Zu "K04207" wurden 35 Artikel gefunden!
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Lu AA33810
Artikelnummer: Cay32913-1
Lu AA33810 is an antagonist of neuropeptide Y (NPY) receptor Y5 (Ki = 1. nM for the human receptor). It is selective for Y5 over Y1, Y2, and Y4 (Kis = >10 µM for all in HEK293 membranes expressing rat receptors). Lu AA33810 also binds the serotonin (5-HT) receptor subtypes 5-HT1A and 5-HT2B (Kis = 478 and 247 nM,...
| Schlagworte: | N-[[trans-4-[(4,5-dihydro[1]benzothiepino[5,4-d]thiazol-2-yl)amino]cyclohexyl]methyl]-methanesulfonamide |
| Anwendung: | NPY receptor Y5 antagonist |
| CAS | 304008-29-5 |
| MW: | 423.62 D |
75,00 €
Anti-NPY5R Biotin Conjugate
Artikelnummer: NSJ-R34109BTN
0.5 mg/ml in 1X TBS, pH7.3, with 0.5% BSA (US sourced) and 0.02% sodium azide. Additional name(s) for this target protein: Neuropeptide Y receptor Y5
| Schlagworte: | Anti-NPY5R, Anti-NPY-Y5 receptor, Anti-Neuropeptide Y receptor type 5, NPY5R Antibody Biotin Conjugate |
| Anwendung: | WB, IHC, ELISA (peptide) |
| Wirt: | Goat |
| Spezies-Reaktivität: | human |
836,00 €
L-152,804
Artikelnummer: Cay42504-10
L-152,804 is an antagonist of neuropeptide Y (NPY) receptor Y5 (IC50s = 26 and 31 nM for the human and rat receptors, respectively). It is selective for Y5 over Y1, Y2, and Y4 receptors (IC50s = >10,000 nM for the human receptors). L-152,804 (30 µg, i.c.v.) reduces bovine pancreatic peptide-induced, but not...
| Schlagworte: | 5,5-dimethyl-2-(2,3,4,9-tetrahydro-3,3-dimethyl-1-oxo-1H-xanthen-9-yl)-1,3-cyclohexanedione |
| Anwendung: | NPY receptor Y5 (NPY5R) antagonist |
| CAS | 6508-43-6 |
| MW: | 366.45 D |
ab 118,00 €
NTNCB (hydrochloride)
Artikelnummer: Cay43216-1
NTNCB is an antagonist of neuropeptide Y (NPY) receptor Y5 (Ki = 8 nM). It is selective for neuropeptide Y5 over Y1 receptors (Ki = >10,000 nM). NTNCB (10 and 20 µM) suppresses colony formation by PC3 and DU145 prostate cancer cells. In vivo, NTNCB (1, 3, and 10 mg/kg per day) reduces tumor volume in a PC3 mouse...
| Schlagworte: | 2-nitro-N-[[trans-4-[[[(1,2,3,4-tetrahydro-2-naphthalenyl)methyl]amino]methyl]cyclohexyl]methyl]-benzenesulfonamide,... |
| Anwendung: | NPY receptor Y5 antagonist |
| CAS | 191931-56-3 |
| MW: | 508.07 D |
ab 44,00 €
MK-0557
Artikelnummer: Cay22134-1
MK-0557 is a potent antagonist of the neuropeptide Y (NPY) receptor Y5 (Kis = 1.3, 0.79, 0.74, and 1.4 nM for human, rhesus monkey, mouse, and rat receptors, respectively). It is >7,500-fold selective for Y5 over other receptors and lacks activity in a panel of 180 receptors, enzymes, and ion channels at...
| Schlagworte: | trans-N-[1-(2-fluorophenyl)-1H-pyrazol-3-yl]-1'-oxo-spiro[cyclohexane-1,3'(1'H)-furo[3,4-c]pyridine]-4-carboxamide |
| Anwendung: | NPY5R antagonist |
| CAS | 328232-95-7 |
| MW: | 406.4 D |
ab 56,00 €
Anti-Neuropeptide Y receptor Y5, Internal
Artikelnummer: ARG63772.100
Protein function: Receptor for neuropeptide Y and peptide YY. The activity of this receptor is mediated by G proteins that inhibit adenylate cyclase activity. Seems to be associated with food intake. Could be involved in feeding disorders. [The UniProt Consortium]
| Schlagworte: | Anti-NPYR5, Anti-NPY5R, Anti-NPY5-R, Anti-NPYY5-R, Anti-Y5 receptor, Anti-NPY-Y5 receptor, Anti-Neuropeptide Y receptor... |
| Anwendung: | ELISA, IHC (paraffin), IP, WB |
| Wirt: | Goat |
| Spezies-Reaktivität: | human |
871,00 €
Human NPY5R ELISA Kit
Artikelnummer: G-HUFI02669.96
| Anwendung: | ELISA |
| Spezies-Reaktivität: | human |
698,00 €
Anti-NPY5R
Artikelnummer: NSJ-R34109-100UG
0.5 mg/ml in 1X TBS, pH7.3, with 0.5% BSA (US sourced) and 0.02% sodium azide. Additional name(s) for this target protein: Neuropeptide Y receptor Y5 Protein function: Receptor for neuropeptide Y and peptide YY. The activity of this receptor is mediated by G proteins that inhibit adenylate cyclase activity. Seems to...
| Schlagworte: | Anti-NPY5R, Anti-NPYR5, Anti-NPY5-R, Anti-NPYY5-R, Anti-Y5 receptor, Anti-NPY-Y5 receptor, Anti-Neuropeptide Y receptor... |
| Anwendung: | WB, IHC, IP, ELISA (peptide) |
| Wirt: | Goat |
| Spezies-Reaktivität: | human |
836,00 €
![[Leu31,Pro34] Neuropeptide Y (human) (trifluoroacetate salt)](https://www.biomol.com/media/image/5d/a3/65/Cay24712-1_200x200.png "[Leu31,Pro34] Neuropeptide Y (human) (trifluoroacetate salt)")
[Leu31,Pro34] Neuropeptide Y (human) (trifluoroacetate salt)
Artikelnummer: Cay24712-1
[Leu31,Pro34] Neuropeptide Y (NPY) is an agonist of the NPY receptors Y1 and Y5 with Ki values of 0.11 and 0.17 nM, respectively, for human and 0.08 and 0.18 nM, respectively, for rhesus monkey receptors. It reduces forskolin-induced cAMP accumulation in L-M(TK-) cells expressing human and rat Y4 receptors (EC50s =...
| Schlagworte: | [Leu31,Pro34] NPY, 31-L-leucine-34-L-proline-neuropeptide Y (human), trifluoroacetate salt |
| Anwendung: | NPY1-R / NPY5-R agonist |
| MW: | 4240.7 D |
ab 228,00 €
CGP 71683 (hydrochloride)
Artikelnummer: Cay28778-1
CGP 71683 is an antagonist of neuropeptide Y (NPY) receptor Y5 (IC50 = 1.4 nM in a radioligand binding assay). It is selective for Y5 over Y1, Y2, and Y4 receptors (IC50s = 2,765, 7,187, and 5,637 nM, respectively). It inhibits NPY-induced increases in BT-549 cell growth and MDA-MB-231 cell migration when used at a...
| Schlagworte: | CGP 71683A, N-[[trans-4-[[(4-amino-2-quinazolinyl)amino]methyl]cyclohexyl]methyl]-1-naphthalenesulfonamide, monohydrochloride |
| Anwendung: | Neuropeptide Y (NPY) receptor Y5 antagonist |
| CAS | 192322-50-2 |
| MW: | 512.1 D |
ab 49,00 €
Velneperit
Artikelnummer: Cay33850-1
Velneperit is a nonpeptide antagonist of neuropeptide Y (NPY) receptor Y5 (Ki = 5.3 nM). It is selective for Y5 over Y1, Y2, and Y4 receptors, as well as a panel of 44 receptors, ion channels, transporters and enzymes, at 10 µM. Velneperit inhibits NPY-induced decreases in forskolin-induced cAMP production in CHO-K1...
| Schlagworte: | S-2367, trans-4-[[(1,1-dimethylethyl)sulfonyl]amino]-N-[5-(trifluoromethyl)-2-pyridinyl]-cyclohexanecarboxamide |
| Anwendung: | NPY receptor Y5 antagonist |
| CAS | 342577-38-2 |
| MW: | 407.5 D |
ab 57,00 €
![[cPP1-7,NPY19-23,Ala31,Aib32,Gln34] - Pancreatic Polypeptide (human) (acetate)](https://www.biomol.com/media/image/be/bf/17/Cay36718-1_200x200.png "[cPP1-7,NPY19-23,Ala31,Aib32,Gln34] - Pancreatic Polypeptide (human) (acetate)")
[cPP1-7,NPY19-23,Ala31,Aib32,Gln34] - Pancreatic...
Artikelnummer: Cay36718-1
[cPP1-7,NPY19-23,Ala31,Aib32,Gln34] - Pancreatic polypeptide is an agonist of the neuropeptide Y (NPY) receptor Y5. It inhibits cAMP production induced by forskolin (Cay-11018) in HEK293 cells expressing the human Y5 receptor (EC50 = 17 nM). [cPP1-7,NPY19-23,Ala31,Aib32,Gln34] - Pancreatic polypeptide selectively...
| Schlagworte: | glycyl-L-prolyl-L-seryl-L-glutaminyl-L-prolyl-L-threonyl-L-tyrosyl-L-prolylglycyl-L-alpha-aspartyl-L-asparaginyl-L-alanyl-... |
| Anwendung: | NPY receptor Y5 (NPY5R) agonist |
| MW: | 4207.7 D |
ab 92,00 €