Zu "K04201" wurden 30 Artikel gefunden!
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PG-106 (trifluoroacetate salt)
Artikelnummer: Cay41553-1
PG-106 is a cyclic peptidomimetic antagonist of melanocortin receptor 3 (MC3R, IC50 = 210 nM). It is selective for MC3R over MC4R and MC5R at 10 µM. InChI:...
| Schlagworte: | Ac-Nle-c[Asp-betaAla-DNal(2')-Arg-Trp-Lys]-NH2,... |
| Anwendung: | Melanocortin 3 receptor (MC3R) antagonist |
| MW: | 1008,18 D |
ab 75,00 €
CHO-K1/MC3/Galpha15 Stable Cell Line
Artikelnummer: GSC-M00242
Recombinant CHO-K1 cells stably overexpress human melanocortin 3 receptor (MC3R) on the surface and contain high levels of G protein Galphas to couple with the receptor in downstream signaling pathways.
| Schlagworte: | MC3R, Melanocortin receptor 3 |
11.424,00 €
![[D-Trp8]-gamma-MSH (trifluoroacetate salt)](https://www.biomol.com/media/image/68/1d/4d/Cay14037-1_200x200.png "[D-Trp8]-gamma-MSH (trifluoroacetate salt)")
[D-Trp8]-gamma-MSH (trifluoroacetate salt)
Artikelnummer: Cay14037-1
[D-Trp8]-gamma-MSH is a melanocortin receptor 3 (MC3R) agonist and an analog of gamma-melanocyte-stimulating hormone (gamma-MSH). It selectively induces cAMP accumulation in cells expressing MC3R over cells expressing MC4R or MC5R (EC50s = 0.33, 100, and 82 nM, respectively, for the human receptors). In vivo,...
| Schlagworte: | L-tyrosyl-L-valyl-L-methionylglycyl-L-histidyl-L-phenylalanyl-L-arginyl-D-tryptophyl-L-alpha-aspartyl-L-arginyl-L-phenylal... |
| Anwendung: | MC3R agonist |
| MW: | 1570.8 D |
ab 93,00 €
Anti-Melanocortin 3 Receptor
Artikelnummer: ARG55379.100
Protein function: Receptor for MSH (alpha, beta and gamma) and ACTH. This receptor is mediated by G proteins which activate adenylate cyclase. Required for expression of anticipatory patterns of activity and wakefulness during periods of limited nutrient availability and for the normal regulation of circadian clock...
| Schlagworte: | Anti-MC3R, Anti-MC3-R, Anti-Melanocortin receptor 3 |
| Anwendung: | WB, FC |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human |
616,00 €
Anti-MC3R
Artikelnummer: NSJ-R35931-100UG
0.5 mg/ml in 1X TBS, pH7.3, with 0.5% BSA (US sourced) and 0.02% sodium azide. Additional name(s) for this target protein: Melanocortin 3 Receptor Protein function: Receptor for MSH (alpha, beta and gamma) and ACTH. This receptor is mediated by G proteins which activate adenylate cyclase. Required for expression of...
| Schlagworte: | Anti-MC3R, Anti-MC3-R, Anti-Melanocortin receptor 3, MC3R Antibody |
| Anwendung: | WB, ELISA (peptide) |
| Wirt: | Goat |
| Spezies-Reaktivität: | human |
836,00 €
ACTH (1-13) (human, mouse, rat, porcine, bovine, ovine)...
Artikelnummer: Cay27150-1
ACTH (1-13) is a peptide fragment of adrenocorticotropic hormone (ACTH, Cay-24257), a peptide hormone found in the brain that is involved in the biological stress response. An acetylated form of ACTH (1-13), alpha-melanocyte stimulating hormone (alpha-MSH), is formed in the intermediate lobe of the pituitary gland...
| Schlagworte: | SYSMEHFRWGKPV-OH, alpha1-13-corticotropin, trifluoroacetate salt |
| Anwendung: | Peptide fragment, MC3R / MC4R agonist |
| MW: | 1623.8 D |
ab 110,00 €
AP1189 (acetate)
Artikelnummer: Cay37400-1
AP1189 is a biased agonist of melanocortin receptor 1 (MC1R) and MC3R. It induces ERK1 and ERK2 phosphorylation but not canonical cAMP production in HEK293 cells expressing human MC1R or MC3R when used at concentrations ranging from 10 pM to 1 mM. AP1189 (0.1-10 nM) reduces zymosan-induced IL-1beta, IL-6, and...
| Schlagworte: | 2-[3-[1-(2-nitrophenyl)-1H-pyrrol-2-yl]-2-propen-1-ylidene]-hydrazinecarboximidamide, acetate |
| Anwendung: | Biased MC1R / MC3R agonist |
| CAS | 959850-74-9 |
| MW: | 358.4 D |
ab 60,00 €
Anti-MC3R
Artikelnummer: CSB-PA261897.100
Host Species: Rabbit. Isotype: IgG. Buffer: Rabbit IgG in pH7.3 PBS, 0.05% NaN3, 50% Glycerol. Storage: Upon receipt, store at -20°C or -80°C. Avoid repeated freeze. Purification Method: Antigen Affinity Purified. Target Name: MC3R. Antigen Species: Human
| Schlagworte: | Anti-MC3R, Anti-MC3-R, Anti-Melanocortin receptor 3, BMIQ9 antibody, MC3 antibody, MC3 R antibody, MC3 Receptor antibody,... |
| Anwendung: | ELISA, WB |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human, mouse, rat |
284,00 €
AP1189 acetate
Artikelnummer: TGM-T9596-100mg
Description: AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors. Target: Melanocortin Receptor. Smiles: O=[N+](C1=CC=CC=C1N2C(/C=C/C=N/NC(N)=N)=CC=C2)[O-].CC(O)=O. References: Montero-Melendez T, et al. Biased agonism as a novel strategy to harness the proresolving properties of...
| Anwendung: | Biased MC1R / MC3R agonist |
| CAS | 959850-74-9 |
| MW: | 358.35 D |
ab 39,00 €
TCMCB07 (trifluoroacetate salt)
Artikelnummer: Cay41545-1
TCMCB07 is a peptide antagonist of melanocortin receptor 1 (MC1R), MC3R, MC4R, and MC5R (IC50s = 19.5, 0.59, 13.58, and 8.07 nM, respectively, for the human receptors). It is also an antagonist of dog MC1R, MC3R, MC4R, and MC5R receptors (IC50s = 53.64, 1.46, 7.14, and 11.22 nM, respectively). TCMCB07 (10 mg/kg)...
| Schlagworte: | Ac-Nle-Asp-Pro-D-2Nal-Arg-Trp-Lys-D-Val-D-Pro-NH2, Mifomelatide,... |
| Anwendung: | MC1R/MC3R/MC4R/MC5R peptide antagonist |
| MW: | 1230.5 D |
ab 58,00 €
MC3R Protein (human), hFc Tag
Artikelnummer: DIM-PME101797.10
Tag: C-Human Fc tag. This gene encodes a G-protein-coupled receptor for melanocyte-stimulating hormone and adrenocorticotropic hormone that is expressed in tissues other than the adrenal cortex and melanocytes. This gene maps to the same region as the locus for benign neonatal epilepsy. Mice deficient for this gene...
| Schlagworte: | MC3R, MC3-R, Melanocortin receptor 3, Human MC3R Protein, hFc Tag |
| Exprimiert in: | Human cells |
| Ursprungsart: | human |
| MW: | >30.1 kD |
ab 132,00 €
Nanodisc Human MC3R-Strep Protein
Artikelnummer: G-HDFP1069.10
Protein function: Receptor for MSH (alpha, beta and gamma) and ACTH. This receptor is mediated by G proteins which activate adenylate cyclase. Required for expression of anticipatory patterns of activity and wakefulness during periods of limited nutrient availability and for the normal regulation of circadian clock...
| Schlagworte: | MC3R, MC3-R, Melanocortin receptor 3 |
| Exprimiert in: | Human cells |
| Ursprungsart: | human |
1.605,00 €