab 1.520,00 €
SCH 58261
Artikelnummer: TGM-T6979-100mg
Description: SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a. Target: Adenosine Receptor. Smiles: Nc1nc2n(CCc3ccccc3)ncc2c2nc(nn12)-c1ccco1. References: Zocchi C, et al. J Pharmacol Exp Ther. 1996, 276(2), 398-404.
| Schlagworte: | SCH58261 |
| Anwendung: | Adenosine A2A-Receptor antagonist |
| CAS | 160098-96-4 |
| MW: | 345.36 D |
ab 34,00 €