Zu "K04215" wurden 372 Artikel gefunden!
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CHO-K1/OPRM1/Galpha15 Stable Cell Line
Artikelnummer: GSC-M00304
Recombinant CHO-K1 cells stably overexpress human opioid receptor mu 1 (OPRM1) on the surface and contain high levels of G protein Galphai and Galphaq to couple with the receptor in downstream signaling pathways.
| Schlagworte: | OPRM1, Mu opiate receptor, Mu opioid receptor, Mu-type opioid receptor |
11.424,00 €
Fentanyl-KLH conjugate
Artikelnummer: ABD-50567
Small compounds (drugs or peptides) are not sufficiently complex by themselves to induce an immune response or be processed in a manner that elicits production of specific antibodies. For antibody production to be successful with small antigens, they must be chemically conjugated with immunogenic carrier proteins...
| Anwendung: | Antigen |
658,00 €
SR 17018
Artikelnummer: Cay24480-5
SR 17018 is an orally bioavailable and brain-penetrant agonist of µ-opioid receptors. It is functionally selective for G protein-coupled receptor signaling (EC50 = 97 nM for GTPgammaS binding in CHO cells expressing µ-opioid receptors) over beta-arrestin 2 recruitment (EC50 = >10,000 nM) at the µ-opioid receptor. SR...
| Schlagworte: | 5,6-dichloro-1-[1-[(4-chlorophenyl)methyl]-4-piperidinyl]-1,3-dihydro-2H-benzimidazol-2-one |
| Anwendung: | µ-opioid receptor agonist |
| CAS | 2134602-45-0 |
| MW: | 410.7 D |
ab 73,00 €
Nalmefene (hydrochloride)
Artikelnummer: Cay28266-10
A µ- and kappa-opioid receptor antagonist (Kis = 0.91 and 1.03 nM, respectively, in CHO membranes expressing the human receptors), selective for µ- and kappa-opioid receptors over delta-opioid receptors (Ki = 13.26 nM in CHO membranes expressing the human receptors), decreases self-administration of alcohol in...
| Schlagworte: | NIH 10365, (5a)-17-(cyclopropylmethyl)-4,5-epoxy-6-methylene-morphinan-3,14-diol, monohydrochloride |
| Anwendung: | µ/kappa-opioid receptor antagonist |
| CAS | 58895-64-0 |
| MW: | 375.9 D |
ab 38,00 €
O-Desmethyl-cis-tramadol-d6 (hydrochloride) (CRM)
Artikelnummer: Cay42181-100
An internal standard for the quantification of O-desmethyl-cis-tramadol by GC- or LC-MS, intended for research and forensic applications. Formulation: A 100 µg/ml solution in methanol. InChI:...
| Schlagworte: | O-Desmethyltramadol-d6, ODMT-d6, 3-((1R,2R)-2-((bis(methyl-d3)amino)methyl)-1-hydroxycyclohexyl)phenol, monohydrochloride |
| Anwendung: | Certified reference material, GC-MS, LC-MS, internal standard, quantification, opioid |
| CAS | 1261393-87-6 |
| MW: | 291.85 D |
340,00 €
Loperamide hydrochloride
Artikelnummer: LKT-L5660.5
A mu-opioid agonist that is an antidiarrhoeal drug which inhibits intestinal motility and secretion. It has been shown to suppress the calcium-influx in dorsal root ganglion neurons.
| Anwendung: | mu-opioid agonist |
| CAS | 34552-83-5 |
| MW: | 513,51 D |
ab 128,00 €
meta-Methylfentanyl-d5 (hydrochloride)
Artikelnummer: Cay42416-1
meta-Methylfentanyl-d5 (hydrochloride) (Cay-42416) is intended for use as an internal standard for the quantification of meta-Methylfentanyl (Cay-22633, Cay-36371) by GC- or LC-MS. meta-Methylfentanyl is an analytical reference standard categorized as an opioid. meta-Methylfentanyl-d5 is regulated as a Schedule I...
| Schlagworte: | m-Methylfentanyl-d5, N-(3-methylphenyl)-N-[1-(2-(phenyl-d5)ethyl)-4-piperidinyl]-propanamide, monohydrochloride |
| Anwendung: | Analytical reference standard, GC-MS, LC-MS, internal standard, quantification, opioid |
| MW: | 391.99 D |
ab 221,00 €
meta-Fluorofentanyl-d5 (hydrochloride)
Artikelnummer: Cay42429-1
meta-Fluorofentanyl-d5 (hydrochloride) (Cay-42429) is intended for use as an internal standard for the quantification of meta-fluorofentanyl (Cay-19424, Cay-38142) by GC- or LC-MS. meta-Fluorofentanyl is categorized as an opioid. meta-Fluorofentanyl-d5 is regulated as a Schedule I compound in the United States. This...
| Schlagworte: | m-FF-d5, m-Fluorofentanyl-d5, N-(3-fluorophenyl)-N-[1-(2-phenylethyl-d5)-4-piperidinyl]-propanamide, monohydrochloride |
| Anwendung: | Analytical reference standard, internal standard, quantification, opioid |
| MW: | 395.95 D |
ab 221,00 €
3,4-MDiPA (hydrochloride)
Artikelnummer: Cay42415-1
3,4-MDiPA (hydrochloride) (Cay-42415) is an analytical reference standard categorized as an amphetamine. 3,4-MDiPA has analgesic activity in mice. This product is intended for research and forensic applications.. Solulibility: PBS (pH 7.2): Sparingly soluble: 1-10 mg/ml: .
| Schlagworte: | 3,4-MDiPr, 3,4-Methylenedioxy-N-isopropylamphetamine, N-isopropyl MDA,... |
| Anwendung: | Analytical reference standard, amphetamine |
| CAS | 74341-76-7 |
| MW: | 257.76 D |
ab 122,00 €
para-Methylfentanyl-d5 (hydrochloride)
Artikelnummer: Cay42417-1
para-Methylfentanyl-d5 (hydrochloride) (Cay-42417) is intended for use as an internal standard for the quantification of para-methylfentanyl (Cay-41384, Cay-20038) by GC- or LC-MS. para-Methylfentanyl is categorized as an opioid. It has antinociceptive activity. para-Methylfentanyl is regulated as a Schedule I...
| Schlagworte: | p-Methylfentanyl-d5, N-(4-methylphenyl)-N-[1-(2-(phenyl-d5)ethyl)-4-piperidinyl]-propanamide, monohydrochloride |
| Anwendung: | Analytical reference standard, internal standard, quantification, opioid |
| MW: | 391.99 D |
ab 221,00 €
Naloxonazine (hydrochloride)
Artikelnummer: Cay21950-50
Naloxonazine is a µ-opioid receptor antagonist (Ki = 0.054 nM in a radioligand binding assay). It is selective for µ-opioid over kappa- and delta-opioid receptors (Kis = 11 and 8.6 nM, respectively, in radioligand binding assays) and selectively binds to high-affinity µ1-opioid over µ- and delta-opioid receptors...
| Schlagworte: | NLXZ, (5alpha)-[(5alpha)-4,5-epoxy-3,14-dihydroxy-17-(2-propenyl)morphinan-6-ylidene]hydrazone,... |
| Anwendung: | µ-opioid receptor (OPRM1) antagonist |
| CAS | 880759-65-9 |
| MW: | 723.7 D |
ab 110,00 €
DAMGO (trifluoroacetate salt)
Artikelnummer: Cay21553-5
DAMGO is a selective peptide agonist of the µ-opioid receptor (Kis = 1.18, 1,430, and 213 nM for human µ-, delta-, and kappa-opioid receptors, respectively). DAMGO displays higher efficacy than morphine (Cay-ISO60147) for µ-opioid-induced nociception in rats.Formal Name:...
| Schlagworte: | [D-Ala2, N-Me-Phe4, Gly5-ol]-Enkephalin, DAGO, NIH 10891, RX-783006,... |
| Anwendung: | µ-opioid receptor agonist |
| MW: | 513.6 D |
ab 75,00 €