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TBCA
TBCA

Artikelnummer: TGM-T21915-10mg

Description: TBCA (Casein Kinase II Inhibitor III, TBCA) is a highly selective CK2 (casein kinase II) inhibitor, IC50 = 110 nM, Ki = 77 nM. TBCA shows selectivity for CK2 over CK1, DYRK1A and a panel of 27 other kinases. Target: Casein Kinase. Smiles: OC(=O)\C=C\c1cc(Br)c(Br)c(Br)c1Br. References: Pagano MA, et al....
Schlagworte: Casein Kinase II Inhibitor III, TBCA
CAS 934358-00-6
MW: 463.74 D
ab 37,00 €
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TBCA
TBCA

Artikelnummer: Cay14831-1

Casein kinase 2 (CK2) is a kinase with many targets and diverse roles in cell signaling and disease. TBCA is a selective, cell-permeable inhibitor of CK2 (IC50 = 0.11 µM, Ki = 77 nM) that has minimal effect on a panel of 28 other kinases. It induces cell death in Jurkat adult T cell leukemia cells (DC50 = 7.7 µM),...
Schlagworte: Casein Kinase II Inhibitor III, Tetrabromocinnamic Acid, (2E)-3-(2,3,4,5-tetrabromophenyl)-2-propenoic acid
Anwendung: Selective, cell-permeable Casein kinase 2 (CK2) inhibitor
CAS 934358-00-6
MW: 463.7 D
ab 58,00 €
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