Zu "K04137" wurden 52 Artikel gefunden!
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CHO-K1/ADRA1D Stable Cell Line
Artikelnummer: GSC-M00340
Recombinant CHO-K1 cells stably overexpress human adrenoceptor alpha 1D (ADRA1D) on the surface and contain high levels of G protein Galphaq to couple with the receptor in downstream signaling pathways.
| Schlagworte: | ADRA1D, Alpha-1D adrenoreceptor, Alpha-adrenergic receptor 1a, Alpha-1A adrenergic receptor, Alpha-1D adrenergic receptor |
11.424,00 €
(-)-Norepinephrine (bitartrate hydrate)
Artikelnummer: Cay16673-250
(-)-Norepinephrine is the endogenous isomer of (±)-norepinephrine (Cay-35580) that acts as a neurotransmitter and hormone and is biosynthesized from dopamine by dopamine beta-hydroxylase. It is an agonist of adrenergic receptors (Ki values are 330, 56, and 740 nM for alpha1, alpha2, and beta1 adrenoceptors,...
| Schlagworte: | Arterenol, Levarterenol, L-Noradrenaline, NE, 4-[(1R)-2-amino-1-hydroxyethyl]-1,2-benzenediol... |
| Anwendung: | Adrenergic receptor agonist, dopamine beta-hydroxylase metabolite |
| CAS | 108341-18-0 |
| MW: | 337.3 D |
ab 50,00 €
Acetylcholine (chloride)
Artikelnummer: Cay23829-5
Acetylcholine is a neurotransmitter that binds to nicotinic and muscarinic acetylcholine receptors (AChRs) in the central and peripheral nervous systems. It mediates motor function at the neuromuscular junction but also has functions in the parasympathetic and sympathetic nervous systems. It is involved in learning...
| Schlagworte: | ACh, 2-(acetyloxy)-N,N,N-trimethyl-ethanaminium, monochloride |
| Anwendung: | alpha1-Adrenergic receptor agonist |
| CAS | 60-31-1 |
| MW: | 181.7 D |
56,00 €
Phentolamine (mesylate)
Artikelnummer: Cay16135-100
Phentolamine is a reversible antagonist of alpha-adrenergic receptors, non-specifically binding all alpha1- and alpha2-adrenoceptors with nanomolar affinities. Formulations containing phentolamine have been used in the treatment of hypertensive emergencies, as well as chronic and emergent pain.Formal Name:...
| Schlagworte: | 3-[[(4,5-dihydro-1H-imidazol-2-yl)methyl](4-methylphenyl)amino]-phenol, monomethanesulfonate |
| Anwendung: | alpha1/2-adrenergic receptor antagonist |
| CAS | 65-28-1 |
| MW: | 377.5 D |
ab 67,00 €
Prazosin (hydrochloride)
Artikelnummer: Cay15023-100
Prazosin is an antagonist of alpha1-adrenergic receptors (alpha1-ARs). It selectively binds to alpha1-ARs with Ki values of 0.2, 0.25, and 0.32 nM for the human recombinant alpha1A-, alpha1B-, and alpha1D-ARs, respectively, over alpha2-ARs (Kis = 340 and 3.7 nM in alpha2A-AR-expressing HT-29 cells and...
| Schlagworte: | CP 12,299-1, NSC 292810, [4-(4-amino-6,7-dimethoxy-2-quinazolinyl)-1-piperazinyl]-2-furanyl-methanone, monohydrochloride |
| Anwendung: | Antihypertensive agent, melatonin MT3 receptor antagonist |
| CAS | 19237-84-4 |
| MW: | 419.9 D |
ab 49,00 €
Urapidil hydrochloride
Artikelnummer: LKT-U6802.500
White solid. An alpha1-adrenergic antagonist. In addition, it has high affinity and selectivity for central 5-hydroxytryptamine binding sites and inhibits platelet aggregation.
| Anwendung: | alpha1-adrenergic antagonist |
| CAS | 64887-14-5 |
| MW: | 423,93 D |
ab 193,00 €
Synephrine
Artikelnummer: LKT-S9753.1
A biogenic amine present in herbal products and citrus juices. It has antidepressant-like effects by stimulating alpha1-adrenoceptors in mice.
| Anwendung: | alpha-adrenergic receptor agonist |
| CAS | 94-07-5 |
| MW: | 167,21 D |
ab 64,00 €
Methyl 5,6,7,8-Tetradehydro Risperidone
Artikelnummer: Cay17801-10
Risperidone (Cay-13629) is a benzisoxazole derivative used for treating schizophrenia, and also the psychotic, affective, or behavioral symptoms associated with other disorders. Methyl 5,6,7,8-tetradehydro risperidone is used as an internal standard used in the quantitative analysis of risperidone.Formal Name:...
| Schlagworte: | 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-2,7-dimethyl-4H-pyrido[1,2-a]pyrimidin-4-one |
| Anwendung: | Internal standard |
| CAS | 106266-08-4 |
| MW: | 420.5 D |
ab 56,00 €
Risperidone E-oxime
Artikelnummer: Cay22156-10
Risperidone E-oxime is a potential impurity found in commercial preparations of risperidone. Risperidone (Cay-13629) is a longer-acting benzisoxazole derivative used for treating schizophrenia, and also the psychotic, affective, or behavioral symptoms associated with other disorders. This second-generation...
| Schlagworte: | 3-[2-[4-[(E)-(2,4-difluorophenyl)(hydroxyimino)methyl]-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]py... |
| Anwendung: | Potential impurity |
| CAS | 691007-09-7 |
| MW: | 430.5 D |
ab 93,00 €
Tamsulosin (hydrochloride)
Artikelnummer: Cay24020-50
Tamsulosin is a potent antagonist of alpha1-adrenergic receptors (alpha1-ARs, Ki = 0.229 nM in a radioligand binding assay). It is 3,800-fold selective for alpha1-ARs over alpha2-ARs (Ki = 871 nM). Tamsulosin antagonizes norepinephrine-induced contraction of isolated rabbit aorta (pA2 = 10.11) but has no effect on...
| Schlagworte: | LY253351, YM-12617-1, 5-[(2R)-2-[[2-(2-ethoxyphenoxy)ethyl]amino]propyl]-2-methoxy-benzenesulfonamide, monohydrochloride |
| Anwendung: | alpha1-Adrenergic receptor antagonist |
| CAS | 106463-17-6 |
| MW: | 445 D |
ab 72,00 €
Silodosin
Artikelnummer: LKT-S3346.100
A potent and highly selective antagonist of human alpha 1a-adrenoceptor.
| Schlagworte: | KAD 3213, KMD 3213 |
| Anwendung: | Antagonist of human alpha 1a-adrenoceptor |
| CAS | 160970-54-7 |
| MW: | 495,53 D |
ab 140,00 €
Terazosin hydrochloride dihydrate
Artikelnummer: LKT-T1670.1
An alpha1-selective blocker. Its inhibitory effect on prostate tumor growth may be the result of antiangiogenic activity.
| Anwendung: | Alpha1-adrenergic receptor antagonist |
| CAS | 70024-40-7 |
| MW: | 459,93 D |
ab 134,00 €