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Pergolide (mesylate)
Pergolide (mesylate)

Artikelnummer: Cay26085-25

Pergolide is a potent dopamine D1 and D2 receptor agonist (Kis = 111 and 0.495 nM, respectively, for rat striatal receptors). It depresses dopaminergic firing in paralyzed rats (ED50 = 2-selective antagonist spiperone or the dopamine D1-selective antagonist SCH 23390 (Cay-15631). Pergolide (0.025 and 0.05 mg/kg)...
Schlagworte: LY127809, NSC 319773, 8beta-[(methylthio)methyl]-6-propyl-ergoline, monomethanesulfonate
Anwendung: Dopamine D1-receptor agonist, dopamine D2-receptor agonist
CAS 66104-23-2
MW: 410.6 D
ab 73,00 €
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Pergolide mesylate
Pergolide mesylate

Artikelnummer: TGM-T2226-10mg

Description: Pergolide mesylate salt(LY127809) is a long-acting dopamine agonist which has been used to treat PARKINSON DISEASE and HYPERPROLA CTINEMIA but withdrawn from some markets due to potential for HEART VALVE DISEASES. Target: 5-HT Receptor, Adrenergic Receptor, Dopamine Receptor. Smiles:...
Schlagworte: Pergolide mesylate salt, LY127809, Pergolide methanesulfonate
Anwendung: Targets dopamine receptor D1 (DRD1)
CAS 66104-23-2
MW: 410.59 D
ab 45,00 €
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