Zu "K04140" wurden 58 Artikel gefunden!
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Romifidine (hydrochloride)
Artikelnummer: Cay36693-50
Romifidine is an alpha2-adrenergic receptor (alpha2-AR) agonist. Epidural administration of romifidine (50 µg/kg) induces antinociception and sedation in donkeys. It also induces bradycardia in horses when administered at doses ranging from 0.04 to 0.12 mg/kg. Formulations containing romifidine have been used as...
| Schlagworte: | STH 2130, N-(2-bromo-6-fluorophenyl)-4,5-dihydro-1H-imidazol-2-amine, monohydrochloride |
| Anwendung: | Alpha2-AR agonist |
| CAS | 65896-14-2 |
| MW: | 294.6 D |
ab 93,00 €
Dexmedetomidine
Artikelnummer: Cay39544-250
Dexmedetomidine is an agonist of alpha2-adrenergic receptors (alpha2-ARs). It selectively binds to alpha2-ARs over alpha1-ARs (Kis = 0.015 and 5 nM, respectively). In vivo, dexmedetomidine (50 µg/kg) prevents increases in cardiac troponin I (CTnI), a marker of myocardial injury, as well as reduces myocardial...
| Schlagworte: | MPV 1440, 5-[(1S)-1-(2,3-dimethylphenyl)ethyl]-1H-imidazole |
| Anwendung: | Alpha2-AR agonist, sedative-hypnotic |
| CAS | 113775-47-6 |
| MW: | 200.3 D |
ab 53,00 €
Rat ADRa2C (Adrenergic Receptor Alpha 2C) ELISA Kit
Artikelnummer: ELK-ELK6355.48
The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Rat ADRa2C. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Rat ADRa2C. Next,...
| Schlagworte: | Adra2c, Alpha-2CAR, Alpha-2C adrenoceptor, Alpha-2C adrenoreceptor, Alpha-2C adrenergic receptor, Alpha-2 adrenergic... |
| Anwendung: | ELISA |
| Spezies-Reaktivität: | rat |
ab 365,00 €
Human ADRa2C (Adrenergic Receptor Alpha 2C) ELISA Kit
Artikelnummer: ELK-ELK3967.48
The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Human ADRa2C. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Human ADRa2C....
| Schlagworte: | ADRA2C, ADRA2L2, Alpha-2CAR, Alpha-2C adrenoceptor, Alpha-2C adrenoreceptor, Alpha-2C adrenergic receptor, Alpha-2... |
| Anwendung: | ELISA |
| Spezies-Reaktivität: | human |
ab 365,00 €
Xylazine
Artikelnummer: Cay14113-25
Xylazine is an agonist of alpha2-adrenergic receptors (Ki = 194 nM). It is an analog of clonidine, an alpha2-adrenergic receptor agonist used to reduce blood pressure. Xylazine is used for sedation, anesthesia, and analgesia in non-human mammals. This product is also available as an analytical reference standard...
| Schlagworte: | N-(2,6-dimethylphenyl)-5,6-dihydro-4H-1,3-thiazin-2-amine |
| Anwendung: | alpha2 adrenergic receptor agonist |
| CAS | 7361-61-7 |
| MW: | 220.3 D |
ab 48,00 €
Xylazine (hydrochloride)
Artikelnummer: Cay36692-5
Xylazine is an agonist of alpha2-adrenergic receptors (Ki = 194 nM). It is an analog of clonidine, an alpha2-adrenergic receptor agonist used to reduce blood pressure. Xylazine is used for sedation, anesthesia, and analgesia in non-human mammals. This product is also available as an analytical reference standard...
| Schlagworte: | BAY-Va 1470, N-(2,6-dimethylphenyl)-5,6-dihydro-4H-1,3-thiazin-2-amine, monohydrochloride |
| Anwendung: | Alpha2-adrenergic receptors agonist |
| CAS | 23076-35-9 |
| MW: | 256.8 D |
ab 35,00 €
Atipamezole (hydrochloride)
Artikelnummer: Cay9001181-5
Atipamezole is an antagonist of alpha2A-adrenergic receptors (alpha2A-ARs, Ki = 1.86 nM). It is selective for alpha2A-ARs over alpha2B- and alpha1-ARs (Kis = 1,949.83 and 13,300 nM, respectively), as well as over 40 receptors, ion channels, and transporters (IC50s = 540->10,000 nM). Atipamezole (0.04, 0.08, and 1.2...
| Schlagworte: | Antisedan(R), 5-(2-ethyl-2,3-dihydro-1H-inden-2-yl)-1H-imidazole, monohydrochloride |
| Anwendung: | alpha2-adrenergic receptor antagonist |
| CAS | 104075-48-1 |
| MW: | 248.8 D |
ab 97,00 €
Dexmedetomidine (hydrochloride)
Artikelnummer: Cay15581-5
Dexmedetomidine is the (S)-enantiomer of medetomidine, an imidazole compound that binds to alpha2-adrenoceptors (Ki = 1.08 nM) with high affinity and selectivity compared to that of alpha1-adrenoceptors (Ki = 1.8 µM). Dexmedetomidine produces analgesic, sedative, and anxiolytic effects through both presynaptic...
| Schlagworte: | Dex, Precedex, 5-[(1S)-1-(2,3-dimethylphenyl)ethyl]-1H-imidazole, monohydrochloride |
| Anwendung: | alpha2-adrenergic receptor agonist |
| CAS | 145108-58-3 |
| MW: | 236.7 D |
ab 66,00 €
Guanabenz (hydrochloride)
Artikelnummer: Cay10851-25
Guanabenz is an alpha2-adrenergic receptor agonist (effective concentrations 10-100 nM) with hypotensive effects. It also competes for imidazoline I2-binding sites in brown adipose tissue (Ki = 97 nM).Formal Name: 2-[(2,6-dichlorophenyl)methylene]-hydrazinecarboximidamide, monohydrochloride. CAS Number: 23113-43-1....
| Schlagworte: | Wytensin, 2-[(2,6-dichlorophenyl)methylene]-hydrazinecarboximidamide, monohydrochloride |
| Anwendung: | alpha2-adrenergic receptor agonist |
| CAS | 23113-43-1 |
| MW: | 267.5 D |
ab 61,00 €
Quercetin 3-O-glucuronide
Artikelnummer: Cay21289-1
Quercetin 3-O-glucuronide is a pharmacologically active flavonol glucuronide isolated from H. perforatum (St. John's wort) that inhibits the alpha2c adrenergic receptor (Ki = 4,060 nM in halpha2c preparations).{33869,33870, 33974} Quercetin 3-O-glucuronide (0.6 mg/kg) reduced the time rats spent immobile in the...
| Schlagworte: | Miquelianin, Quercetin 3-O-beta-D-glucuronide,... |
| Anwendung: | alpha-2C adrenergic receptor inhibitor |
| CAS | 22688-79-5 |
| MW: | 478.4 D |
ab 66,00 €
Clonidine (hydrochloride)
Artikelnummer: Cay15949-500
Clonidine is an agonist of alpha2-adrenergic receptors (alpha2-ARs, Kis = 61.66, 69.18, and 134.9 nM for alpha2A-, alpha2B-, and alpha2C-ARs, respectively). It stimulates [35S]GTPgammaS binding to HEK293 cell membranes expressing the human receptors with EC50 values of 26.92, 56.23, and 912.01 nM for alpha2A-,...
| Schlagworte: | ST 155, N-(2,6-dichlorophenyl)-4,5-dihydro-1H-imidazol-2-amine, monohydrochloride |
| Anwendung: | alpha2-adrenergic receptor agonist |
| CAS | 4205-91-8 |
| MW: | 266.6 D |
ab 43,00 €
Rauwolscine (hydrochloride)
Artikelnummer: Cay15596-50
Rauwolscine is a natural alkaloid that acts as a selective and reversible alpha2-adrenergic receptor antagonist (Ki = 12 nM). It is a stereoisomer of yohimbine, which potently antagonizes both alpha1- and alpha2-adrenergic receptors. Rauwolscine also acts as a receptor antagonist at the serotonin 5-HT2B receptor (Ki...
| Schlagworte: | Isoyohimbine, NSC 407307, alpha-Yohimbine, (16beta,17alpha,20alpha)-17-hydroxy-yohimban-16-carboxylic acid, methyl ester,... |
| Anwendung: | Selective, reversible alpha2-adrenergic receptor antagonist |
| CAS | 6211-32-1 |
| MW: | 390.9 D |
ab 50,00 €