Zu "3562-84-3" wurden 2 Artikel gefunden!
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Benzbromarone
Artikelnummer: Cay19768-500
Benzbromarone is an inhibitor of the urate anion transporter (IC50 = 0.3 µM for hURAT1) that prevents renal urate resorption. It also potently inhibits CYP2C9 (Ki = 20 nM), a major cytochrome P450 enzyme involved in the metabolic clearance of a wide range of therapeutic agents. Several analogs of benzabromarone have...
| Schlagworte: | MJ10061, NSC 85433, (3,5-dibromo-4-hydroxyphenyl)(2-ethyl-3-benzofuranyl)-methanone |
| Anwendung: | Urate anion transporter inhibitor, CYP2C9 inhibitor |
| CAS | 3562-84-3 |
| MW: | 424.1 D |
ab 49,00 €
Benzbromarone
Artikelnummer: TGM-T1274-100mg
Description: Benzbromarone (Desuric) is a CYP2C9 inhibitor with Ki value of 19.3 nM. Target: Xanthine Oxidase, Apoptosis, P450. Smiles: C(=O)(C=1C=2C(OC1CC)=CC=CC2)C3=CC(Br)=C(O)C(Br)=C3. References: Locuson CW 2nd, et al. Drug Metab Dispos, 2003, 31(7), 967-971.
| Schlagworte: | Desuric, Normurat, Urinorm |
| Anwendung: | Targets SLC22A12 (URAT1) |
| CAS | 3562-84-3 |
| MW: | 424.08 D |
ab 32,00 €
