Zu "K04265" wurden 94 Artikel gefunden!
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5'-Methylthioadenosine
Artikelnummer: TGM-T8227-25mg
Description: 4-Methyl-2-oxopentanoic acid is an abnormal metabolite, a neurotoxin and a metabolic toxin. Target: Endogenous Metabolite. Smiles: CSC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12. References: Avila MA, et al. Methylthioadenosine. Int J Biochem Cell Biol. 2004 Nov,36(11):2125-30.
| Schlagworte: | 5'-S-Methyl-5'-thioadenosine, 5'-Deoxy-5'-(methylthio)adenosine, Methylthioadenosine, 5'-(Methylthio)-5'-deoxyadenosine |
| Anwendung: | Intermediate, adenosine receptor agonist |
| CAS | 2457-80-9 |
| MW: | 297.33 D |
ab 40,00 €
2-Chloroadenosine
Artikelnummer: TGM-T7736-100mg
Description: 2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, and A3 receptors( Ki:300, 80, and 1,900 nM, respectively). Target: Adenosine Receptor. Smiles: NC1=C2N=CN(C3OC(CO)C(O)C3O)C2=NC(Cl)=N1. References: Ates N , Ilbay G , Sahin D . Suppression of...
| Anwendung: | Adenosine A1/A2A/A3 receptor agonist |
| CAS | 146-77-0 |
| MW: | 301.69 D |
ab 31,00 €
Adenosine amine congener
Artikelnummer: TGM-T7683-100mg
Description: Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,. Target: Adenosine Receptor. Smiles: NCCNC(=O)Cc1ccc(NC(=O)Cc2ccc(Nc3ncnc4n(cnc34)[C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)cc2)cc1. References: Vlajkovic S M , Lee K H , Wong A C Y , et al. Adenosine amine congener...
| Schlagworte: | ADAC |
| Anwendung: | Adenosine A1 receptor agonist |
| CAS | 96760-69-9 |
| MW: | 576.6 D |
ab 67,00 €
MIPS521
Artikelnummer: TGM-T9330-100mg
Description: MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R. Target: Adenosine Receptor. Smiles: Nc1scc(c1C(=O)c1ccc(Cl)cc1)-c1cc(cc(c1)C(F)(F)F)C(F)(F)F. References: receptor-mediated analgesia[J]. Nature.
| Schlagworte: | {2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone |
| Anwendung: | Adenosine A1 receptor positive allosteric modulator |
| CAS | 1146188-19-3 |
| MW: | 449.8 D |
ab 33,00 €
A1AR Protein, Human, Recombinant (His)
Artikelnummer: TGM-TMPH-00892-100ug
Description: Receptor for adenosine. The activity of this receptor is mediated by G proteins which inhibit adenylyl cyclase. A1AR Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 39.3 kDa and the accession number is P30542.
| Schlagworte: | ADORA1, Adenosine receptor A1 |
| MW: | 39.3 kD |
ab 1.941,00 €
5'-Deoxy-5'-methylthioadenosine-d3
Artikelnummer: TGM-TMID-0168-1mg
Description: 5'-Deoxy-5'-methylthioadenosine-d3 is a deuterated compound of 5'-Deoxy-5'-methylthioadenosine. 5'-Deoxy-5'-methylthioadenosine has a CAS number of 2457-80-9. 5'-Methylthioadenosine is produced from S-adenosylmethionine and behaves as a powful inhibitory product. Smiles:...
| Anwendung: | GC-MS, LC-MS, internal standard, quantification |
| CAS | 174838-38-1 |
| MW: | 300.35 D |
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GR79236
Artikelnummer: TGM-TQ0136-2mg
Description: GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions. Target: Adenosine Receptor. Smiles: OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N[C@H]3CCC[C@@H]3O)ncnc12. References: Sneyd JR, et al. Multicentre evaluation of the adenosine...
| Schlagworte: | GR 79236 |
| Anwendung: | Selective adenosine receptor A1 agonist |
| CAS | 124555-18-6 |
| MW: | 351.36 D |
49,00 €
CV1808
Artikelnummer: TGM-T19696-10mg
Description: CV-1808 is a coronary vasodilator, antihypertensive, and antipsychotic following systemic administration in vivo. CV-1808 is an adenosine A2 receptor agonist. Target: Others. Smiles: [H][C@]1(O[C@H](CO)[C@@H](O)[C@H]1O)n1cnc2c(N)nc(Nc3ccccc3)nc12. References: Cornfield LJ, Hu S, Hurt SD, Sills MA....
| Schlagworte: | CV-1808, CV 1808 |
| Anwendung: | Adenosine receptor agonist. |
| CAS | 53296-10-9 |
| MW: | 358.35 D |
ab 112,00 €
N6-Cyclopentyladenosine
Artikelnummer: TGM-T16263-100mg
Description: N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor, mimicking its action with Ki values of 2.3 nM, 790 nM, and 43 nM for human A1, A2A, and A3 receptors, respectively. CPA is used to modulate cellular signaling, neurotransmission, and other biological processes. Target:...
| Schlagworte: | CPA, UK-80882 |
| Anwendung: | Adenosine 1 receptor agonist |
| CAS | 41552-82-3 |
| MW: | 335.36 D |
ab 31,00 €
Rolofylline
Artikelnummer: TGM-T16782-100mg
Description: Rolofylline (KW-3902) is a selective adenosine A1 receptor antagonist utilized in research on acute congestive heart failure, renal dysfunction, and neurodegenerative disorders. Target: Adenosine Receptor. Smiles: CCCn1c2[nH]c(nc2c(=O)n(CCC)c1=O)C12CC3CC1CC(C2)C3. References: Slawsky MT, et al....
| Schlagworte: | MK-7418, KF-15372, KW-3902 |
| Anwendung: | Targets adenosine receptor A1 (ADORA1) |
| CAS | 136199-02-5 |
| MW: | 356.46 D |
ab 40,00 €
Tecadenoson
Artikelnummer: TGM-T17023-100mg
Description: Tecadenoson (CVT-510) is a selective A1 adenosine receptor agonist. Target: Adenosine Receptor. Smiles: OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N[C@@H]3CCOC3)ncnc12. References: Snowdy S, et al. A comparison of an A1 adenosine receptor agonist (CVT-510) with diltiazem for slowing of AVnodal conduction...
| Schlagworte: | CVT-510 |
| Anwendung: | Targets adenosine receptor A1 (ADORA1) |
| CAS | 204512-90-3 |
| MW: | 337.33 D |
ab 46,00 €
Tonapofylline
Artikelnummer: TGM-T17117-100mg
Description: Tonapofylline is an orally active and selective antagonist of the A1 adenosine receptor (Ki: 7.4 nM for human A1). Tonapofylline can be used in studies about heart failure. Target: Adenosine Receptor. Smiles: CCCn1c2nc([nH]c2c(=O)n(CCC)c1=O)C12CCC(CCC(O)=O)(CC1)CC2. References: Kiesman WF, et al. Potent...
| Schlagworte: | BG 9928 |
| Anwendung: | Targets adenosine receptor A1 (ADORA1) |
| CAS | 340021-17-2 |
| MW: | 416.51 D |
ab 37,00 €