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Astemizole
Artikelnummer: Cay16967-25
Astemizole is a non-sedating antihistamine that antagonizes the histamine H1 receptor with a Ki value of 4.4 nM. It is considerably less potent at muscarinic acetylcholine receptors (Ki = 2.4 µM). Astemizole is also a potent blocker of ether-a-go-go-related gene (ERG) potassium channels (IC50 = ~1 nM) that has been...
| Schlagworte: | NSC 329963, 1-[(4-fluorophenyl)methyl]-N-[1-[2-(4-methoxyphenyl)ethyl]-4-piperidinyl]-1H-benzimidazol-2-amine |
| Anwendung: | Histamine H1 receptor antagonist |
| CAS | 68844-77-9 |
| MW: | 458.6 D |
ab 73,00 €
Astemizole
Artikelnummer: TGM-T1278-10mg
Description: Astemizole (Laridal) is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 receptors, with less anticholinergic effects compared to related agents. It is a long-acting, non-sedative antihistaminic used in the treatment...
| Schlagworte: | Histaminos, Paralergin, Laridal |
| Anwendung: | Targets histamine receptor H1 (HRH1) |
| CAS | 68844-77-9 |
| MW: | 458.57 D |
ab 40,00 €
