Zu "K04150" wurden 57 Artikel gefunden!
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Betazole (hydrochloride)
Artikelnummer: Cay41712-10
Betazole is a histamine H2 receptor agonist. It induces acid secretion in isolated human gastric glands (EC50 = 120 µM), an effect mediated by histamine H2 receptors. Betazole (3-10 mg/kg) increases pepsin and acid levels in gastric juice in dogs.Formal Name: 1H-pyrazole-3-ethanamine, dihydrochloride. CAS Number:...
| Schlagworte: | Ametazole, Gastramine, 1H-pyrazole-3-ethanamine, dihydrochloride |
| Anwendung: | Histamine H2 receptor agonist |
| CAS | 138-92-1 |
| MW: | 184.1 D |
ab 67,00 €
Donetidine
Artikelnummer: TGM-T68056-100mg
Description: Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders. Target: Histamine Receptor. Smiles: C(C=1C(=O)NC(NCCSCC=2OC(CN(C)C)=CC2)=NC1)C3=CC(=O)NC=C3. References: Machálková M, et al. A label-free MALDI TOF MS-based method for studying the kinetics and inhibitor screening of...
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 99248-32-5 |
| MW: | 415.51 D |
ab 130,00 €
Cimetidine hydrochloride
Artikelnummer: TGM-T60584-100mg
Description: Cimetidine (SKF-92334) hydrochloride is an orally active inverse histamine H2 receptor antagonist with a Ki of 0.6 µM, demonstrating anti-cancer and anti-inflammatory activity, and is a gastric acid reducer useful in the research of duodenal and gastric ulcers [1] [2] [5]. Target: Others. Smiles:...
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 70059-30-2 |
| MW: | 288.8 D |
ab 1.520,00 €
Sufotidine
Artikelnummer: TGM-T68146-10mg
Description: Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist. Target: Histamine Receptor. Smiles: C(C1=CC(OCCCNC2=NC(CS(C)(=O)=O)=NN2C)=CC=C1)N3CCCCC3. References: Rogers MJ, et al. The effects of 15 days of dosing with placebo, sufotidine 600 mg nocte or sufotidine 600 mg twice daily...
| Schlagworte: | AH-25352X, AH 25352X, AH25352X |
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 80343-63-1 |
| MW: | 421.56 D |
ab 248,00 €
Tiotidine
Artikelnummer: TGM-T13163-1mL
Description: Tiotidine is a selective histamine H2-receptor antagonist (pA2=7.3-7.8 for guinea-pig right atrium). Target: Others. Smiles: CN\C(NC#N)=N/CCSCc1csc(NC(N)=N)n1. References: Barth H, et al. Structural requirements of imidazole compounds to be inhibitors or activators of histaminemethyltransferase:...
| Schlagworte: | ICI 125211 |
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 69014-14-8 |
| MW: | 312.42 D |
ab 54,00 €
Niperotidine
Artikelnummer: TGM-T12228-100mg
Description: Niperotidine is an antagonist of histamine H2-receptor. Target: Histamine Receptor. Smiles: CN(C)Cc1ccc(CSCCN\C(NCc2ccc3OCOc3c2)=C\[N+]([O-])=O)o1. References: Gasbarrini G, et al. Acute liver injury related to the use of Niperotidine. J Hepatol. 1997 Sep,27(3):583-6.
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 84845-75-0 |
| MW: | 434.51 D |
ab 1.520,00 €
Famotidine
Artikelnummer: TGM-T1627-2g
Description: Famotidine (MK-208) is a propanimidamide and histamine H2-receptor antagonist with antacid activity. As a competitive inhibitor of histamine H2-receptors on the basolateral membrane of parietal cells, famotidine reduces basal and nocturnal gastric acid secretion, thereby decreasing gastric volume,...
| Schlagworte: | MK-208 |
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 76824-35-6 |
| MW: | 337.45 D |
49,00 €
Nizatidine
Artikelnummer: TGM-T1575-1g
Description: Nizatidine (Acinon) is a competitive and reversible histamine H2-receptor antagonist with antacid activity. Target: Histamine Receptor, AChE. Smiles: CN\C(NCCSCc1csc(CN(C)C)n1)=C\[N+]([O-])=O. References: Lin TM, et al. J Pharmacol Exp Ther, 1986, 239(2), 406-410.
| Schlagworte: | Axid, Acinon, Zanizal |
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 76963-41-2 |
| MW: | 331.46 D |
30,00 €
Lavoltidine succinate
Artikelnummer: TGM-T32608-25mg
Description: Lavoltidine succinate is a biochemical. Target: Others. Smiles: OC(=O)CCC(O)=O.Cn1nc(CO)nc1NCCCOc1cccc(CN2CCCCC2)c1
| Schlagworte: | AH23844A, AH-23844A, AH 23844A |
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 86160-82-9 |
| MW: | 477.562 D |
1.520,00 €
Methantheline Bromide
Artikelnummer: TGM-T33314-100mg
Description: Methantheline Bromide is a synthetic spasmolytic used to relieve cramps or spasms of the stomach, bowel, and bladder. It is also useful for intestinal or gastric ulcers (peptic ulcer disease), intestinal problems, pancreatitis, gastritis, biliary dysmotility, pyloric or urinary problems. Target: Others....
| Schlagworte: | Frenogastrico, Dixamone bromide, Asabaine, Banthine, Methanthelinium bromide |
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 53-46-3 |
| MW: | 420.34 D |
ab 1.520,00 €
Dalcotidine
Artikelnummer: TGM-T31195-100mg
Description: Dalcotidine (KU 1257) is a novel histamine H2 receptor antagonist with histamine H9 receptor antagonistic activity and antisecretory effects.The Ki value for binding to guinea pig cerebral cortex was 0.040 The KB value for antagonism of histamine-induced positive chronotropic responses in the right...
| Schlagworte: | KU 1257, KU-1257 |
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 120958-90-9 |
| MW: | 319.44 D |
ab 142,00 €
Ranitidine
Artikelnummer: TGM-T3610-100mg
Description: Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors). It is used to treat gastrointestinal ulcers. Target: P450, Antibacterial, Histamine Receptor. Smiles: C(N(C)C)C=1OC(CSCCNC(=CN(=O)=O)NC)=CC1. References: Fedorowicz Z. et al,...
| Schlagworte: | HSDB 3925, Ranitidin |
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 66357-35-5 |
| MW: | 314.4 D |
ab 37,00 €