Zu "53882-12-5" wurden 2 Artikel gefunden!
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Lodoxamide
Artikelnummer: TGM-T4566-100mg
Description: Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis. Target: Histamine Receptor, GPR. Smiles: OC(=O)C(=O)Nc1cc(cc(NC(=O)C(O)=O)c1Cl)C#N. References: Watt GD, et al. Protective effect opf lodoxamide...
| Schlagworte: | Lodoxamidum |
| Anwendung: | Antiallergic, Antiasthmatic |
| CAS | 53882-12-5 |
| MW: | 311.63 D |
ab 40,00 €
Lodoxamide
Artikelnummer: Cay23994-25
Lodoxamide is a potent agonist of GPR35 with an EC50 value of 1.61 nM in a beta-arrestin-2 interaction assay using CHO-K1 cells expressing the human receptor. It inhibits histamine release induced by compound 48/80 (Cay-22173), anti-IgE, or A23187 (Cay-11016) in isolated rat peritoneal mast cells (IC50s = 0.1-50 µM)...
| Schlagworte: | 2,2'-[(2-chloro-5-cyano-1,3-phenylene)diimino]bis[2-oxo-acetic acid] |
| Anwendung: | GPR35 agonist |
| CAS | 53882-12-5 |
| MW: | 311.6 D |
ab 133,00 €
