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Capadenoson
Capadenoson

Artikelnummer: Cay28422-1

Capadenoson is an orally bioavailable, non-nucleoside adenosine (A) receptor partial agonist. It binds selectively to human A1 and A2B (EC50s = 0.66 and 1.1 nM, respectively) over A2A and A3 receptors (EC50s = 1,413 and 240 nM, respectively) expressed in CHO cells. Capadenoson (0.6 µM) decreases electrical...
Schlagworte: BAY 68-4986,...
Anwendung: Adenosine (A) receptor partial agonist
CAS 544417-40-5
MW: 520 D
ab 76,00 €
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Capadenoson
Capadenoson

Artikelnummer: TGM-TQ0125-10mg

Description: Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist. Target: Adenosine Receptor. Smiles: Nc1nc(SCc2csc(n2)-c2ccc(Cl)cc2)c(C#N)c(-c2ccc(OCCO)cc2)c1C#N. References: Bott-Flügel L, et al. Selective attenuation of norepinephrine release and stress-induced heart rate increase by partial...
Schlagworte: BAY 68-4986
Anwendung: Adenosine (A) receptor partial agonist
CAS 544417-40-5
MW: 520.03 D
ab 29,00 €
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