Zu "79183-37-2" wurden 2 Artikel gefunden!
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VU0119498
Artikelnummer: TGM-T8224-100mg
Description: VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 µM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent. Target: AChR. Smiles: Brc1ccc(CN2C(=O)C(=O)c3ccccc23)cc1. References: Lu Zhu , Mario Rossi,et al.Allosteric Modulation of beta-Cell M 3 Muscarinic...
| Anwendung: | Muscarinic acetylcholine receptor M1 / M3 / M5 positive allosteric modulator |
| CAS | 79183-37-2 |
| MW: | 316.15 D |
ab 31,00 €
VU0119498
Artikelnummer: Cay36132-100
VU0119498 is a positive allosteric modulator (PAM) of M1, M3, and M5 muscarinic acetylcholine receptors (mAChRs, EC50s = 6.04, 6.38, and 4.08 µM, respectively, in calcium mobilization assays). It is selective for M1, M3, and M5 mAChRs over M2 and M4 mAChRs in CHO cells expressing the human receptors. VU0119498 (20...
| Schlagworte: | 1-[(4-bromophenyl)methyl]-1H-indole-2,3-dione |
| Anwendung: | Muscarinic acetylcholine receptor M1 / M3 / M5 positive allosteric modulator |
| CAS | 79183-37-2 |
| MW: | 316.2 D |
ab 78,00 €
