Zu "510733-97-8" wurden 2 Artikel gefunden!
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ATC 0175
Artikelnummer: Cay42376-10
An MC1R antagonist (IC50 = 7.23 nM), selective for MC1R over MC2R (IC50 = >10,000 nM) but does antagonize 5-HT2B and 5-HT1A receptors (IC50s = 9.66 and 16.9 nM, respectively), inhibits MCH-induced [35S]GTPgammaS binding and calcium influx in HEK293 cells expressing human MC1R at 3 nM, reduces stress-induced...
| Schlagworte: | N-[cis-4-[[4-(dimethylamino)-2-quinazolinyl]amino]cyclohexyl]-3,4-difluoro-benzamide, monohydrochloride |
| Anwendung: | MC1R antagonist |
| CAS | 510733-97-8 |
| MW: | 461.94 D |
ab 102,00 €
ATC 0175 hydrochloride
Artikelnummer: TGM-T22591-100mg
Description: ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective. ATC 0175 hydrochloride has affinity for MCH1R, MCH2R, MCH1, 5-HT2B receptors and 5-HT1A receptors with IC50s of 13.5 nM, >10,000 nM, 13 nM, 9.66 nM and 16.9 nM, respectively....
| CAS | 510733-97-8 |
| MW: | 461.93 D |
ab 68,00 €
