Zu "K04143" wurden 73 Artikel gefunden!

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Solabegron HCl
Solabegron HCl

Artikelnummer: TGM-T12970L-100mg

Description: Solabegron (GW-427,353), is a selective agonist of beta3 adrenergic receptors. In addition, Solabegron has been shown to produce visceral analgesia by releasing somatostatin from fat cells. Target: Others. Smiles: C(O)(=O)C=1C=C(C=CC1)C2=CC(NCCNC[C@H](O)C3=CC(Cl)=CC=C3)=CC=C2.Cl. References: Rosa GM,...
Schlagworte: GW-427,353, GW427353, GW 427,353, GW427,353, GW-427353
Anwendung: Targets adrenergic receptor beta-3 (ADRB3)
CAS 451470-34-1
MW: 447.35 D
ab 1.671,00 €
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Mirabegron
Mirabegron

Artikelnummer: TGM-T1671-100mg

Description: Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome. Target: Adrenergic Receptor. Smiles: N(C(CC1=CSC(N)=N1)=O)C2=CC=C(CCNC[C@H](O)C3=CC=CC=C3)C=C2. References: Takasu T, et al. J Pharmacol Exp Ther, 2007, 321(2), 642-647.
Schlagworte: YM178
Anwendung: Targets adrenergic receptor beta-3 (ADRB3)
CAS 223673-61-8
MW: 396.51 D
ab 31,00 €
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Vibegron
Vibegron

Artikelnummer: TGM-T35052-100mg

Description: Vibegron (MK-4618) is an effective and selective Beta 3 adrenergic receptor agonist, used to treat overactive bladder (OAB). Target: Others. Smiles: O[C@@H]([C@H]1CC[C@@H](Cc2ccc(NC(=O)[C@@H]3CCc4nccc(=O)n34)cc2)N1)c1ccccc1. References: Edmondson SD, Zhu C, Kar NF, Di Salvo J, Nagabukuro H, Sacre-Salem...
Schlagworte: MK-4618, MK4618, MK 4618
Anwendung: Targets adrenergic receptor beta-3 (ADRB3)
CAS 1190389-15-1
MW: 444.53 D
ab 2.573,00 €
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Fasobegron
Fasobegron

Artikelnummer: TGM-T31748-100mg

Description: Fasobegron is a agonist of beta3-adrenoreceptor . Target: Others. Smiles: O(C)C=1C=C(C=CC1C(O)=O)C2=CC=C(CCNC[C@H](O)C3=CC(Cl)=CC=C3)C=C2
Anwendung: Targets adrenergic receptor beta-3 (ADRB3)
CAS 643094-49-9
MW: 425.91 D
ab 1.671,00 €
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L755507
L755507

Artikelnummer: TGM-T6872-100mg

Description: L755507 is an effective, selective agonist of beta3-AR(IC50=35 nM). Target: CRISPR/Cas9, Adrenergic Receptor. Smiles: CCCCCCNC(=O)Nc1ccc(cc1)S(=O)(=O)Nc1ccc(CCNC[C@H](O)COc2ccc(O)cc2)cc1. References: Parmee ER, et al. Bioorg Med Chem Lett. 1998, 8(9):1107-1112.
Anwendung: Partial beta-3 adrenergic receptor agonist
CAS 159182-43-1
MW: 584.73 D
ab 45,00 €
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Amibegron
Amibegron

Artikelnummer: TGM-T71216-100mg

Description: Amibegron is a selective agonist for the beta3 adrenergic receptor. It is the first orally active beta3 agonist developed that is capable of entering the central nervous system. Amibegron has antidepressant and anxiolytic effects. Target: Others. Smiles:...
Anwendung: Targets adrenergic receptor beta-3 (ADRB3)
CAS 121524-08-1
MW: 403.9 D
ab 1.520,00 €
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Anti-ADRB3
Anti-ADRB3

Artikelnummer: CSB-PA007545.100

Host Species: Rabbit. Isotype: IgG. Buffer: Liquid in PBS containing 50% glycerol, 0.5% BSA and 0.02% sodium azide. Storage: Upon receipt, store at -20°C or -80°C. Avoid repeated freeze. Purification Method: The antibody was affinity-purified from rabbit antiserum by affinity-chromatography using epitope-specific...
Schlagworte: Anti-ADRB3, Anti-ADRB3R, Anti-Beta-3 adrenoceptor, Anti-Beta-3 adrenoreceptor, Anti-Beta-3 adrenergic receptor, ADR B3...
Anwendung: ELISA, WB
Wirt: Rabbit
Spezies-Reaktivität: human, mouse, rat
ab 126,00 €
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Anti-ADRB3
Anti-ADRB3

Artikelnummer: CSB-PA120361.100

Host Species: Rabbit. Isotype: IgG. Buffer: -20°C, pH7.4 PBS, 0.05% NaN3, 40% Glycerol. Storage: Upon receipt, store at -20°C or -80°C. Avoid repeated freeze. Purification Method: Antigen affinity purification. Target Name: ADRB3. Antigen Species: Human
Schlagworte: Anti-ADRB3, Anti-ADRB3R, Anti-Beta-3 adrenoceptor, Anti-Beta-3 adrenoreceptor, Anti-Beta-3 adrenergic receptor, ADR B3...
Anwendung: ELISA, IHC
Wirt: Rabbit
Spezies-Reaktivität: human
ab 167,00 €
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Anti-ADRB3
Anti-ADRB3

Artikelnummer: CSB-PA235900.100

Host Species: Rabbit. Isotype: IgG. Buffer: -20°C, pH7.4 PBS, 0.05% NaN3, 40% Glycerol. Storage: Upon receipt, store at -20°C or -80°C. Avoid repeated freeze. Purification Method: Antigen affinity purification. Target Name: ADRB3. Antigen Species: Human
Schlagworte: Anti-ADRB3, Anti-ADRB3R, Anti-Beta-3 adrenoceptor, Anti-Beta-3 adrenoreceptor, Anti-Beta-3 adrenergic receptor, ADR B3...
Anwendung: ELISA, WB, IHC
Wirt: Rabbit
Spezies-Reaktivität: human, mouse
ab 167,00 €
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Anti-ADRB3
Anti-ADRB3

Artikelnummer: CSB-PA779661.100

Host Species: Rabbit. Isotype: IgG. Buffer: -20°C, pH7.4 PBS, 0.05% NaN3, 40% Glycerol. Storage: Upon receipt, store at -20°C or -80°C. Avoid repeated freeze. Purification Method: Antigen affinity purification. Target Name: ADRB3. Antigen Species: Human
Schlagworte: Anti-ADRB3, Anti-ADRB3R, Anti-Beta-3 adrenoceptor, Anti-Beta-3 adrenoreceptor, Anti-Beta-3 adrenergic receptor, ADR B3...
Anwendung: ELISA, IHC
Wirt: Rabbit
Spezies-Reaktivität: human
ab 167,00 €
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Anti-ADRB3
Anti-ADRB3

Artikelnummer: CSB-PA831980.100

Host Species: Rabbit. Isotype: IgG. Buffer: -20°C, pH7.4 PBS, 0.05% NaN3, 40% Glycerol. Storage: Upon receipt, store at -20°C or -80°C. Avoid repeated freeze. Purification Method: Antigen affinity purification. Target Name: ADRB3. Antigen Species: Human
Schlagworte: Anti-ADRB3, Anti-ADRB3R, Anti-Beta-3 adrenoceptor, Anti-Beta-3 adrenoreceptor, Anti-Beta-3 adrenergic receptor, ADR B3...
Anwendung: ELISA, WB, IHC
Wirt: Rabbit
Spezies-Reaktivität: human
ab 167,00 €
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Mirabegron
Mirabegron

Artikelnummer: Cay17319-10

Mirabegron is an agonist of the beta3-adrenergic receptor (beta3-AR). It induces cAMP accumulation in CHO cells expressing the beta3-AR but not the beta1- or beta2-AR (EC50s = 0.0224, >10, and >10 µM, respectively). Mirabegron reduces contraction induced by carbamoylcholine (Cay-14486) of isolated rat and human...
Schlagworte: YM-178, 2-amino-N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-4-thiazoleacetamide
Anwendung: beta3-adrenergic receptor agonist
CAS 223673-61-8
MW: 396.5 D
ab 52,00 €
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