Zu "875258-85-8" wurden 2 Artikel gefunden!
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YIL 781
Artikelnummer: Cay45211-10
An antagonist of GHS-Ra (Ki = 0.017 µM), is selective for GHS-Ra over the motilin receptor (Ki = 6 µM) and a panel of 30 receptors and enzymes (Kis = > 10 µM), prevents ghrelin-induced decreases in insulin secretion in glucose-stimulated isolated rat pancreatic islets at concentration of 1 µM, increases plasma...
| Schlagworte: | (S)-6-(4-fluorophenoxy)-3-((1-isopropylpiperidin-3-yl)methyl)-2-methylquinazolin-4(3H)-one |
| Anwendung: | GHS-R1alpha antagonist |
| CAS | 875258-85-8 |
| MW: | 409.51 D |
ab 151,00 €
YIL 781
Artikelnummer: TGM-T23543-100mg
Description: YIL 781 is a selective ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM), showing a weak affinity for kinesin receptors (K = 6 µM). YIL 781 improves glucose homeostasis in vivo and in vitro by blocking ghrelin secretion. Target: GHSR. Smiles:...
| CAS | 875258-85-8 |
| MW: | 409.5 D |
ab 42,00 €
