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Takeda103A
Artikelnummer: TGM-T24850-100mg
Description: Takeda103A (CMPD103A) is the GRK2-dependent bovine tubulin oxidation effective inhibitor. Target: GRK. Smiles: CCCn1c(CNc2cccc(c2)C(=O)NCc2c(F)cccc2F)nnc1-c1ccncn1. References: Waldschmidt HV, Homan KT, Cruz-Rodríguez O, et al. Structure-Based Design, Synthesis, and Biological Evaluation of Highly...
| Schlagworte: | CMPD103A, Takeda 103 A, CMPD-103A, Takeda-103-A, Takeda-103A |
| Anwendung: | GRK2 inhibitor |
| CAS | 865609-72-9 |
| MW: | 463.48 D |
ab 77,00 €
Takeda-103A
Artikelnummer: Cay41027-1
Takeda-103A is an inhibitor of G protein-coupled receptor kinase 2 (GRK2). It selectively inhibits phosphorylation of bovine rod outer segments by GRK2 (IC50 = 54 nM) over phosphorylation by GRK1 and GRK5 at concentrations up to 125 µM. Takeda-103A also inhibits phosphorylation of bovine rod outer segments by GRK2...
| Schlagworte: | N-[(2,6-difluorophenyl)methyl]-3-[[[4-propyl-5-(4-pyrimidinyl)-4H-1,2,4-triazol-3-yl]methyl]amino]-benzamide |
| Anwendung: | GRK2 inhibitor |
| CAS | 865609-72-9 |
| MW: | 463.5 D |
ab 108,00 €
