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Hesperadin
Hesperadin

Artikelnummer: TGM-T6532-10mg

Description: Hesperadin(IC50=250 nM) effectively inhibits Aurora B. It potently reduces the activity of AMPK, MAPKAP-K1, MKK1, Lck, CHK1 and PHK, but it could not inhibit MKK1 activity in vivo. Target: Parasite, Aurora Kinase, Autophagy, Influenza Virus. Smiles:...
Anwendung: Multi-kinase inhibitor
CAS 422513-13-1
MW: 516.65 D
ab 34,00 €
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Hesperadin
Hesperadin

Artikelnummer: Cay24199-1

Hesperadin is a multi-kinase inhibitor. It inhibits human Aurora kinase B (IC50 = 250 nM) and its T. brucei homolog Aurora kinase-1 (IC50 = 40 nM) in in vitro kinase assays. Hesperadin (1 µM) inhibits AMPK, LCK, MKK1, MAPKAP-K1, CHK1, and PHK in a panel of 25 kinases. It also inhibits MEKK2 in ATPase and...
Schlagworte: N-[2,3-dihydro-2-oxo-3-[(3Z)-phenyl[[4-(1-piperidinylmethyl)phenyl]amino]methylene]-1H-indol-5-yl]-ethanesulfonamide
Anwendung: Multi-kinase inhibitor
CAS 422513-13-1
MW: 516.7 D
ab 67,00 €
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