Zu "K04149" wurden 221 Artikel gefunden!
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Promethazine-d3 (hydrochloride)
Artikelnummer: Cay38299-1
Promethazine-d3 (Cay-38299) is intended for use as an internal standard for the quantification of promethazine (Cay-21331, Cay-22450) by GC- or LC-MS. Promethazine is categorized as a phenothiazine. It has been associated with misuse in conjunction with opioids or sedatives. Formulations containing promethazine have...
| Schlagworte: | N,alpha-dimethyl-N-(methyl-d3)-10H-phenothiazine-10-ethanamine, monohydrochloride |
| Anwendung: | GC-MS, LC-MS internal standard, quantification, phenothiazine |
| CAS | 1435933-86-0 |
| MW: | 323.9 D |
ab 513,00 €
Norastemizole
Artikelnummer: Cay41828-1
Norastemizole is a histamine H1 receptor antagonist (IC50 = 4.1 nM) and an active metabolite of the histamine H1 receptor antagonist and ether-a-go-go (ERG) channel blocker astemizole (Cay-16967). It is formed from astemizole by the cytochrome P450 (CYP) isoform 3A4 (CYP3A4). Norastemizole also inhibits currents in...
| Schlagworte: | Tecastemizole, 1-[(4-fluorophenyl)methyl]-N-4-piperidinyl-1H-benzimidazol-2-amine |
| Anwendung: | Astemizole active metabolite, histamine H1 receptor antagonist |
| CAS | 75970-99-9 |
| MW: | 324.4 D |
ab 52,00 €
Promethazine-d3 (hydrochloride) (CRM)
Artikelnummer: Cay39606-100
Promethazine-d3 (hydrochloride) (CRM) (Cay-39606) is intended for use as an internal standard for the quantification of promethazine (Cay-21331, Cay-22450) by GC- or LC-MS. Promethazine is categorized as a phenothiazine. It has been associated with misuse in conjunction with opioids or sedatives. Formulations...
| Schlagworte: | N,alpha-dimethyl-N-(methyl-d3)-10H-phenothiazine-10-ethanamine, monohydrochloride |
| Anwendung: | GC-MS, LC-MS, internal standard, quantification, phenothiazine, Histamine receptor H1 antagonist |
| CAS | 1435933-86-0 |
| MW: | 323.9 D |
172,00 €
Epinastine
Artikelnummer: TGM-T60366-5mg
Description: Epinastine (WAL801), a potent, selective, and orally-active antihistamine and mast cell stabilizer, functions as a histamine H1 receptor antagonist. It also inhibits IL-8 release from human eosinophils, showcasing antiallergic action [1] [2] [3] [4]. Target: Others. Smiles: NC1=NCC2N1c1ccccc1Cc1ccccc21
| Anwendung: | Targets histamine receptor H1 (HRH1) |
| CAS | 80012-43-7 |
| MW: | 249.31 D |
31,00 €
Tripelennamine
Artikelnummer: TGM-T60392-100mg
Description: Tripelennamine, an ethylenediamine derivative, acts as a potent histamine H1-receptor antagonist, effectively reducing the organism's allergic response to histamine. It is utilized in researching conditions such as rhinitis, conjunctivitis, and allergic and anaphylactic reactions [1] [2] [3]. Target:...
| Anwendung: | Targets histamine receptor H1 (HRH1) |
| CAS | 91-81-6 |
| MW: | 255.36 D |
ab 4.526,00 €
Phenindamine
Artikelnummer: TGM-T60424-100mg
Description: Phenindamine (Nu 1504) is an H1-receptor antagonist with antihistamine properties[1]. Target: Others. Smiles: CN1CC=2C(C=3C(C2CC1)=CC=CC3)C4=CC=CC=C4
| Anwendung: | Targets histamine receptor H1 (HRH1) |
| CAS | 82-88-2 |
| MW: | 261.36 D |
ab 1.520,00 €
Rupatadine Fumarate
Artikelnummer: TGM-T6242-100mg
Description: Rupatadine Fumarate (Rinialer) (UR-12592 Fumarate) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 uM. Target: Autophagy, PAFR, Histamine Receptor. Smiles: OC(=O)\C=C\C(O)=O.Cc1cncc(CN2CC\C(CC2)=C2/c3ccc(Cl)cc3CCc3cccnc23)c1. References: Merlos M, et al. J Pharmacol Exp Ther, 1997, 280(1),...
| Schlagworte: | Alergoliber, Rinialer, Rupafin |
| Anwendung: | Targets histamine receptor H1 (HRH1) |
| CAS | 182349-12-8 |
| MW: | 532.03 D |
ab 33,00 €
Buclizine
Artikelnummer: TGM-T62421-100mg
Description: Buclizine is an orally active antihistamine, antiallergic compound. buclizine is also a strong teratogen in rats and exhibits antitumour effects. Target: Others. Smiles: CC(C)(C)c1ccc(CN2CCN(CC2)C(c2ccccc2)c2ccc(Cl)cc2)cc1
| Anwendung: | Targets histamine receptor H1 (HRH1) |
| CAS | 82-95-1 |
| MW: | 433.03 D |
ab 1.520,00 €
Chlorpheniramine
Artikelnummer: TGM-T60498-100mg
Description: Chlorpheniramine is an H1 anti-histamine agent for IgE-mediated inflammation that is commonly used for allergic diseases. Target: Others. Smiles: C(CCN(C)C)(C1=CC=C(Cl)C=C1)C2=CC=CC=N2
| Anwendung: | Targets histamine receptor H1 (HRH1) |
| CAS | 132-22-9 |
| MW: | 274.79 D |
ab 1.520,00 €
Triprolidine
Artikelnummer: TGM-T60514-100mg
Description: Triprolidine is an orally active antagonist of H1R. Triprolidine has spinal cord motor and sensory block effects. Triprolidine can be used in allergic rhinitis research[1] [2] [3]. Target: Others. Smiles: CC1=CC=C(C=C1)C(=C/CN1CCCC1)\C1=NC=CC=C1
| Anwendung: | Targets histamine receptor H1 (HRH1) |
| CAS | 486-12-4 |
| MW: | 278.39 D |
ab 1.520,00 €
Cyproheptadine
Artikelnummer: TGM-T60576-500mg
Description: Cyproheptadine is a potent, orally active antagonist of the 5-HT 2A receptor with antidepressant, antiserotonergic, antiplatelet, and thromboprotective effects, useful in thromboembolic disorders research [1] [2]. Target: Others. Smiles: CN1CCC(CC1)=C1C2=C(C=CC=C2)C=CC2=C1C=CC=C2
| Anwendung: | Targets histamine receptor H1 (HRH1) |
| CAS | 129-03-3 |
| MW: | 287.4 D |
1.130,00 €
Tripelennamine citrate
Artikelnummer: TGM-T62669-100mg
Description: Tripelennamine citrate is an ethylenediamine derivative and is a potent histamine H1 receptor antagonist. tripelennamine citrate reduces histamine-induced allergic reactions in the body. tripelennamine citrate can be used to study rhinitis, conjunctivitis, allergic and anaphylactic reactions. Target:...
| Anwendung: | Targets histamine receptor H1 (HRH1) |
| CAS | 6138-56-3 |
| MW: | 447.488 D |
ab 1.520,00 €