Zu "K03915" wurden 27 Artikel gefunden!
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ELN441958
Artikelnummer: Cay43214-1
ELN441958 is a bradykinin B1 receptor antagonist (Ki = 0. nM). It is selective for the bradykinin B1 receptor over a panel of greater than 100 enzymes and receptors at 10 µM but does bind to the µ-, delta-, and kappa-opioid receptors and M1 muscarinic receptor (Kis = 0. 0. 1. and 0. µM, respectively). ELN441958...
| Schlagworte: | 7-chloro-2,3-dihydro-2-[3-[[9-(4-pyridinyl)-3,9-diazaspiro[5.5]undec-3-yl]carbonyl]phenyl]-1H-isoindol-1-one |
| Anwendung: | Bradykinin B1 receptor antagonist |
| CAS | 913064-47-8 |
| MW: | 501.03 D |
ab 88,00 €
SCH 79797 (hydrochloride)
Artikelnummer: Cay14633-1
SCH 79797 is a non-peptide antagonist of proteinase-activated receptor 1 (PAR1). It blocks binding of the high affinity thrombin receptor-activating peptide (haTRAP) (IC50 = 70 nM) as well as platelet aggregation induced by either haTRAP or alpha-thrombin (IC50 = 0.3 and 3 µM, respectively). SCH 79797 has no...
| Schlagworte: | N3-cyclopropyl-7-[[4-(1-methylethyl)phenyl]methyl]-7H-pyrrolo[3,2-f]quinazoline-1,3-diamine, monohydrochloride |
| Anwendung: | PAR1 antagonist |
| CAS | 1216720-69-2 |
| MW: | 444.4 D |
ab 68,00 €
Anti-Bradykinin receptor B1, Internal
Artikelnummer: ARG64653.100
Protein function: This is a receptor for bradykinin. Could be a factor in chronic pain and inflammation. [The UniProt Consortium]
| Schlagworte: | Anti-B1R, Anti-BDKRB1, Anti-BRADYB1, Anti-BK-1 receptor, Anti-B1 bradykinin receptor |
| Anwendung: | ELISA, WB |
| Wirt: | Goat |
| Spezies-Reaktivität: | human |
871,00 €
Anti-BDKRB1
Artikelnummer: NSJ-R34695-100UG
0.5 mg/ml in 1X TBS, pH7.3, with 0.5% BSA (US sourced) and 0.02% sodium azide. Additional name(s) for this target protein: Bradykinin receptor B1 Protein function: This is a receptor for bradykinin. Could be a factor in chronic pain and inflammation. [The UniProt Consortium]
| Schlagworte: | Anti-B1R, Anti-BDKRB1, Anti-BRADYB1, Anti-BK-1 receptor, Anti-B1 bradykinin receptor, BDKRB1 Antibody |
| Anwendung: | WB, ELISA (peptide) |
| Wirt: | Goat |
| Spezies-Reaktivität: | human |
836,00 €
![Bradykinin [DPhe7]](https://www.biomol.com/media/image/48/97/89/LKT-B6809-1_200x200.png "Bradykinin [DPhe7]")
Bradykinin [DPhe7]
Artikelnummer: LKT-B6809.1
| Anwendung: | Vasodilatory peptide |
| MW: | 1110.29 D |
ab 90,00 €
Lys-(Des-Arg9)-Bradykinin (trifluoroacetate salt)
Artikelnummer: Cay29922-10
Lys-(Des-Arg9)-Bradykinin is a naturally occurring peptide agonist of the bradykinin B1 receptor (Ki = 0.12 nM in HEK293 cells expressing the human receptor). It is selective for bradykinin B1 over B2 receptors (IC50 = >30,000 nM in CHO cells expressing the human receptor). Lys-(Des-Arg9)-Bradykinin increases both...
| Schlagworte: | (Des-Arg10)-Kallidin, (Des-Arg10)-KD, KRPPGFSPF-OH, Lys-(Des-Arg9)-BK, N2-L-lysyl-9-de-L-arginine-Bradykinin,... |
| Anwendung: | Bradykin in B1 receptor peptide agonist |
| MW: | 1032.2 D |
ab 68,00 €
Lys-(Des-Arg9, Leu8)-Bradykinin (trifluoroacetate salt)
Artikelnummer: Cay35462-10
Lys-(Des-Arg9, Leu8)-Bradykinin is a bradykinin B1 receptor antagonist (Ki = 0.43 nM for the rabbit aorta receptor). It is selective for the bradykinin B1 over the B2 receptor (Ki = >10 µM for the rabbit ileum receptor). Lys-(Des-Arg9, Leu8)-Bradykinin inhibits contractions induced by the bradykinin B1 receptor...
| Schlagworte: | [Des-Arg10,Leu9]-Kallidin, [Des-Arg10,Leu9]-KD, Lys[Leu8]Des-Arg9-BK, Lys[Leu8]Des-Arg9-Bradykinin,... |
| Anwendung: | Bradykinin B1 receptor antagonist |
| MW: | 998.2 D |
ab 111,00 €
SSR 240612
Artikelnummer: Cay25544-1
SSR 240612 is a selective, non-peptide antagonist of the bradykinin B1 receptor (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors, respectively). It inhibits the contraction of rabbit aorta and rat ileum induced by the B1 receptor agonist des-Arg9-bradykinin (des-Arg9-BK) ex vivo in a concentration-dependent...
| Schlagworte: | (3R)-3-(1,3-benzodioxol-5-yl)-N-[(6-methoxy-2-naphthalenyl)sulfonyl]-beta-alanyl-4-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]me... |
| Anwendung: | Bradykinin B1 receptor antagonist |
| CAS | 464930-42-5 |
| MW: | 793.4 D |
ab 158,00 €
SCH79797 dihydrochloride
Artikelnummer: TGM-T12870-100mg
Description: SCH79797 dihydrochloride is an effective and selective antagonist of protease activated receptor 1 (PAR1) with an IC50 of 70 nM and a Ki of 35 nM. SCH79797 dihydrochloride has antiproliferative and pro-apoptotic effects. Target: Protease-activated Receptor, Apoptosis, Others. Smiles:...
| Anwendung: | PAR1 antagonist |
| CAS | 1216720-69-2 |
| MW: | 444.4 D |
ab 31,00 €
Bradykinin (acetate)
Artikelnummer: TGM-T21610-100mg
Description: Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system. It is a inflammatory mediator and also recognized as a neuromediator and regulator of several vascular and renal functions. Enzymatically produced from kallidin in the blood, it is a powerful vasodilator that...
| Anwendung: | peptide hormone |
| CAS | 6846-03-3 |
| MW: | 1120.26 D |
ab 36,00 €
SSR240612
Artikelnummer: TGM-T5048-100mg
Description: SSR240612 is a potent, orally active, specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 nM for B1 receptors and 358-481 nM for B2 receptors, respectively). Target: Bradykinin Receptor. Smiles:...
| Anwendung: | Bradykinin B1 receptor antagonist |
| CAS | 464930-42-5 |
| MW: | 793.41 D |
ab 233,00 €
R 715 (trifluoroacetate salt)
Artikelnummer: Cay36890-1
R 715 is a bradykinin B1 receptor antagonist. It inhibits contractions induced by bradykinin (Cay-37408) in isolated human umbilical cords, which express bradykinin B1 receptors (pA2 = 8.49). R 715 (200, 400, and 600 µg/kg) decreases the latency to tail withdrawal in the tail-flick test in a mouse model of diabetic...
| Schlagworte: | [Ac-Lys-[D-betaNal7,Ile8]des-Arg9]-BK, Ac-Lys-Arg-Pro-Pro-Gly-Phe-Ser-D2Nal-Ile-OH,... |
| Anwendung: | Bradykinin B1 receptor antagonist |
| MW: | 1140.3 D |
ab 310,00 €