Zu "768404-03-1" wurden 2 Artikel gefunden!
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5-BDBD
Artikelnummer: TGM-T22518-100mg
Description: 5-BDBD is a potent and selective P2X4 receptor antagonist. 5-BDBD inhibits rP2X4R-mediated currents with an IC50 of 0.75 µM. 5-BDBD completely blocked the basal and acute hyperalgesia induced by NTG. Target: P2X Receptor. Smiles: Brc1cccc(c1)C1=NCC(=O)Nc2c1oc1ccccc21. References: Coddou C, et al....
| CAS | 768404-03-1 |
| MW: | 355.19 D |
ab 35,00 €
5-BDBD
Artikelnummer: Cay42034-1
A P2X4 receptor antagonist (IC50 = 0.75 µM), selective for P2X4 over P2X1, P2X2a, P2X2b, and P2X7 but does inhibit P2X3 by 35.9% at 10 µM, decreases fEPSP slopes in rat hippocampal slices at 10 µM, inhibits nitroglycerin-induced mechanical hyperalgesia in a mouse model of chronic migraine at 28 mg/kg, decreases...
| Schlagworte: | 5-(3-bromophenyl)-1,3-dihydro-2H-benzofuro[3,2-e]-1,4-diazepin-2-one |
| Anwendung: | P2X4 receptor antagonist |
| CAS | 768404-03-1 |
| MW: | 355.2 D |
ab 38,00 €
