Zu "83846-83-7" wurden 3 Artikel gefunden!
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Ketanserin (tartrate)
Artikelnummer: Cay22058-100
Ketanserin is a potent antagonist of the serotonin (5-HT) receptor that is selective for 5-HT2 (IC50 = 6.3 nM, Ki = 2.1 nM). It has no activity at 5-HT1 receptors but does have activity at histamine type 1, alpha1-adrenergic, and dopamine receptors with Ki values of 10, 10, and 220 nM, respectively. Ketanserin...
| Schlagworte: | 3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]-2,4(1H,3H)-quinazolinedione (2R,3R)-2,3-dihydroxybutanedioate |
| Anwendung: | HTR2A antagonist |
| CAS | 83846-83-7 |
| MW: | 545.5 D |
ab 109,00 €
(+)-Ketanserin tartrate salt
Artikelnummer: LKT-K1679.10
Ketanserin is an inhibitor of 5-HT2A receptors that exhibits antihypertensive, vasodilatory, analgesic, and pro-angiogenic activities. In animal models of hypertension, ketanserin decreases blood pressure and improves baroreceptor sensitivity and vagal tonic activity, improving left ventricular remodeling and...
| Anwendung: | 5-HT2A-receptor antagonist, Alpha1-adrenergic receptor antagonist, H1-receptor antagonist |
| CAS | 83846-83-7 |
| MW: | 545.52 D |
ab 60,00 €
Ketanserin . tartrate
Artikelnummer: AG-CR1-0014-M010
Selective 5-HT2A serotonin receptor antagonist, ATP-sensitive potassium channel inhibitor, hERG potassium channel blocker.
| Schlagworte: | 3-[2-[4-(4-Fluorobenzoyl)-1-piperdinyl)ethyl]-2,4(1H,3H)-quinazolinedione tartrate |
| Anwendung: | Potassium channel inhibitor, 5-HT2A serotonin receptor antagonist |
| CAS | 83846-83-7 |
| MW: | 395,4 D |
ab 33,00 €
