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QLT0267
QLT0267

Artikelnummer: Cay34309-10

QLT0267 is an inhibitor of integrin-linked kinase (ILK, IC50 = 26 nM). It is greater than 10-fold selective for ILK over cyclin-dependent kinase 1 (Cdk1), Cdk2, and Cdk5, as well as greater than 1,000-fold selective for ILK over C-terminal Src kinase (CSK), DNA-PK, Pim-1, Akt, PKC, and casein kinase 2 (CK2), at 10...
Schlagworte: 4-((4-methoxyphenyl)diazenyl)-1H-pyrazole-3,5-diamine
Anwendung: ILK inhibitor
CAS 866409-68-9
MW: 232.2 D
ab 247,00 €
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QLT0267
QLT0267

Artikelnummer: TGM-T84998-10mg

Description: QLT0267 is an inhibitor targeting integrin-linked kinase (ILK, IC50= 26 nM), showing over 10-fold selectivity against cyclin-dependent kinases 1, 2, and 5 (Cdk1, Cdk2, and Cdk5), and over 1,000-fold selectivity against C-terminal Src kinase (CSK), DNA-PK, Pim-1, Akt, PKC, and casein kinase 2 (CK2) at a...
Anwendung: ILK inhibitor
CAS 866409-68-9
MW: 232.24 D
ab 241,00 €
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